Evidence map›Paper›PMID 34138563›Full record

ArticleJournal of medicinal chemistry2021

Asymmetric Synthesis and Biological Screening of Quinoxaline-Containing Synthetic Lipoxin A

Monica de Gaetano, Catherine Tighe, Kevin Gahan, Andrea Zanetti, Jianmin Chen, Justine Newson, Antonino Cacace, Mariam Marai, Andrew Gaffney, Eoin Brennan and 7 more

Open access · hybridAbstract read
In one paragraph

Article in Journal of medicinal chemistry, 2021. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 11 papers.

0numbers the graph read from it
0cells of the map it votes in
11citing papers in PubMed
1.8field-weighted citation impact, top 15% of its field
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

11 citing papers in PubMed, 30 citations in OpenAlex.

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4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

17 authors at 5 institutions in 4 countries.

Monica de GaetanoSchool of Medicine, Diabetes Complications Research Centre, UCD Conway Institute, University College Dublin, Belfield, Dublin D04 N2E5, Ireland.
Catherine TigheCentre for Synthesis and Chemical Biology, School of Chemistry, UCD Conway Institute, University College Dublin, Belfield, Dublin D04 N2E5, Ireland.
Kevin GahanCentre for Synthesis and Chemical Biology, School of Chemistry, UCD Conway Institute, University College Dublin, Belfield, Dublin D04 N2E5, Ireland.
Andrea ZanettiCentre for Synthesis and Chemical Biology, School of Chemistry, UCD Conway Institute, University College Dublin, Belfield, Dublin D04 N2E5, Ireland.
Jianmin ChenWilliam Harvey Research Institute, Queen Mary University London, London EC1M 6BQ, U.K.
Justine NewsonCentre for Clinical Pharmacology, University College London, London WC1E 6JF, U.K.
Antonino CacaceSchool of Medicine, Diabetes Complications Research Centre, UCD Conway Institute, University College Dublin, Belfield, Dublin D04 N2E5, Ireland.
Mariam MaraiSchool of Medicine, Diabetes Complications Research Centre, UCD Conway Institute, University College Dublin, Belfield, Dublin D04 N2E5, Ireland.
Andrew GaffneySchool of Medicine, Diabetes Complications Research Centre, UCD Conway Institute, University College Dublin, Belfield, Dublin D04 N2E5, Ireland.
Eoin BrennanSchool of Medicine, Diabetes Complications Research Centre, UCD Conway Institute, University College Dublin, Belfield, Dublin D04 N2E5, Ireland.
Phillip KantharidisDepartment of Diabetes, Central Clinical School, Monash University, Melbourne, VIC 3004, Australia.
Mark E CooperDepartment of Diabetes, Central Clinical School, Monash University, Melbourne, VIC 3004, Australia.
Xavier LeroyDomain Therapeutics SA, 67400 Strasbourg, Illkirch, France.
Mauro PerrettiWilliam Harvey Research Institute, Queen Mary University London, London EC1M 6BQ, U.K.
Derek GilroyCentre for Clinical Pharmacology, University College London, London WC1E 6JF, U.K.
Catherine GodsonSchool of Medicine, Diabetes Complications Research Centre, UCD Conway Institute, University College Dublin, Belfield, Dublin D04 N2E5, Ireland.
Patrick J GuiryCentre for Synthesis and Chemical Biology, School of Chemistry, UCD Conway Institute, University College Dublin, Belfield, Dublin D04 N2E5, Ireland.ORCID 0000-0002-2612-8569
University College Dublin · IEMonash University · AUUniversity College London · GBWilliam Harvey Research Institute · GBDomain Therapeutics (France) · FR

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Failure to resolve inflammation underlies many prevalent pathologies. Recent insights have identified lipid mediators, typified by lipoxins (LXs), as drivers of inflammation resolution, suggesting potential therapeutic benefit. We report the asymmetric preparation of novel quinoxaline-containing synthetic-LXA

Indexed as

AnimalsAnti-Inflammatory Agents, Non-SteroidalCells, CulturedCell SurvivalDose-Response Relationship, DrugDrug Evaluation, PreclinicalHumansInflammationLipopolysaccharidesMiceMolecular StructureMonocytesNF-kappa BQuinoxalinesReceptors, Formyl PeptideReceptors, LipoxinAnti-Inflammatory Agents, Non-SteroidalFPR2 protein, humanLipopolysaccharidesNF-kappa BQuinoxalinesReceptors, Formyl PeptideReceptors, LipoxinTNF protein, humanTumor Necrosis Factor-alpha

Identifiers

PMID34138563
PMCPMC8279484
OpenAlexW3172854200

What Socratic holds

Textmetadata
LicenceCC BY
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.