ArticleBritish journal of pharmacology2023
The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors.
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Article in British journal of pharmacology, 2023. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 97 papers, 1 of them a synthesis that pooled it.
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97citing papers in PubMed, 1 pooled it
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Who cites it
97 citing papers in PubMed, 1 synthesis or guideline pooled it.
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37 more citing papers are in PubMed but not listed here.
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Authors and funding
166 authors.
Stephen P H AlexanderSchool of Life Sciences, University of Nottingham Medical School, Nottingham, NG7 2UH, UK.ORCID 0000-0003-4417-497X
Arthur ChristopoulosMonash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, 3052, Australia.ORCID 0000-0003-4442-3294
Anthony P DavenportClinical Pharmacology Unit, University of Cambridge, Cambridge, CB2 0QQ, UK.ORCID 0000-0002-2096-3117
Eamonn KellySchool of Physiology, Pharmacology and Neuroscience, University of Bristol, Bristol, BS8 1TD, UK.
Alistair A MathieSchool of Engineering, Arts, Science and Technology, University of Suffolk, Ipswich, IP4 1QJ, UK.ORCID 0000-0001-6094-2890
John A PetersNeuroscience Division, Medical Education Institute, Ninewells Hospital and Medical School, University of Dundee, Dundee, DD1 9SY, UK.ORCID 0000-0002-4277-4245
Emma L VealeMedway School of Pharmacy, The Universities of Greenwich and Kent at Medway, Anson Building, Central Avenue, Chatham Maritime, Chatham, Kent, ME4 4TB, UK.ORCID 0000-0002-6778-9929
Jane F ArmstrongCentre for Discovery Brain Sciences, University of Edinburgh, Edinburgh, EH8 9XD, UK.ORCID 0000-0002-0524-0260
Elena FaccendaCentre for Discovery Brain Sciences, University of Edinburgh, Edinburgh, EH8 9XD, UK.ORCID 0000-0001-9855-7103
Simon D HardingCentre for Discovery Brain Sciences, University of Edinburgh, Edinburgh, EH8 9XD, UK.ORCID 0000-0002-9262-8318
Jamie A DaviesCentre for Discovery Brain Sciences, University of Edinburgh, Edinburgh, EH8 9XD, UK.ORCID 0000-0001-6660-4032
Maria Pia AbbracchioUniversity of Milan, Milan, Italy.ORCID 0000-0002-7833-3388
George AbrahamClinical Pharmacology Unit, University of Cambridge, Cambridge, CB2 0QQ, UK.
Alexander AgoulnikFlorida International University, Miami, USA.
Wayne AlexanderEmory University, Atlanta, USA.
Khaled Al-HosainiKing Saud University, Riyadh, Kingdom of Saudi Arabia.
Magnus BäckKarolinska University Hospital, Stockholm, Sweden.ORCID 0000-0003-0853-5141
Jillian G BakerSchool of Life Sciences, University of Nottingham Medical School, Nottingham, NG7 2UH, UK.
Nicholas M BarnesUniversity of Birmingham, Birmingham, UK.
Ross BathgateFlorey Institute of Neuroscience and Mental Health, Melbourne, Australia.ORCID 0000-0001-6301-861X
Jean-Martin BeaulieuUniversity of Toronto, Toronto, Canada.ORCID 0000-0002-0446-7447
Annette G Beck-SickingerLeipzig University, Leipzig, Germany.ORCID 0000-0003-4560-8020
Maik BehrensTechnical University of Munich, Freising, Germany.ORCID 0000-0003-2082-8860
Kenneth E BernsteinCedars-Sinai Medical Center, Los Angeles, USA.ORCID 0000-0001-8097-3272
Bernhard BettlerUniversity of Basel, Basel, Switzerland.ORCID 0000-0003-0842-8207
Nigel J M BirdsallThe Francis Crick Institute, London, UK.
Victoria BlahoSanford Burnham Prebys Medical Discovery Institute, La Jolla, USA.ORCID 0000-0001-8499-2278
Francois BoulayUniversity of Grenoble Alpes, Grenoble, France.
Corinne BousquetFrench Institute of Health and Medical Research (INSERM), Toulouse, France.ORCID 0000-0002-2501-0593
Hans Bräuner-OsborneUniversity of Copenhagen, Copenhagen, Denmark.ORCID 0000-0001-9495-7388
Geoffrey BurnstockUniversity College London, London, UK.ORCID 0000-0001-8152-7979
Girolamo CalóUniversity of Padova, Padova, Italy.
Justo P CastañoUniversity of Córdoba, Córdoba, Spain.
Kevin J CattNational Institute of Health, Bethesda, USA.
Stefania CerutiUniversity of Milan, Milan, Italy.ORCID 0000-0003-1663-4211
Paul ChazotDurham University, Durham, UK.ORCID 0000-0002-5453-0379
Nan ChiangHarvard University, Boston, USA.ORCID 0000-0003-1963-1585
Bice ChiniUniversity of Milan Bicocca, Vedano al Lambro, Italy.ORCID 0000-0002-1686-284X
Jerold ChunUniversity of California San Diego, La Jolla, USA.ORCID 0000-0003-3964-0921
Antonia CianciulliUniversity of Bari, Bari, Italy.
Olivier CivelliUniversity of California Irvine, Irvine, USA.
Lucie H ClappUniversity College London, London, UK.ORCID 0000-0001-7802-4481
Réjean CoutureUniversity of Montréal, Montréal, Canada.
Helen M CoxKing's College London, London, UK.ORCID 0000-0001-9024-1497
Zsolt CsabaFrench Institute of Health and Medical Research (INSERM), Paris, France.
Claes DahlgrenUniversity of Gothenburg, Gothenburg, Sweden.
Gordon DentKeele University, Keele, UK.ORCID 0000-0001-9419-2952
Steven D DouglasUniversity of Pennsylvania, Pennsylvania, USA.
Pascal DournaudFrench Institute of Health and Medical Research (INSERM), Paris, France.
Satoru EguchiTemple University, Philadelphia, USA.
Emanuel EscherUniversity of Sherbrooke, Sherbrooke, Canada.
Edward J FilardoUniversity of Iowa, Iowa City, USA.
Tung FongLabcorp Drug Development, Somerset, USA.
Marta FumagalliUniversity of Milan, Milan, Italy.ORCID 0000-0002-0158-842X
Raul R GainetdinovSaint Petersburg State University, Saint-Petersburg, Russia.ORCID 0000-0003-2951-6038
Michael L GareljaUniversity of Otago, Dunedin, New Zealand.ORCID 0000-0001-5332-1236
Marc de GasparoMG Consulting Co, Basel, Switzerland.
Craig GerardHarvard University, Boston, USA.
Marvin GershengornNational Institute of Health, Bethesda, USA.
Fernand GobeilUniversity of Sherbrooke, Sherbrooke, Canada.
Theodore L GoodfriendUniversity of Wisconsin, Madison, USA.
Cyril GoudetFrench National Centre for Scientific Research, Montpellier, France.ORCID 0000-0002-8255-3535
Lukas GrätzKarolinska Institute, Stockholm, Sweden.
Karen J GregoryMonash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, 3052, Australia.ORCID 0000-0002-3833-2137
Andrew L GundlachFlorey Institute of Neuroscience and Mental Health, Melbourne, Australia.ORCID 0000-0002-6066-9692
Jörg HamannAmsterdam University, Amsterdam, The Netherlands.ORCID 0000-0002-9448-1727
Julien HansonUniversity of Liège, Liège, Belgium.ORCID 0000-0001-7063-7590
Richard L HaugerUniversity of California San Diego, La Jolla, USA.
Debbie L HayUniversity of Otago, Dunedin, New Zealand.ORCID 0000-0002-9558-5122
Akos HeinemannMedical University of Graz, Graz, Austria.ORCID 0000-0002-8554-2372
Deron HerrSan Diego State University, San Diego, USA.ORCID 0000-0001-5755-0896
Morley D HollenbergUniversity of Calgary, Calgary, Canada.
Nicholas D HollidaySchool of Life Sciences, University of Nottingham Medical School, Nottingham, NG7 2UH, UK.ORCID 0000-0002-2900-828X
Mastgugu HoriuchiEhime University, Ehime, Japan.
Daniel HoyerUniversity of Melbourne, Melbourne, Australia.ORCID 0000-0002-1405-7089
László HunyadySemmelweis University, Budapest, Hungary.
Ahsan HusainEmory University, Atlanta, USA.
Adriaan P IJzermanLeiden University, Leiden, The Netherlands.ORCID 0000-0002-1182-2259
Tadashi InagamiVanderbilt University, Nashville, USA.
Kenneth A JacobsonNational Institute of Health, Bethesda, USA.ORCID 0000-0001-8104-1493
Robert T JensenNational Institute of Health, Bethesda, USA.
Ralf JockersFrench Institute of Health and Medical Research (INSERM), Paris, France.ORCID 0000-0002-4354-1750
Deepa JonnalagaddaSanford Burnham Prebys Medical Discovery Institute, La Jolla, USA.ORCID 0000-0002-1511-8197
Sadashiva KarnikLerner Research Institute, Cleveland, USA.ORCID 0000-0003-0746-2753
Klemens KaupmannNovartis, Basel, Switzerland.ORCID 0000-0001-8903-2508
Jacqueline KempCleveland Clinic Lerner Research Institute, Cleveland, USA.
Charles KennedyStrathclyde University, Glasgow, UK.ORCID 0000-0001-9661-5437
Yasuyuki KiharaSanford Burnham Prebys Medical Discovery Institute, La Jolla, USA.ORCID 0000-0001-7462-3006
Takio KitazawaRakuno Gakuen University, Ebetsu, Japan.
Pawel KozielewiczKarolinska Institute, Stockholm, Sweden.ORCID 0000-0003-1414-3566
Hans-Jürgen KreienkampUniversity of Hamburg, Hamburg, Germany.
Jyrki P KukkonenUniversity of Helsinki, Helsinki, Finland.ORCID 0000-0002-6989-1564
Tobias LangenhanLeipzig University, Leipzig, Germany.ORCID 0000-0002-9061-3809
Dan LarhammarUppsala University, Uppsala, Sweden.ORCID 0000-0002-6736-0663
Katie LeachMonash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, 3052, Australia.ORCID 0000-0002-9280-1803
Davide LeccaUniversity of Milan, Milan, Italy.ORCID 0000-0002-3258-363X
John D LeeUniversity of Queensland, Brisbane, Australia.ORCID 0000-0002-9976-7396
Susan E LeemanBoston University, Boston, USA.
Jérôme LeprinceUniversity of Rouen, Rouen, France.ORCID 0000-0002-7814-9927
Xaria X LiUniversity of Queensland, Queensland, Australia.ORCID 0000-0001-5924-2977
Stephen J LolaitSchool of Physiology, Pharmacology and Neuroscience, University of Bristol, Bristol, BS8 1TD, UK.ORCID 0000-0001-7228-8072
Amelie LuppFriedrich Schiller University Jena, Jena, Germany.
Robyn MacraeUniversity of Cambridge, Cambridge, UK.
Janet MaguireClinical Pharmacology Unit, University of Cambridge, Cambridge, CB2 0QQ, UK.ORCID 0000-0002-9254-7040
Davide MalfaciniUniversity of Padova, Padova, Italy.
Jean MazellaFrench National Centre for Scientific Research (CNRS), Valbonne, France.ORCID 0000-0002-5627-0742
Craig A McArdleSchool of Physiology, Pharmacology and Neuroscience, University of Bristol, Bristol, BS8 1TD, UK.ORCID 0000-0003-4836-5351
Shlomo MelmedCedars-Sinai Medical Center, Los Angeles, USA.
Martin C MichelJohannes Gutenberg University Mainz, Mainz, Germany.ORCID 0000-0003-4161-8467
Laurence J MillerMayo Foundation for Medical Education and Research, Scottsdale, USA.ORCID 0000-0002-4554-3872
Vincenzo MitoloUniversity of Bari, Bari, Italy.
Bernard MouillacFrench National Centre for Scientific Research, Montpellier, France.ORCID 0000-0002-3906-8673
Christa E MüllerUniversity of Bonn, Bonn, Germany.ORCID 0000-0002-0013-6624
Philip M MurphyEdge Hill University, Bethesda, USA.
Jean-Louis NahonFrench National Centre for Scientific Research (CNRS), Valbonne, France.ORCID 0000-0001-9572-7779
Tony NgoSanford Burnham Prebys Medical Discovery Institute, La Jolla, USA.ORCID 0000-0002-6779-2546
Xavier NorelFrench Institute of Health and Medical Research (INSERM), Paris, France.ORCID 0000-0003-0734-3359
Duuamene NyimanuUniversity of Cambridge, Cambridge, UK.
Anne-Marie O'CarrollSchool of Physiology, Pharmacology and Neuroscience, University of Bristol, Bristol, BS8 1TD, UK.ORCID 0000-0001-5255-8506
Stefan OffermannsMax Planck Institute for Heart and Lung Research, Bad Nauheim, Germany.ORCID 0000-0001-8676-6805
Maria Antonietta PanaroUniversity of Bari, Bari, Italy.
Marc ParmentierFree University of Brussels, Brussels, Belgium.
Roger G PertweeUniversity of Aberdeen, Aberdeen, UK.ORCID 0000-0003-3227-2783
Jean-Philippe PinUniversity of Montpellier, Montpellier, France.ORCID 0000-0002-1423-345X
Eric R ProssnitzUniversity of New Mexico, Albuquerque, USA.ORCID 0000-0001-9190-8302
Mark QuinnMontana State University, Bozeman, USA.
Rithwik RamachandranUniversity of Calgary, Calgary, Canada.ORCID 0000-0001-9557-9905
Manisha RaySanford Burnham Prebys Medical Discovery Institute, La Jolla, USA.ORCID 0000-0002-8844-6191
Rainer K ReinscheidFriedrich Schiller University Jena, Jena, Germany.
Philippe RondardUniversity of Montpellier, Montpellier, France.ORCID 0000-0003-1134-2738
G Enrico RovatiUniversity of Milan, Milan, Italy.ORCID 0000-0002-8788-9783
Chiara RuzzaUniversity of Ferrara, Ferrara, Italy.ORCID 0000-0003-1360-202X
Gareth J SangerQueen Mary University of London, London, UK.ORCID 0000-0002-4231-1945
Torsten SchönebergLeipzig University, Leipzig, Germany.ORCID 0000-0001-5313-0237
Gunnar SchulteKarolinska Institute, Stockholm, Sweden.ORCID 0000-0002-2700-7013
Stefan SchulzFriedrich Schiller University Jena, Jena, Germany.
Deborah L SegaloffUniversity of Iowa, Iowa City, USA.
Charles N SerhanHarvard University, Boston, USA.
Khuraijam Dhanachandra SinghCleveland Clinic Lerner Research Institute, Cleveland, USA.ORCID 0000-0003-0506-6896
Craig M SmithDeakin University, Waurn Ponds, Australia.
Leigh A StoddartSchool of Life Sciences, University of Nottingham Medical School, Nottingham, NG7 2UH, UK.ORCID 0000-0002-4469-0600
Yukihiko SugimotoKumamoto University, Kumamoto, Japan.ORCID 0000-0001-6973-932X
Roger SummersMonash University, Melbourne, Australia.ORCID 0000-0002-8367-4056
Valerie P TanUniversity of California San Diego, La Jolla, USA.ORCID 0000-0002-7308-1601
David ThalMonash University, Melbourne, Australia.ORCID 0000-0002-0325-2524
Walter Wally ThomasUniversity of Queensland, Queensland, Australia.
Pieter B M W M TimmermansKosan Biosciences Inc., San Francisco, USA.
Kalyan TirupulaCleveland Clinic Lerner Research Institute, Cleveland, USA.
Lawrence TollFlorida Atlantic University, Jupiter, USA.ORCID 0000-0002-4501-7573
Giovanni TulipanoUniversity of Brescia, Brescia, Italy.
Hamiyet UnalCleveland Clinic, Cleveland, USA.
Thomas UngerMaastricht University, Maastricht, The Netherlands.
Celine ValantMonash University, Melbourne, Australia.ORCID 0000-0002-2509-7465
Patrick VanderheydenFree University of Brussels, Brussels, Belgium.
David VaudryUniversity of Rouen, Rouen, France.
Hubert VaudryUniversity of Rouen, Rouen, France.
Jean-Pierre VilardagaUniversity of Pittsburgh, Pittsburgh, USA.
Christopher S WalkerUniversity of Auckland, Auckland, New Zealand.ORCID 0000-0001-8151-4123
Ji Ming WangNational Institute of Health, Frederick, USA.
Donald T WardUniversity of Manchester, Manchester, UK.ORCID 0000-0003-1342-9458
Hans-Jürgen WesterTechnical University of Munich, Munich, Germany.
Gary B WillarsUniversity of Leicester, Leicester, UK.
Tom Lloyd WilliamsUniversity of Cambridge, Cambridge, UK.
Trent M WoodruffUniversity of Queensland, Queensland, Australia.ORCID 0000-0003-1382-911X
Chengcan YaoUniversity of Edinburgh, Edinburgh, UK.ORCID 0000-0003-3754-2842
Richard D YeThe Chinese University of Hong Kong, Shenzhen, China.
Funding
Altered reverse transcriptase-dependent gene diversification mechanisms in Alzheimer's disease brainsR01AG065541 · NIA · SANFORD BURNHAM PREBYS MEDICAL DISCOVERY INSTITUTE · PI JEROLD CHUN · 2022 to 2024
$2.8MCancer Research UK 25246Medical Research Council MR/R008167/1NHLBI NIH HHS R01 HL132351NIA NIH HHS R01 AG065541
Abstract
The Concise Guide to PHARMACOLOGY 2023/24 is the sixth in this series of biennial publications. The Concise Guide provides concise overviews, mostly in tabular format, of the key properties of approximately 1800 drug targets, and about 6000 interactions with about 3900 ligands. There is an emphasis on selective pharmacology (where available), plus links to the open access knowledgebase source of drug targets and their ligands (https://www.guidetopharmacology.org), which provides more detailed views of target and ligand properties. Although the Concise Guide constitutes almost 500 pages, the material presented is substantially reduced compared to information and links presented on the website. It provides a permanent, citable, point-in-time record that will survive database updates. The full contents of this section can be found at http://onlinelibrary.wiley.com/doi/bph.16177. G protein-coupled receptors are one of the six major pharmacological targets into which the Guide is divided, with the others being: ion channels, nuclear hormone receptors, catalytic receptors, enzymes and transporters. These are presented with nomenclature guidance and summary information on the best available pharmacological tools, alongside key references and suggestions for further reading. The landscape format of the Concise Guide is designed to facilitate comparison of related targets from material contemporary to mid-2023, and supersedes data presented in the 2021/22, 2019/20, 2017/18, 2015/16 and 2013/14 Concise Guides and previous Guides to Receptors and Channels. It is produced in close conjunction with the Nomenclature and Standards Committee of the International Union of Basic and Clinical Pharmacology (NC-IUPHAR), therefore, providing official IUPHAR classification and nomenclature for human drug targets, where appropriate.
Indexed as
Databases, PharmaceuticalReceptors, G-Protein-CoupledHumansIon ChannelsLigandsReceptors, Cytoplasmic and NuclearIon ChannelsLigandsReceptors, Cytoplasmic and NuclearReceptors, G-Protein-Coupled
Identifiers
What Socratic holds
Textmetadata
LicenceCC BY
Read underepoch 390
Registered trials
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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.