Evidence map›Paper›PMID 30862686›Full record

ArticleMolecular cancer research : MCR2019

Metabolic Detection of Bruton's Tyrosine Kinase Inhibition in Mantle Cell Lymphoma Cells.

Seung-Cheol Lee, Alexander A Shestov, Lili Guo, Qian Zhang, Jeffrey C Roman, Xiaobin Liu, Hong Y Wang, Stephen Pickup, Kavindra Nath, Pin Lu and 8 more

Open access · bronzeAbstract read
In one paragraph

Article in Molecular cancer research : MCR, 2019. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 14 papers.

0numbers the graph read from it
0cells of the map it votes in
14citing papers in PubMed
1.6field-weighted citation impact, top 17% of its field
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

14 citing papers in PubMed, 22 citations in OpenAlex.

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  12. Liquid Chromatography-Mass Spectrometry for Clinical Metabolomics: An Overview.Advances in experimental medicine and biology · 2021
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4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

18 authors at 3 institutions in 1 country.

Seung-Cheol Lee *Department of Radiology, University of Pennsylvania, Philadelphia, Pennsylvania. wasik@pennmedicine.upenn.edu seungch@pennmedicine.upenn.edu glickson@pennmedicine.upenn.edu.
Alexander A Shestov *Department of Radiology, University of Pennsylvania, Philadelphia, Pennsylvania.
Lili GuoDepartment of Systems Pharmacology and Translational Therapeutics, University of Pennsylvania, Philadelphia, Pennsylvania.
Qian ZhangDepartment of Pathology and Laboratory Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.
Jeffrey C RomanDepartment of Radiology, University of Pennsylvania, Philadelphia, Pennsylvania.
Xiaobin LiuDepartment of Pathology and Laboratory Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.
Hong Y WangDepartment of Pathology and Laboratory Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.ORCID 0000-0003-0773-1212
Stephen PickupDepartment of Radiology, University of Pennsylvania, Philadelphia, Pennsylvania.
Kavindra NathDepartment of Radiology, University of Pennsylvania, Philadelphia, Pennsylvania.
Pin LuDepartment of Pathology, University of Chicago, Chicago, Illinois.
Samuel HofbauerDepartment of Systems Pharmacology and Translational Therapeutics, University of Pennsylvania, Philadelphia, Pennsylvania.
Clementina MesarosDepartment of Systems Pharmacology and Translational Therapeutics, University of Pennsylvania, Philadelphia, Pennsylvania.
Y Lynn WangDepartment of Pathology, University of Chicago, Chicago, Illinois.ORCID 0000-0003-0773-1212
David S NelsonDepartment of Radiology, University of Pennsylvania, Philadelphia, Pennsylvania.
Stephen J SchusterDepartment of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania.
Ian A BlairDepartment of Systems Pharmacology and Translational Therapeutics, University of Pennsylvania, Philadelphia, Pennsylvania.
Jerry D GlicksonDepartment of Radiology, University of Pennsylvania, Philadelphia, Pennsylvania. wasik@pennmedicine.upenn.edu seungch@pennmedicine.upenn.edu glickson@pennmedicine.upenn.edu.
Mariusz A WasikDepartment of Pathology and Laboratory Medicine, University of Pennsylvania, Philadelphia, Pennsylvania. wasik@pennmedicine.upenn.edu seungch@pennmedicine.upenn.edu glickson@pennmedicine.upenn.edu.
University of Pennsylvania · USTranslational Therapeutics (United States) · USUniversity of Illinois Chicago · US

Funding

Systemic Chemotherapy of Melanoma: NMR Studies of Lonidamine & N-Mustard ActivityR01CA129544 · NCI · UNIVERSITY OF PENNSYLVANIA · PI GLICKSON, JERRY D · 2009 to 2016
$3.2M
Mechanism of Activity of LonidamineR01CA172820 · NCI · UNIVERSITY OF PENNSYLVANIA · PI GLICKSON, JERRY D · 2013 to 2017
$2.8M
NCI NIH HHS R01 CA129544NCI NIH HHS R01 CA172820
6 · The paper itself

Abstract

Current methods to evaluate effects of kinase inhibitors in cancer are suboptimal. Analysis of changes in cancer metabolism in response to the inhibitors creates an opportunity for better understanding of the interplay between cell signaling and metabolism and, from the translational perspective, potential early evaluation of response to the inhibitors as well as treatment optimization. We performed genomic, metabolomic, and fluxomic analyses to evaluate the mechanism of action of the Bruton's tyrosine kinase (BTK) inhibitor ibrutinib (IBR) in mantle cell lymphoma (MCL) cells. Our comprehensive analysis of the data generated by these diverse technologies revealed that IBR profoundly affected key metabolic pathways in IBR-sensitive cells including glycolysis, pentose phosphate pathway, TCA cycle, and glutaminolysis while having much less effects on IBR-poorly responsive cells. Changes in

Indexed as

AdenineAgammaglobulinaemia Tyrosine KinaseBenzeneacetamidesBiomarkers, TumorCell Line, TumorGlutaminaseHumansLymphoma, Mantle-CellMetabolic Networks and PathwaysPiperidinesProtein Kinase InhibitorsProtein-Tyrosine KinasesPyrazolesPyrimidinesSignal TransductionThiadiazolesAdenineAgammaglobulinaemia Tyrosine KinaseBenzeneacetamidesBiomarkers, TumorCB-839GlutaminaseibrutinibPiperidinesProtein Kinase InhibitorsProtein-Tyrosine KinasesPyrazolesPyrimidinesThiadiazoles

Identifiers

PMID30862686
PMCPMC8757533
OpenAlexW2921347480

What Socratic holds

Textmetadata
LicenceTDM
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.