Evidence mapPaperPMID 39312270Full record

ArticlePharmacology research & perspectives2024

Plasma and urinary CP I and CP III concentrations in chimeric mice with human hepatocytes after rifampicin administration.

Yurina Shishido, Tomohiro Yoshida, Keiyu Oshida, Masashi Uchida

Abstract read
In one paragraph

Article in Pharmacology research & perspectives, 2024. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 2 papers.

0numbers the graph read from it
0cells of the map it votes in
2citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

2 citing papers in PubMed.

  1. Article
  2. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

4 authors.

Yurina ShishidoPharmaceutical Research Laboratories, Toray Industries, Inc., Kamakura, Kanagawa, Japan.
Tomohiro YoshidaPharmaceutical Research Laboratories, Toray Industries, Inc., Kamakura, Kanagawa, Japan.
Keiyu OshidaPharmaceutical Research Laboratories, Toray Industries, Inc., Kamakura, Kanagawa, Japan.
Masashi UchidaPharmaceutical Research Laboratories, Toray Industries, Inc., Kamakura, Kanagawa, Japan.ORCID 0009-0007-0541-9715

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

The interest in transporter-mediated drug interactions has been increasing in the field of drug development. In this study, we measured the plasma and urinary concentrations of coproporphyrin (CP) I and CP III as endogenous substrates for organic anion-transporting polypeptide (OATP) using chimeric mice with human hepatocytes (PXB mice) and examined the influence of an OATP inhibitor, rifampicin (RIF). CP I and CP III were actively taken up intracellularly, and RIF inhibited the uptake in a concentration-dependent manner for both CP I and CP III in human hepatocytes (PXB-cells). Single doses of RIF at 10 and 30 mg/kg were orally or intravenously administered to PXB mice and wild-type ICR mice. Plasma concentrations (AUC

Indexed as

CoproporphyrinsHepatocytesMice, Inbred ICRRifampinAdministration, IntravenousAnimalsChimeraDrug InteractionsHumansMaleMiceOrganic Anion Transporterscoproporphyrin ICoproporphyrinsOrganic Anion TransportersRifampincoproporphyrinsorganic anion‐transporting polypeptide (OATP)PXB micerifampicintransporter‐mediated drug interactions

Identifiers

PMID39312270
PMCPMC11418634

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.