Evidence map›Paper›PMID 38352172›Full record

Trial reportDrug design, development and therapy2024

Pharmacokinetic Comparison Between a Fixed-Dose Combination of Atorvastatin/Omega-3-Acid Ethyl Esters and the Corresponding Loose Combination in Healthy Korean Male Subjects.

Juyoung Khwarg, Soyoung Lee, In-Jin Jang, Won-Ho Kang, Hye Jung Lee, Kyu Yeon Kim, Ki-Sun Jeong, Chongho Won, Youn Woong Choi, Dae Chul Ha and 7 more

Open access · goldAbstract readRandomized Controlled Trial
In one paragraph

Trial report in Drug design, development and therapy, 2024. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
–field-weighted citation impact, top 97% of its field
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed, 0 citations in OpenAlex.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

17 authors at 4 institutions in 2 countries.

Juyoung KhwargDepartment of Clinical Pharmacology and Therapeutics, Seoul National University College of Medicine and Hospital, Seoul, Republic of Korea.ORCID 0000-0001-7097-2006
Soyoung LeeDepartment of Clinical Pharmacology and Therapeutics, Seoul National University College of Medicine and Hospital, Seoul, Republic of Korea.ORCID 0000-0001-5799-4489
In-Jin JangDepartment of Clinical Pharmacology and Therapeutics, Seoul National University College of Medicine and Hospital, Seoul, Republic of Korea.ORCID 0000-0002-8384-3139
Won-Ho KangR&D Center, Korea United Pharm. Inc., Seoul, Republic of Korea.
Hye Jung LeeCaleb Multilab, Inc., Seoul, Republic of Korea.
Kyu Yeon KimCaleb Multilab, Inc., Seoul, Republic of Korea.ORCID 0000-0002-1708-9932
Ki-Sun JeongCaleb Multilab, Inc., Seoul, Republic of Korea.ORCID 0000-0002-6181-2665
Chongho WonCaleb Multilab, Inc., Seoul, Republic of Korea.
Youn Woong ChoiR&D Center, Korea United Pharm.Inc., Sejong, Republic of Korea.
Dae Chul HaR&D Center, Korea United Pharm.Inc., Sejong, Republic of Korea.
RaeHoon JungR&D Center, Korea United Pharm.Inc., Sejong, Republic of Korea.
Min-Gu HanR&D Center, Korea United Pharm.Inc., Sejong, Republic of Korea.
Won Tae JungGlobal R&D, Korea United Pharm. Inc., Seoul, Republic of Korea.
Kyu-Yeol NamGlobal R&D, Korea United Pharm. Inc., Seoul, Republic of Korea.
YeSeul KimGlobal R&D, Korea United Pharm. Inc., Seoul, Republic of Korea.
Kyung-Sang YuDepartment of Clinical Pharmacology and Therapeutics, Seoul National University College of Medicine and Hospital, Seoul, Republic of Korea.ORCID 0000-0003-0921-7225
Jaeseong OhDepartment of Clinical Pharmacology and Therapeutics, Seoul National University College of Medicine and Hospital, Seoul, Republic of Korea.ORCID 0000-0001-6275-8587
Korea Pharma (South Korea) · KRCaleb University · NGSeoul National University Hospital · KRSeoul National University · KR

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Purpose: Statins are widely used in combination with omega-3 fatty acids for the treatment of patients with dyslipidemia. The aim of this study was to compare the pharmacokinetic (PK) profiles of atorvastatin and omega-3-acid ethyl esters between fixed-dose combination (FDC) and loose combination in healthy subjects. Methods: A randomized, open-label, single-dose, 2-sequence, 2-treatment, 4-period replicated crossover study was performed. Subjects were randomly assigned to one of the 2 sequences and alternately received four FDC soft capsules of atorvastatin/omega-3-acid ethyl esters (10/1000 mg) or a loose combination of atorvastatin tablets (10 mg × 4) and omega-3-acid ethyl ester soft capsules (1000 mg× 4) for four periods, each period accompanied by a high-fat meal. Serial blood samples were collected for PK analysis of atorvastatin, eicosapentaenoic acid (EPA), and docosahexaenoic acid (DHA). PK parameters were calculated by a non-compartmental analysis. The geometric mean ratio (GMR) and its 90% confidence interval (CI) of the FDC to the loose combination were calculated to compare PK parameters. Results: A total of 43 subjects completed the study as planned. The GMR (90% CI) of FDC to loose combination for maximum concentration (C Conclusion: The FDC of atorvastatin and omega-3-acid ethyl esters showed comparable PK characteristics to the corresponding loose combination, offering a convenient therapeutic option for the treatment of dyslipidemia.

Indexed as

DyslipidemiasEicosapentaenoic AcidArea Under CurveAtorvastatinCross-Over StudiesDocosahexaenoic AcidsDrug CombinationsHealthy VolunteersHumansMaleRepublic of KoreaAtorvastatinDocosahexaenoic AcidsDrug CombinationsEicosapentaenoic Acidcardiovascular diseasepharmacokinetics

Identifiers

PMID38352172
PMCPMC10861834
OpenAlexW4391671052

What Socratic holds

Textmetadata
LicenceCC BY-NC
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.