Evidence mapPaperPMID 33477672Full record

ArticlePharmaceutics2021

Physicochemical Characterization of a Co-Amorphous Atorvastatin-Irbesartan System with a Potential Application in Fixed-Dose Combination Therapy.

Marcin Skotnicki, Barbara Jadach, Agnieszka Skotnicka, Bartłomiej Milanowski, Lidia Tajber, Marek Pyda, Jacek Kujawski

Abstract read
In one paragraph

Article in Pharmaceutics, 2021. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 6 papers.

0numbers the graph read from it
0cells of the map it votes in
6citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

6 citing papers in PubMed.

  1. Article
  2. Article
  3. Article
  4. Article
  5. Article
  6. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

7 authors.

Marcin SkotnickiChair and Department of Pharmaceutical Technology, Poznan University of Medical Sciences, 60-780 Poznan, Poland.ORCID 0000-0002-3325-4109
Barbara JadachChair and Department of Pharmaceutical Technology, Poznan University of Medical Sciences, 60-780 Poznan, Poland.ORCID 0000-0001-5222-4557
Agnieszka SkotnickaChair and Department of Pharmaceutical Technology, Poznan University of Medical Sciences, 60-780 Poznan, Poland.
Bartłomiej MilanowskiChair and Department of Pharmaceutical Technology, Poznan University of Medical Sciences, 60-780 Poznan, Poland.ORCID 0000-0002-6450-174X
Lidia TajberSchool of Pharmacy and Pharmaceutical Sciences, Trinity College Dublin, College Green, 2 Dublin, Ireland.ORCID 0000-0003-1544-6796
Marek PydaDepartment of Biophysics, Poznan University of Medical Sciences, 60-780 Poznan, Poland.
Jacek KujawskiChair and Department of Organic Chemistry, Poznan University of Medical Sciences, 60-780 Poznan, Poland.ORCID 0000-0001-6279-4887

Funding

European Union's Horizon 2020 research and innovation programme under the Marie Skłodowska-Curie 778051Ministry of Science and Higher Education of Poland fund for supporting internationally co-financed projects in 2018-2022 3899/H2020/2018/2Synthesis and Solid State Pharmaceutical Centre (SSPC), financed by a research grant from Science Foundation Ireland (SFI) and co-funded under the European Regional Development Fund 12/RC/2275Wrocław Center for Networking and Supercomputing 327/2014
6 · The paper itself

Abstract

The aim of this study was to characterize a 1:1 molar ratio of a pharmacologically relevant co-amorphous atorvastatin-irbesartan (ATR-IRB) system obtained by quench cooling of the crystalline ATR/IRB physical mixture for potential use in the fixed-dose combination therapy. The system was characterized by employing standard differential scanning calorimetry (DSC), Fourier transform-infrared spectroscopy (FT-IR), and intrinsic dissolution rate studies. Quantum mechanical calculations were performed to obtain information regarding intermolecular interactions in the studied co-amorphous ATR-IRB system. The co-amorphous formulation showed a significant improvement in the intrinsic dissolution rate (IDR) of IRB over pure crystalline as well as its amorphous counterpart. An unusual behavior was observed for ATR, as the IDR of ATR in the co-amorphous formulation was slightly lower than that of amorphous ATR alone. Short-term physical aging studies of up to 8 h proved that the ATR-IRB co-amorphous system remained in the amorphous form. Furthermore, no physical aging occurred in the co-amorphous system. FT-IR, density functional theory calculations, and analysis of

Indexed as

atorvastatinco-amorphous systemdensity functional theorydifferential scanning calorimetryintrinsic dissolution rateirbesartanphysical stability

Identifiers

PMID33477672
PMCPMC7831949

What Socratic holds

Textmetadata
LicenceCC BY
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.