Evidence mapPaperPMID 39760829Full record

ArticleArchives of pharmacal research2025

Physiologically based pharmacokinetic (PBPK) modeling of gliclazide for different genotypes of CYP2C9 and CYP2C19.

Hye-Jung Park, Sang-Ho Lee, Pureum Kang, Chang-Keun Cho, Choon-Gon Jang, Seok-Yong Lee, Yun Jeong Lee, Jung-Woo Bae, Chang-Ik Choi

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Article in Archives of pharmacal research, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 1 paper.

0numbers the graph read from it
0cells of the map it votes in
1citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

1 citing paper in PubMed.

  1. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

9 authors.

Hye-Jung Park *School of Pharmacy, Sungkyunkwan University, Suwon, 16419, Republic of Korea.
Sang-Ho Lee *School of Pharmacy, Sungkyunkwan University, Suwon, 16419, Republic of Korea.
Pureum Kang *School of Pharmacy, Sungkyunkwan University, Suwon, 16419, Republic of Korea.
Chang-Keun ChoSchool of Pharmacy, Sungkyunkwan University, Suwon, 16419, Republic of Korea.
Choon-Gon JangSchool of Pharmacy, Sungkyunkwan University, Suwon, 16419, Republic of Korea.
Seok-Yong LeeSchool of Pharmacy, Sungkyunkwan University, Suwon, 16419, Republic of Korea. sylee@skku.edu.ORCID http://orcid.org/0000-0003-4162-1981
Yun Jeong LeeCollege of Pharmacy, Dankook University, Cheonan, 31116, Republic of Korea.
Jung-Woo BaeCollege of Pharmacy, Keimyung University, Daegu, 42601, Republic of Korea.
Chang-Ik ChoiCollege of Pharmacy, Dongguk University-Seoul, Goyang, 10326, Republic of Korea. cichoi@dongguk.edu.

Funding

Ministry of Science and ICT, South Korea NRF-2019R1A2C1004582Ministry of Science and ICT, South Korea NRF-2019R1C1C1006213
6 · The paper itself

Abstract

Gliclazide is a sulfonylurea hypoglycemic agent used to treat type 2 diabetes. Cytochrome P450 (CYP) 2C9 and CYP2C19 are primarily involved in the hepatic metabolism of gliclazide. The two CYP isozymes are highly polymorphic, and their genetic polymorphisms are known to significantly impact the pharmacokinetics of gliclazide. In the present study, the physiologically based pharmacokinetic (PBPK) model was developed using data from subjects whose pharmacokinetic parameters were influenced by the genetic polymorphisms of the CYP metabolic enzymes. All predicted plasma concentration-time profiles generated by the model showed visual agreement with the observed data, and the pharmacokinetic results were within the twofold error range. Individual simulation results showed additional metrics: average fold error (- 0.19 to 0.07), geometric mean fold error (1.13-1.56), and mean relative deviation (1.18-1.58) for AUC, C

Indexed as

Cytochrome P-450 CYP2C19Cytochrome P-450 CYP2C9GliclazideHypoglycemic AgentsModels, BiologicalAdultFemaleGenotypeHumansMaleMiddle AgedPolymorphism, GeneticCYP2C19 protein, humanCYP2C9 protein, humanCytochrome P-450 CYP2C19Cytochrome P-450 CYP2C9GliclazideHypoglycemic AgentsCYP2C19CYP2C9Genetic polymorphismGliclazidePharmacokineticsPhysiologically based pharmacokinetic (PBPK) model

Identifiers

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.