Evidence map›Paper›PMID 38454939›Full record

ReviewRSC advances2024

Synthesis and pharmacological activity of vinpocetine derivatives.

Zhang Chao Dong, Yang Shi, Li Juan Liu, Ting Ting Feng, Ying Zhou, Bo Wen Pan

Open access · goldAbstract readReview
In one paragraph

Review in RSC advances, 2024. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 5 papers.

0numbers the graph read from it
0cells of the map it votes in
5citing papers in PubMed
2.2field-weighted citation impact, top 13% of its field
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

5 citing papers in PubMed, 9 citations in OpenAlex.

  1. Article
  2. Article
  3. Review
  4. Article
  5. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

6 authors.

Zhang Chao DongCollege of Pharmacy, Guizhou University of Traditional Chinese Medicine Guiyang 550025 China bwpan1105@163.com yingzhou71@126.com.
Yang ShiCollege of Pharmacy, Guizhou University of Traditional Chinese Medicine Guiyang 550025 China bwpan1105@163.com yingzhou71@126.com.
Li Juan LiuCollege of Pharmacy, Guizhou University of Traditional Chinese Medicine Guiyang 550025 China bwpan1105@163.com yingzhou71@126.com.
Ting Ting FengCollege of Pharmacy, Guizhou University of Traditional Chinese Medicine Guiyang 550025 China bwpan1105@163.com yingzhou71@126.com.
Ying ZhouCollege of Pharmacy, Guizhou University of Traditional Chinese Medicine Guiyang 550025 China bwpan1105@163.com yingzhou71@126.com.
Bo Wen PanCollege of Pharmacy, Guizhou University of Traditional Chinese Medicine Guiyang 550025 China bwpan1105@163.com yingzhou71@126.com.ORCID https://orcid.org/0000-0003-0930-4492

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Vinpocetine and its derivatives were extensively employed in the treatment of ischemic stroke, serving as effective cerebrovascular vasodilators. They could also be utilized for neuroprotection, anti-inflammatory purposes, anti-aging interventions, insomnia treatment, and antidepressant effects. However, due to issues such as hepatic first-pass effect, low bioavailability, and poor patient compliance with multiple dosing, the secondary development of Vinpocetine to address these limitations became a prominent area of research. Five primary methodologies were employed for the synthesis of Vinpocetine derivatives. These included substitution on the A ring to modify the 14-ester group, alteration of the 16-ethyl group, simplification of the D and E rings, and modification of the conformation of Vinpocetine. This paper summarized the current synthesis and activity studies of Vinpocetine and its derivatives, with the aim of providing a reference for the discovery of more potent derivatives of Vinpocetine.

Identifiers

PMID38454939
PMCPMC10918451
OpenAlexW4392565948

What Socratic holds

Textmetadata
LicenceCC BY-NC
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.