Evidence mapPaperPMID 35595952Full record

ArticleCommunications biology2022

A precision medicine approach to metabolic therapy for breast cancer in mice.

Ngozi D Akingbesote, Aaron Norman, Wanling Zhu, Alexandra A Halberstam, Xinyi Zhang, Julia Foldi, Maryam B Lustberg, Rachel J Perry

Open access · goldAbstract read
In one paragraph

Article in Communications biology, 2022. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 15 papers.

0numbers the graph read from it
0cells of the map it votes in
15citing papers in PubMed
1.8field-weighted citation impact, top 15% of its field
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

15 citing papers in PubMed, 23 citations in OpenAlex.

  1. Review
  2. Review
  3. Review
  4. Review
  5. Review
  6. Review
  7. Review
  8. Exploring SGLT2 Inhibitors' Activity in Breast Cancer: An Overview.Current topics in medicinal chemistry · 2025
    Review
  9. Obesity-Associated Colorectal Cancer.International journal of molecular sciences · 2024
    Review
  10. Thiazolidinedione enhances the efficacy of anti-PD-1 monoclonal antibody in murine melanoma.American journal of physiology. Endocrinology and metabolism · 2024
    Article
  11. Metabolic underpinnings of cancer-related fatigue.American journal of physiology. Endocrinology and metabolism · 2024
    Review
  12. Dichloroacetate as a novel pharmaceutical treatment for cancer-related fatigue in melanoma.American journal of physiology. Endocrinology and metabolism · 2023
    Article
  13. A review of the impact of energy balance on triple-negative breast cancer.Journal of the National Cancer Institute. Monographs · 2023
    Review
  14. Article
  15. Review
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

8 authors at 1 institution in 1 country.

Ngozi D AkingbesoteDepartment of Celullar and Molecular Physiology, Yale University School of Medicine, New Haven, CT, USA.
Aaron NormanDepartment of Celullar and Molecular Physiology, Yale University School of Medicine, New Haven, CT, USA.
Wanling ZhuDepartment of Celullar and Molecular Physiology, Yale University School of Medicine, New Haven, CT, USA.
Alexandra A HalberstamDepartment of Celullar and Molecular Physiology, Yale University School of Medicine, New Haven, CT, USA.ORCID http://orcid.org/0000-0001-5475-560X
Xinyi ZhangDepartment of Celullar and Molecular Physiology, Yale University School of Medicine, New Haven, CT, USA.ORCID http://orcid.org/0000-0002-3173-0589
Julia FoldiDepartment of Internal Medicine (Hematology/Oncology), Yale University School of Medicine, New Haven, CT, USA.ORCID http://orcid.org/0000-0002-7504-867X
Maryam B LustbergDepartment of Internal Medicine (Hematology/Oncology), Yale University School of Medicine, New Haven, CT, USA.
Rachel J PerryDepartment of Celullar and Molecular Physiology, Yale University School of Medicine, New Haven, CT, USA. rachel.perry@yale.edu.ORCID http://orcid.org/0000-0003-0748-8064
Yale University · US

Funding

Yale Diabetes Research CenterP30DK045735 · YALE UNIVERSITY · 1993 to 2025
$10.2M
INSTITUTIONAL NATIONAL RESEARCH SERVICE AWARDT32GM007324 · YALE UNIVERSITY · 1987 to 2005
$1.3M
NIDDK NIH HHS P30 DK045735NIGMS NIH HHS T32 GM007324
6 · The paper itself

Abstract

Increasing evidence highlights approaches targeting metabolism as potential adjuvants to cancer therapy. Sodium-glucose transport protein 2 (SGLT2) inhibitors are the newest class of antihyperglycemic drugs. To our knowledge, SGLT2 inhibitors have not been applied in the neoadjuvant setting as a precision medicine approach for this devastating disease. Here, we treat lean breast tumor-bearing mice with the SGLT2 inhibitor dapagliflozin as monotherapy and in combination with paclitaxel chemotherapy. We show that dapagliflozin enhances the efficacy of paclitaxel, reducing tumor glucose uptake and prolonging survival. Further, the ability of dapagliflozin to enhance the efficacy of chemotherapy correlates with its effect to reduce circulating insulin in some but not all breast tumors. Our data suggest a genetic signature for breast tumors more likely to respond to dapagliflozin in combination with paclitaxel. In the current study, tumors driven by mutations upstream of canonical insulin signaling pathways responded to this combined treatment, whereas tumors driven by mutations downstream of canonical insulin signaling did not. These data demonstrate that dapagliflozin enhances the response to chemotherapy in mice with breast cancer and suggest that patients with driver mutations upstream of canonical insulin signaling may be most likely to benefit from this neoadjuvant approach.

Indexed as

Breast NeoplasmsDiabetes Mellitus, Type 2Sodium-Glucose Transporter 2 InhibitorsAnimalsFemaleHumansInsulinMicePaclitaxelPrecision MedicineInsulinPaclitaxelSodium-Glucose Transporter 2 Inhibitors

Identifiers

PMID35595952
PMCPMC9122928
OpenAlexW4280588360

What Socratic holds

Textmetadata
LicenceCC BY
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.