Evidence mapPaperPMID 39910656Full record

ArticleCell & bioscience2025

Epsin3 promotes non-small cell lung cancer progression via modulating EGFR stability.

Huiling Su, Jie Shen, Chenzi Gao, Yue Zhao, Wanyu Deng, Bo Qin, Xin Zhang, Juan Lai, Qian Wang, Jie Dou and 1 more

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Article in Cell & bioscience, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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1 · What the graph read from it

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4 · The record

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5 · Who and what money

Authors and funding

11 authors.

Huiling Su *State Key Laboratory of Natural Medicines, School of Life Science & Technology, Pharmaceutical University, 210009, Nanjing, China.
Jie Shen *State Key Laboratory of Natural Medicines, School of Life Science & Technology, Pharmaceutical University, 210009, Nanjing, China.
Chenzi Gao *Key Laboratory of Human Functional Genomics of Jiangsu Province, Department of Biochemistry and Molecular Biology, Nanjing Medical University, 210029, Nanjing, China.
Yue ZhaoState Key Laboratory of Natural Medicines, School of Life Science & Technology, Pharmaceutical University, 210009, Nanjing, China.
Wanyu DengCollege of Life Science, Shangrao Normal University, 334001, Shangrao, China.
Bo QinShaoxing Women and Children's Hospital, 312000, Shaoxing, China.
Xin ZhangGeneMind Biosciences Company Limited, 518001, Shenzhen, China.
Juan LaiGeneMind Biosciences Company Limited, 518001, Shenzhen, China.
Qian WangKey Laboratory of Human Functional Genomics of Jiangsu Province, Department of Biochemistry and Molecular Biology, Nanjing Medical University, 210029, Nanjing, China. wqian@njmu.edu.cn.
Jie DouState Key Laboratory of Natural Medicines, School of Life Science & Technology, Pharmaceutical University, 210009, Nanjing, China. doujie@cpu.edu.cn.
Min GuoState Key Laboratory of Natural Medicines, School of Life Science & Technology, Pharmaceutical University, 210009, Nanjing, China. 1020152471@cpu.edu.cn.ORCID http://orcid.org/0000-0003-4945-5877

Funding

Education Department Science and Technology Foundation of Jiangxi GJJ211720Guangdong Provincial Introduction of Innovative Research and Development Team SRPG23-GZNL2023A02008Major Project of Guangzhou National Laboratory SRPG22-002National Natural Science Foundation of China 81700756National Natural Science Foundation of China 82260603Postgraduate Research & Practice Innovation Program of Jiangsu Province KYCX23_0860
6 · The paper itself

Abstract

backgroundThe abnormal expression and overactivation of the epidermal growth factor receptor (EGFR), a typical cancer marker for non-small cell lung cancer (NSCLC), are closely related to the tumorigenesis and progression of NSCLC. However, the endocytosis mechanism of EGFR in lung cancer is not yet known. Epsin3 (EPN3), a member of the endocytic adaptor protein family, is essential for the endocytosis of multiple receptors. In this study, we aimed to investigate the role of EPN3 in modulating EGFR function, its effects on NSCLC progression, and its potential involvement in tyrosine kinase inhibitor (TKI) resistance, which remains a significant hurdle in NSCLC treatment.

resultsOur findings revealed that the expression of EPN3 is significantly up-regulated in NSCLC patients. Elevated EPN3 expression was proportional to shorter overall survival in patients with NSCLC. Functional analyses revealed that EPN3 directly interacts with EGFR, enhancing its recycling to the plasma membrane and preventing its degradation via the lysosomal pathway. This stabilization of EGFR led to sustained downstream signalling, promoting NSCLC cell proliferation and migration. Notably, mutations in the EGFR tyrosine kinase domain, which typically confer resistance to TKIs, did not alter the regulatory effect of EPN3.

conclusionsEPN3 enhances EGFR signalling by promoting its recycling and stability, contributing to NSCLC progression and TKI resistance. Targeting EPN3 could offer a novel therapeutic strategy to overcome drug resistance in EGFR-driven NSCLC.

Indexed as

EGFREpsin3Non-small cell lung cancerTKI resistance

Identifiers

PMID39910656
PMCPMC11800460

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.