Evidence mapPaperPMID 25475828Full record

ArticleDiabetes, obesity & metabolism2015

Liraglutide, leptin and their combined effects on feeding: additive intake reduction through common intracellular signalling mechanisms.

S E Kanoski, Z Y Ong, S M Fortin, E S Schlessinger, H J Grill

Open access · greenAbstract read
In one paragraph

Article in Diabetes, obesity & metabolism, 2015. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 17 papers.

0numbers the graph read from it
0cells of the map it votes in
17citing papers in PubMed
1.3field-weighted citation impact, top 22% of its field
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

17 citing papers in PubMed, 39 citations in OpenAlex.

  1. Article
  2. Article
  3. Article
  4. Review
  5. Review
  6. Article
  7. Review
  8. Article
  9. Incendiary Leptin.Nutrients · 2020
    Review
  10. Glucagon-like peptide 1 (GLP-1).Molecular metabolism · 2019 · on this map
    Review
  11. Article
  12. Review
  13. Endogenous Glucagon-like Peptide-1 Receptor Signaling in the Nucleus Tractus Solitarius is Required for Food Intake Control.Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology · 2017
    Article
  14. Article
  15. GLP-1 and weight loss: unraveling the diverse neural circuitry.American journal of physiology. Regulatory, integrative and comparative physiology · 2016
    Review
  16. Leptin applications in 2015: what have we learned about leptin and obesity?Current opinion in endocrinology, diabetes, and obesity · 2015
    Review
  17. Liraglutide and obesity: a review of the data so far.Drug design, development and therapy · 2015
    Review
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

5 authors at 3 institutions in 1 country.

S E KanoskiDepartment of Biological Sciences, University of Southern California, Los Angeles, CA, USA.
Z Y Ong
S M Fortin
E S Schlessinger
H J Grill
University of Pennsylvania · USUniversity of Illinois Chicago · USUniversity of Southern California · US

Funding

NEURAL HIERARCHY IN THE MODULATION OF INGESTIVE BEHAVIORR01DK021397 · UNIVERSITY OF PENNSYLVANIA · 1986 to 2005
$2.7M
NIDDK NIH HHS DK097147NIDDK NIH HHS DK102478NIDDK NIH HHS DK21397NIDDK NIH HHS K01 DK097147NIDDK NIH HHS R01 DK021397NIDDK NIH HHS R03 DK102478NIDDK NIH HHS R56 DK021397
6 · The paper itself

Abstract

aimTo investigate the behavioural and intracellular mechanisms by which the glucagon like peptide-1 (GLP-1) receptor agonist, liraglutide, and leptin in combination enhance the food intake inhibitory and weight loss effects of either treatment alone.

methodsWe examined the effects of liraglutide (a long-acting GLP-1 analogue) and leptin co-treatment, delivered in low or moderate doses subcutaneously (s.c.) or to the third ventricle, respectively, on cumulative intake, meal patterns and hypothalamic expression of intracellular signalling proteins [phosphorylated signal transducer and activator of transcription-3 (pSTAT3) and protein tyrosine phosphatase-1B (PTP1B)] in lean rats.

resultsA low-dose combination of liraglutide (25 µg/kg) and leptin (0.75 µg) additively reduced cumulative food intake and body weight, a result mediated predominantly through a significant reduction in meal frequency that was not present with either drug alone. Liraglutide treatment alone also reduced meal size; an effect not enhanced with leptin co-administration. Moderate doses of liraglutide (75 µg/kg) and leptin (4 µg), examined separately, each reduced meal frequency, cumulative food intake and body weight; only liraglutide reduced meal size. In combination these doses did not further enhance the anorexigenic effects of either treatment alone. Ex vivo immunoblot analysis showed elevated pSTAT3 in the hypothalamic tissue after liraglutide-leptin co-treatment, an effect which was greater than that of leptin treatment alone. In addition, s.c. liraglutide reduced the expression of PTP1B (a negative regulator of leptin receptor signalling), revealing a potential mechanism for the enhanced pSTAT3 response after liraglutide-leptin co-administration.

conclusionsCollectively, these results show novel behavioural and molecular mechanisms underlying the additive reduction in food intake and body weight after liraglutide-leptin combination treatment.

Indexed as

Weight LossAnimalsAppetite DepressantsBody WeightDrug Therapy, CombinationEatingGlucagon-Like Peptide 1HypothalamusIncretinsLeptinLiraglutideMaleObesityProtein Tyrosine Phosphatase, Non-Receptor Type 1RatsRats, Sprague-DawleyAppetite DepressantsGlucagon-Like Peptide 1IncretinsLeptinLiraglutideProtein Tyrosine Phosphatase, Non-Receptor Type 1STAT3 Transcription Factorexendin-4GLP-1obesityratsynergyweight loss

Identifiers

PMID25475828
PMCPMC4320650
OpenAlexW2146727082

What Socratic holds

Texttitle and abstract
LicenceTDM
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.