Evidence map›Paper›PMID 36076974›Full record

ArticleInternational journal of molecular sciences2022

Intrarectal Capsazepine Administration Modulates Colonic Mucosal Health in Mice.

Vibhu Kumar, Vijay Kumar, Kirti Devi, Ajay Kumar, Rehan Khan, Ravindra Pal Singh, Sivasubramanian Rajarammohan, Kanthi Kiran Kondepudi, Kanwaljit Chopra, Mahendra Bishnoi

Open access · goldAbstract read
In one paragraph

Article in International journal of molecular sciences, 2022. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 6 papers, 1 of them a synthesis that pooled it.

0numbers the graph read from it
0cells of the map it votes in
6citing papers in PubMed, 1 pooled it
1.8field-weighted citation impact, top 15% of its field
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

6 citing papers in PubMed, 1 synthesis or guideline pooled it, 11 citations in OpenAlex.

  1. Pooled it
  2. Review
  3. Review
  4. Review
  5. Article
  6. Frontiers in nutrition · 2023
    Review
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

10 authors at 5 institutions in 3 countries.

Vibhu KumarTR(i)P for Health Laboratory, Centre for Excellence in Functional Foods, Department of Food and Nutritional Biotechnology, National Agri-Food Biotechnology Institute (NABI), Sector 81, Mohali 140306, India.
Vijay KumarTR(i)P for Health Laboratory, Centre for Excellence in Functional Foods, Department of Food and Nutritional Biotechnology, National Agri-Food Biotechnology Institute (NABI), Sector 81, Mohali 140306, India.
Kirti DeviTR(i)P for Health Laboratory, Centre for Excellence in Functional Foods, Department of Food and Nutritional Biotechnology, National Agri-Food Biotechnology Institute (NABI), Sector 81, Mohali 140306, India.
Ajay KumarInstitute of Nanoscience and Technology (INST), Sector 81, Mohali 140306, India.ORCID 0000-0001-7649-4578
Rehan KhanInstitute of Nanoscience and Technology (INST), Sector 81, Mohali 140306, India.
Ravindra Pal SinghTR(i)P for Health Laboratory, Centre for Excellence in Functional Foods, Department of Food and Nutritional Biotechnology, National Agri-Food Biotechnology Institute (NABI), Sector 81, Mohali 140306, India.
Sivasubramanian RajarammohanTR(i)P for Health Laboratory, Centre for Excellence in Functional Foods, Department of Food and Nutritional Biotechnology, National Agri-Food Biotechnology Institute (NABI), Sector 81, Mohali 140306, India.ORCID 0000-0002-4686-8361
Kanthi Kiran KondepudiTR(i)P for Health Laboratory, Centre for Excellence in Functional Foods, Department of Food and Nutritional Biotechnology, National Agri-Food Biotechnology Institute (NABI), Sector 81, Mohali 140306, India.ORCID 0000-0001-8036-7555
Kanwaljit ChopraUniversity Institute of Pharmaceutical Sciences, Panjab University, Chandigarh 160014, India.
Mahendra BishnoiTR(i)P for Health Laboratory, Centre for Excellence in Functional Foods, Department of Food and Nutritional Biotechnology, National Agri-Food Biotechnology Institute (NABI), Sector 81, Mohali 140306, India.ORCID 0000-0002-7785-1204
National Agri-Food Biotechnology Institute · INInstitute of Nano Science and TechnologyFriedrich-Alexander-Universität Erlangen-Nürnberg · DEPanjab University · INUniversity of Florida · US

Funding

Department of Biotechnology National Agri Food Biotechnology Institute
6 · The paper itself

Abstract

Antagonism of transient receptor potential vanniloid-1 (TRPV1) and desensitization of transient receptor potential ankyrin-1 (TRPA1) nociceptors alleviate inflammatory bowel diseases (IBD)-associated chronic pain. However, there is limited literature available about their role in regulating the mucosal layer, its interaction with host physiology, and luminal microbial community. The present study focuses on the effects' intra rectal administration of capsazepine (modulator of TRPA1/TRPV1 expressing peptidergic sensory neurons) on colonic mucus production and gut health. We performed histological analysis, gut permeability alteration, gene expression changes, metabolite profiling, and gut microbial abundance in the ileum, colon, and cecum content of these animals. Intra rectal administration of capsazepine modulates TRPA1/TRPV1-positive nociceptors (behavioral pain assays) and resulted in damaged mucosal lining, increased gut permeability, and altered transcriptional profile of genes for goblet cell markers, mucus regulation, immune response, and tight junction proteins. The damage to mucosal lining prevented its role in enterosyne (short chain fatty acids) actions. These results suggest that caution must be exercised before employing TRPA1/TRPV1 modulation as a therapeutic option to alleviate pain caused due to IBD.

Indexed as

Inflammatory Bowel DiseasesTransient Receptor Potential ChannelsAnimalsCapsaicinColonMicePainTRPA1 Cation ChannelTRPV Cation ChannelsCapsaicincapsazepineTransient Receptor Potential ChannelsTRPA1 Cation ChannelTRPV Cation ChannelscapsazepinemucinnociceptorsTRPA1TRPV1

Identifiers

PMID36076974
PMCPMC9455796
OpenAlexW4293001020

What Socratic holds

Textmetadata
LicenceCC BY
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.