Evidence mapPaperPMID 33236485Full record

ArticleDiabetes, obesity & metabolism2021

Weight-loss response to naltrexone/bupropion is modulated by the Taq1A genetic variant near DRD2 (rs1800497): A pilot study.

Jamie A Mullally, Wendy K Chung, Charles A LeDuc, Tirissa J Reid, Gerardo Febres, Steven Holleran, Rajasekhar Ramakrishnan, Judith Korner

Open access · greenAbstract read
In one paragraph

Article in Diabetes, obesity & metabolism, 2021. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 10 papers, 1 of them a synthesis that pooled it.

0numbers the graph read from it
0cells of the map it votes in
10citing papers in PubMed, 1 pooled it
1.5field-weighted citation impact, top 17% of its field
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

10 citing papers in PubMed, 1 synthesis or guideline pooled it, 11 citations in OpenAlex.

  1. Pooled it
  2. Review
  3. Article
  4. Review
  5. Review
  6. Weight Loss Interventions for Adults With Obesity-Related Asthma.The journal of allergy and clinical immunology. In practice · 2024
    Article
  7. Article
  8. Anti-Inflammatory Effects of Peripheral Dopamine.International journal of molecular sciences · 2023
    Review
  9. Article
  10. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

8 authors at 2 institutions in 1 country.

Jamie A MullallyWestchester Medical Center, Valhalla, New York.ORCID 0000-0002-6633-0884
Wendy K ChungColumbia University Irving Medical Center, New York, New York.
Charles A LeDucColumbia University Irving Medical Center, New York, New York.
Tirissa J ReidColumbia University Irving Medical Center, New York, New York.
Gerardo FebresColumbia University Irving Medical Center, New York, New York.
Steven HolleranColumbia University Irving Medical Center, New York, New York.
Rajasekhar RamakrishnanColumbia University Irving Medical Center, New York, New York.
Judith KornerColumbia University Irving Medical Center, New York, New York.
Columbia University Irving Medical Center · USWestchester Medical Center · US

Funding

Clinical and Translational Science AwardUL1TR001873 · COLUMBIA UNIVERSITY HEALTH SCIENCES · 2025 to 2025
$10.0M
RESEARCH TRAININGP30DK026687 · ST. LUKE'S-ROOSEVELT INST FOR HLTH SCIS · 1986 to 2025
$7.5M
MOLECULAR GENETIC ANALYSIS OF HUMAN OBESITYR01DK052431 · ROCKEFELLER UNIVERSITY · 1996 to 2005
$3.6M
MECHANISMS OF BETA CELL FAILURER01DK064819 · COLUMBIA UNIVERSITY HEALTH SCIENCES · 2003 to 2025
$1.8M
TRAINING PROGRAM IN ENDOCRINOLOGY AND METABOLISMT32DK007271 · COLUMBIA UNIV NEW YORK MORNINGSIDE · 1986 to 2005
$1.7M
NCATS NIH HHS UL1 TR001873NIDDK NIH HHS P30 DK026687NIDDK NIH HHS R01 DK052431NIDDK NIH HHS R01 DK064819NIDDK NIH HHS T32 DK007271
6 · The paper itself

Abstract

Naltrexone/bupropion (NB) is a US Food and Drug Administration-approved antiobesity medication. Clinical trials have shown variable weight loss, with responders and non-responders. NB is believed to act on central dopaminergic pathways to suppress appetite. The Taq1A polymorphism near DRD2 (rs1800497) is associated with the density of striatal dopamine D2 receptors, with individuals carrying the A allele (AA or AG; termed A1+) having 30%-40% fewer dopamine binding sites than those who do not carry the A allele (GG; termed A1-). We performed a pilot study to assess the association of the rs1800497 ANKK1 c.2137G > A (p.Glu713Lys) variant with weight loss with NB treatment in 33 subjects. Mean (SD) weight loss was 5.9% (3.2%) for the A1+ genotype group (n = 15) and 4.2% (4.2%) for the A1- genotype group (n = 18). The mean weight loss for the A1+ genotype group was significantly greater than the predefined clinically significant 4% weight-loss target (one-sample t-test, P = .035), whereas the mean weight loss for the A1- genotype group was not (P = .85). Individuals with the A1+ genotype appear to respond better to NB than A1- individuals.

Indexed as

BupropionNaltrexoneGenotypeHumansPilot ProjectsPolymorphism, Single NucleotideProtein Serine-Threonine KinasesReceptors, Dopamine D2Weight LossANKK1 protein, humanBupropionDRD2 protein, humanNaltrexoneProtein Serine-Threonine KinasesReceptors, Dopamine D2antiobesity drugdrug mechanismobesity therapypharmacogeneticsweight control

Identifiers

PMID33236485
PMCPMC8106923
OpenAlexW3108851982

What Socratic holds

Textmetadata
LicenceTDM
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.