Evidence mapPaperPMID 39819475Full record

ArticleBMC cancer2025

Prostate cancer cells elevate glycolysis and G6PD in response to caffeic acid phenethyl ester-induced growth inhibition.

Tzu-Ping Lin, Pei-Chun Chen, Ching-Yu Lin, Bi-Juan Wang, Ying-Yu Kuo, Chien-Chih Yeh, Jen-Chih Tseng, Chieh Huo, Cheng-Li Kao, Li-Jane Shih and 4 more

Abstract read
In one paragraph

Article in BMC cancer, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 2 papers.

0numbers the graph read from it
0cells of the map it votes in
2citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

2 citing papers in PubMed.

  1. Article
  2. Review
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

14 authors.

Tzu-Ping Lin *Faculty of Medicine, National Yang Ming Chiao Tung University, Hsinchu City, 30010, Taiwan.
Pei-Chun Chen *Institute of Cellular and System Medicine, National Health Research Institutes, Miaoli County, 35053, Taiwan.
Ching-Yu LinInstitute of Cellular and System Medicine, National Health Research Institutes, Miaoli County, 35053, Taiwan.
Bi-Juan WangInstitute of Cellular and System Medicine, National Health Research Institutes, Miaoli County, 35053, Taiwan.
Ying-Yu KuoInstitute of Cellular and System Medicine, National Health Research Institutes, Miaoli County, 35053, Taiwan.
Chien-Chih YehDepartment of Education and Medical Research, Taoyuan Armed Forces General Hospital, Taoyuan City, 325208, Taiwan.
Jen-Chih TsengInstitute of Cellular and System Medicine, National Health Research Institutes, Miaoli County, 35053, Taiwan.
Chieh HuoInstitute of Cellular and System Medicine, National Health Research Institutes, Miaoli County, 35053, Taiwan.
Cheng-Li KaoDivision of Urology, Departments of Surgery, Tri-Service General Hospital, National Defense Medical Center, Taipei City, 114202, Taiwan.
Li-Jane ShihDivision of Colon and Rectal Surgery, Department of Surgery, Tri-Service General Hospital, National Defense Medical Center, Taipei City, 114202, Taiwan.
Jen-Kun ChenInstitute of Biomedical Engineering and Nanomedicine, National Health Research Institutes, Miaoli County, 35053, Taiwan.
Chia-Yang LiGraduate Institute of Medicine, College of Medicine, Kaohsiung Medical University, Kaohsiung City, 80708, Taiwan.
Tzyh-Chyuan HourNeuroscience Research Center, Kaohsiung Medical University, Kaohsiung City, 80708, Taiwan.
Chih-Pin ChuuInstitute of Cellular and System Medicine, National Health Research Institutes, Miaoli County, 35053, Taiwan. cpchuu@nhri.edu.tw.

Funding

Ministry of Science and Technology, Taiwan NSTC 111-2811-B-400-029; NSTC 112-2320-B-400-008; NSTC 112-2314-B-400-031; NSTC 112-2314-B-037-128National Health Research Institutes CS-110-PP-03; CS-111-PP-03; CS-113-SP-04Taoyuan Armed Forces General Hospital TYAFGH-A-111008, TYAFGH-A-112006, TYAFGH-A-113007
6 · The paper itself

Abstract

backgroundCaffeic acid phenethyl ester (CAPE) is the main bioactive component of poplar type propolis. We previously reported that treatment with caffeic acid phenethyl ester (CAPE) suppressed the cell proliferation, tumor growth, as well as migration and invasion of prostate cancer (PCa) cells via inhibition of signaling pathways of AKT, c-Myc, Wnt and EGFR. We also demonstrated that combined treatment of CAPE and docetaxel altered the genes involved in glycolysis and tricarboxylic acid (TCA) cycle. We therefore suspect that CAPE treatment may interfere glucose metabolism in PCa cells.

methodsSeahorse Bioenergetics platform was applied to analyzed the extra cellular acidification rate (ECAR) and oxygen consumption rate (OCR) of PCa cells under CAPE treatment. UPLC-MSMS with Multiple Reaction Monitoring (MRM), PCR, and western blot were used to analyze the effects of CAPE on metabolites, genes, and proteins involved in glycolysis, TCA cycle and pentose phosphate pathway in PCa cells. Flow cytometry and ELISA were used to determine the level of reactive oxygen species in PCa cells being treated with CAPE.

resultsSeahorse Bioenergetics analysis revealed that ECAR, glycolysis, OCR, and ATP production were elevated in C4-2B cells under CAPE treatment. Protein levels of glucose-6-phosphate dehydrogenase (G6PD), phosphogluconate dehydrogenase (PGD), glutaminase (GLS), phospho-AMPK Thr172 as well as abundance of pyruvate, lactate, ribulose-5-phosphate, and sedoheptulose-7-phosphate were increased in CAPE-treated C4-2B cells. ROS level decreased 48 h after treatment with CAPE. Co-treatment of AMPK inhibitor with CAPE exhibited additive growth inhibition on PCa cells.

conclusionsOur study indicated that PCa cells attempted to overcome the CAPE-induced stress by upregulation of glycolysis and G6PD but failed to impede the growth inhibition caused by CAPE. Concurrent treatment of CAPE and inhibitors targeting glycolysis may be effective therapy for advanced PCa.

Indexed as

Caffeic AcidsGlucosephosphate DehydrogenaseGlycolysisPhenylethyl AlcoholProstatic NeoplasmsCell Line, TumorCell ProliferationCitric Acid CycleEnergy MetabolismHumansMaleReactive Oxygen Speciescaffeic acid phenethyl esterCaffeic AcidsGlucosephosphate DehydrogenasePhenylethyl AlcoholReactive Oxygen SpeciesCaffeic acid phenethyl esterG6PDGlycolysisLactateProstate cancerPyruvate

Identifiers

PMID39819475
PMCPMC11737093

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.