Evidence map›Paper›PMID 39408903›Full record

ArticleInternational journal of molecular sciences2024

Enantioselective Binding of Proton Pump Inhibitors to Alpha1-Acid Glycoprotein and Human Serum Albumin-A Chromatographic, Spectroscopic, and In Silico Study.

Gergely Dombi, Levente Tyukodi, Máté Dobó, Gergely Molnár, Zsuzsanna Rozmer, Zoltán-István Szabó, Béla Fiser, Gergő Tóth

Abstract read
In one paragraph

Article in International journal of molecular sciences, 2024. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 6 papers.

0numbers the graph read from it
0cells of the map it votes in
6citing papers in PubMed
–field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

6 citing papers in PubMed.

  1. Article
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  3. Review
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4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

8 authors.

Gergely DombiDepartment of Pharmaceutical Chemistry, Semmelweis University, Hogyes E. 9, 1092 Budapest, Hungary.
Levente TyukodiDepartment of Pharmaceutical Chemistry, University of Pécs, 7624 Pécs, Hungary.ORCID 0000-0002-8983-1876
Máté DobóDepartment of Pharmaceutical Chemistry, Semmelweis University, Hogyes E. 9, 1092 Budapest, Hungary.
Gergely MolnárDepartment of Pharmaceutical Chemistry, Semmelweis University, Hogyes E. 9, 1092 Budapest, Hungary.
Zsuzsanna RozmerDepartment of Pharmaceutical Chemistry, University of Pécs, 7624 Pécs, Hungary.
Zoltán-István SzabóDepartment of Pharmaceutical Industry and Management, Faculty of Pharmacy, George Emil Palade University of Medicine, Pharmacy, Science, and Technology of Targu Mures, Gh. Marinescu 38, 540142 Targu Mures, Romania.ORCID 0000-0002-8740-0212
Béla FiserInstitute of Chemistry, University of Miskolc, 3515 Miskolc, Hungary.ORCID 0000-0003-0603-4626
Gergő TóthDepartment of Pharmaceutical Chemistry, Semmelweis University, Hogyes E. 9, 1092 Budapest, Hungary.ORCID 0000-0001-5341-319X

Funding

Hungarian Academy of Sciences the János Bolyai Research ScholarshipMinistry for Culture and Innovation ÚNKP-23-3-II-SE-3 (M.D), ÚNKP-23-2-III-SE-6 (G.D) and 2023-2.1.1-ÚNKP-2023-00002 (L. Ty.)National Research, Development and Innovation Fund TKP2021-NVA-14National Research, Development and Innovation Office, Hungary NKFIH FK 146930
6 · The paper itself

Abstract

The enantioselective binding of three proton pump inhibitors (PPIs)-omeprazole, rabeprazole, and lansoprazole-to two key plasma proteins, α1-acid glycoprotein (AGP) and human serum albumin (HSA), was characterized. The interactions between PPI enantiomers and proteins were investigated using a multifaceted analytical approach, including high-performance liquid chromatography (HPLC), fluorescence and UV spectroscopy, as well as in silico molecular docking. HPLC analysis demonstrated that all three PPIs exhibited enantioseparation on an AGP-based chiral stationary phase, suggesting stereoselective binding to AGP, while only lansoprazole showed enantioselective binding on the HSA-based column. Quantitatively, the

Indexed as

Molecular Docking SimulationOrosomucoidProtein BindingProton Pump InhibitorsSerum Albumin, HumanChromatography, High Pressure LiquidHumansOmeprazoleRabeprazoleSpectrometry, FluorescenceStereoisomerismThermodynamicsOmeprazoleOrosomucoidProton Pump InhibitorsRabeprazoleSerum Albumin, HumanAGPHPLCHSAprotein bindingproton pump inhibitorstransport proteins

Identifiers

PMID39408903
PMCPMC11477000

What Socratic holds

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Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.