Evidence mapPaperPMID 39985181Full record

ArticleThe international journal of neuropsychopharmacology2025

Synergistic effects of memantine and alpha7 nicotinic acetylcholine receptor agonist PHA-543613 to improve memory of aged rats.

Nóra Bruszt, Zsolt Kristóf Bali, Lili Veronika Nagy, Kornélia Bodó, Péter Engelmann, István Hernádi

Abstract read
In one paragraph

Article in The international journal of neuropsychopharmacology, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 3 papers.

0numbers the graph read from it
0cells of the map it votes in
3citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

3 citing papers in PubMed.

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4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

6 authors.

Nóra BrusztTranslational Neuroscience Research Group, Centre for Neuroscience, Szentágothai Research Centre, University of Pécs, Pécs, Hungary.
Zsolt Kristóf BaliTranslational Neuroscience Research Group, Centre for Neuroscience, Szentágothai Research Centre, University of Pécs, Pécs, Hungary.ORCID 0000-0003-0712-0788
Lili Veronika NagyTranslational Neuroscience Research Group, Centre for Neuroscience, Szentágothai Research Centre, University of Pécs, Pécs, Hungary.
Kornélia BodóDepartment of Immunology and Biotechnology, Medical School, University of Pécs, Pécs, Hungary.
Péter EngelmannDepartment of Immunology and Biotechnology, Medical School, University of Pécs, Pécs, Hungary.
István HernádiTranslational Neuroscience Research Group, Centre for Neuroscience, Szentágothai Research Centre, University of Pécs, Pécs, Hungary.

Funding

Medical School Research Foundation of the University of Pécs KA-2022-03National Research Development and Innovation Fund TKP2021-EGANational Research, Development and Innovation FundNational Research, Development and Innovation Fund of the Hungarian Government TKP2021-EGA-10UNKP-22-3 New National Excellence Program
6 · The paper itself

Abstract

backgroundCombination treatments based on pharmacological interactions at α7 nicotinic acetylcholine receptors (nAChRs) are promising therapeutic approaches for neurocognitive disorders.

methodsHere, we tested the cognitive efficacy of combinations of memantine with an α7 nAChR-selective agonist (PHA-543613) in naturally aged rats. Age-related changes in the expression of some key genes and proteins were also measured using quantitative polymerase chain reaction (PCR) and enzyme-linked immunosorbent assay (ELISA).

resultsAged rats showed marked cognitive decline in the novel object recognition test, and they also exhibited cholinergic changes such as mRNA upregulation of α7 nAChRs. Upregulation of interleukin-1β, macrophage inflammatory protein 1α, CX3CL1, intercellular adhesion molecule 1, and ciliary neurotrophic factor mRNA was also detected in aged rats. Combination treatment of memantine and PHA-543613 successfully alleviated the age-related decline of recognition memory of rats by exceeding the effects of the corresponding monotreatments.

conclusionsResults indicate a positive interaction between memantine and PHA-543613, which also reflects a putative role of α7 nAChRs in the cognitive enhancer effects of memantine. These findings may facilitate the development of combination therapies for age-related neurocognitive disorders.

Indexed as

Agingalpha7 Nicotinic Acetylcholine ReceptorAzabicyclo CompoundsMemantineNicotinic AgonistsNootropic AgentsQuinuclidinesAnimalsDrug SynergismDrug Therapy, CombinationMaleRatsRats, Sprague-DawleyRecognition, Psychologyalpha7 Nicotinic Acetylcholine ReceptorAzabicyclo CompoundsChrna7 protein, ratMemantineNicotinic AgonistsNootropic AgentsQuinuclidinesagingalpha7 nicotinic acetylcholine receptorbehaviorcytokineneurocognitive disorder

Identifiers

PMID39985181
PMCPMC11929953

What Socratic holds

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.