Evidence mapPaperPMID 36897161Full record

Trial reportThe Journal of clinical endocrinology and metabolism2023

Defining Predictors of Weight Loss Response to Lorcaserin.

Aristea Sideri Gugger, Cara Dimino, Sunil K Panigrahi, Laurel Mayer, Richard M Smiley, Judith Korner, Sharon L Wardlaw

Registry-linked trialOpen access · bronzeAbstract readRandomized Controlled Trial
In one paragraph

Trial report in The Journal of clinical endocrinology and metabolism, 2023. The graph could read no effect estimate from its abstract, so it casts no vote on the map. It is linked to trial NCT03353220 (Central Mechanisms and Predictors of Lorcaserin-Induced Weight Loss), which is not on this map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
0.2field-weighted citation impact, top 56% of its field
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

NCT03353220 phase4terminatednot on this map

Central Mechanisms and Predictors of Lorcaserin-Induced Weight Loss

TypeinterventionalSponsorColumbia UniversityRan2018 to 2020Enrolled32ConditionsOverweight and ObesityArmsBelviq, Placebo
3 · Its place in the literature

Who cites it

0 citing papers in PubMed, 1 citations in OpenAlex.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

7 authors at 1 institution in 1 country.

Aristea Sideri GuggerDepartment of Medicine, Columbia University Vagelos College of Physicians and Surgeons, New York, NY 10032, USA.ORCID 0000-0003-0961-1038
Cara DiminoDepartment of Medicine, Columbia University Vagelos College of Physicians and Surgeons, New York, NY 10032, USA.
Sunil K PanigrahiDepartment of Medicine, Columbia University Vagelos College of Physicians and Surgeons, New York, NY 10032, USA.
Laurel MayerDepartment of Psychiatry, Columbia University Vagelos College of Physicians and Surgeons, New York, NY 10032, USA.
Richard M SmileyDepartment of Anesthesiology, Columbia University Vagelos College of Physicians and Surgeons, New York, NY 10032, USA.
Judith KornerDepartment of Medicine, Columbia University Vagelos College of Physicians and Surgeons, New York, NY 10032, USA.
Sharon L WardlawDepartment of Medicine, Columbia University Vagelos College of Physicians and Surgeons, New York, NY 10032, USA.ORCID 0000-0002-9659-7360
Columbia University · US

Funding

Clinical and Translational Science AwardUL1TR001873 · COLUMBIA UNIVERSITY HEALTH SCIENCES · 2025 to 2025
$10.0M
OBESITY RESEARCH CENTER TRAINING PROGRAMT32DK007559 · ST. LUKE'S-ROOSEVELT INST FOR HLTH SCIS · 1989 to 2025
$1.7M
NCATS NIH HHS UL1 TR001873NIDDK NIH HHS R01 DK093920NIDDK NIH HHS T32 DK007559NIH HHS R01-DK093920
6 · The paper itself

Abstract

contextIndividual responses to weight loss (WL) medications vary widely and prediction of response remains elusive.

objectiveWe investigated biomarkers associated with use of lorcaserin (LOR), a 5HT2cR agonist that targets proopiomelanocortin (POMC) neurons that regulate energy and glucose homeostasis, to identify predictors of clinical efficacy.

methodsThirty individuals with obesity were treated with 7 days of placebo and LOR in a randomized crossover study. Nineteen participants continued on LOR for 6 months. Cerebrospinal fluid (CSF) POMC peptide measurements were used to identify potential biomarkers that predict WL. Insulin, leptin, and food intake during a meal were also studied.

resultsLOR induced a significant decrease in CSF levels of the POMC prohormone and an increase in its processed peptide β-endorphin after 7 days; β-endorphin/POMC increased by 30% (P < .001). This was accompanied by a substantial decrease in insulin, glucose, and homeostasis model assessment of insulin resistance before WL. Changes in CSF POMC peptides persisted after WL (6.9%) at 6 months that were distinct from prior reports after diet alone. Changes in POMC, food intake, or other hormones did not predict WL. However, baseline CSF POMC correlated negatively with WL (P = .07) and a cutoff level of CSF POMC was identified that predicted more than 10% WL.

conclusionOur results provide evidence that LOR affects the brain melanocortin system in humans and that effectiveness is increased in individuals with lower melanocortin activity. Furthermore, early changes in CSF POMC parallel WL-independent improvements in glycemic indexes. Thus, assessment of melanocortin activity could provide a way to personalize pharmacotherapy of obesity with 5HT2cR agonists.

Indexed as

beta-EndorphinPro-OpiomelanocortinBenzazepinesCross-Over StudiesGlucoseHumansInsulinMelanocortinsObesityWeight LossBenzazepinesbeta-EndorphinGlucoseInsulinlorcaserinMelanocortinsPro-Opiomelanocortincerebrospinal fluidinsulinlorcaserinobesityproopiomelanocortin

Identifiers

PMID36897161
PMCPMC10438887
OpenAlexW4323805052

What Socratic holds

Textmetadata
Read underepoch 390

Registered trials

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.