Evidence mapPaperPMID 40214461Full record

ArticleCells2025

Empagliflozin Plays Vasoprotective Role in Spontaneously Hypertensive Rats via Activation of the SIRT1/AMPK Pathway.

Monika Kloza, Anna Krzyżewska, Hanna Kozłowska, Sandra Budziak, Marta Baranowska-Kuczko

Abstract read
In one paragraph

Article in Cells, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 5 papers.

0numbers the graph read from it
0cells of the map it votes in
5citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

5 citing papers in PubMed.

  1. Article
  2. Article
  3. Review
  4. Review
  5. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

5 authors.

Monika KlozaDepartment of Experimental Physiology and Pathophysiology, Medical University of Białystok, 15-222 Białystok, Poland.ORCID 0000-0001-7374-0999
Anna KrzyżewskaDepartment of Experimental Physiology and Pathophysiology, Medical University of Białystok, 15-222 Białystok, Poland.ORCID 0000-0001-5986-3757
Hanna KozłowskaDepartment of Experimental Physiology and Pathophysiology, Medical University of Białystok, 15-222 Białystok, Poland.ORCID 0000-0002-2105-3350
Sandra BudziakDepartment of Experimental Physiology and Pathophysiology, Medical University of Białystok, 15-222 Białystok, Poland.ORCID 0009-0001-1794-9947
Marta Baranowska-KuczkoDepartment of Experimental Physiology and Pathophysiology, Medical University of Białystok, 15-222 Białystok, Poland.ORCID 0000-0002-7238-2656

Funding

National Science Center NCN/1/MI/22/001/2213
6 · The paper itself

Abstract

Empagliflozin (EMPA), a sodium-glucose co-transporter 2 (SGLT2) inhibitor, prevents endothelial dysfunction, but its effects on vascular tone in hypertension remain unclear. This study investigated whether EMPA modulates vasomotor tone via sirtuin 1 (SIRT1) and AMP-activated protein kinase (AMPK) pathways in spontaneously hypertensive rats (SHR) and controls (Wistar Kyoto rats, WKY). Functional (wire myography, organ bath) and biochemical (Western blot) studies were conducted on the third-order of the superior mesenteric arteries (sMAs) and/or aortas. EMPA induced concentration-dependent relaxation of preconstricted sMAs in both groups. In SHR, EMPA enhanced acetylcholine (Ach)-induced relaxation in sMAs and aortas and reduced constriction induced by phenylephrine (Phe) and U46619 in sMAs. The SIRT1 inhibitor (EX527) abolished EMPA's effects on Ach-mediated relaxation and U46619-induced vasoconstriction, while AMPK inhibition reduced Ach-mediated relaxation and Phe-induced vasoconstriction. SHR showed increased SGLT2 and SIRT1 expression and decreased pAMPK/AMPK levels in sMAs. In conclusion, EMPA might exert vasoprotective effects in hypertension by enhancing endothelium-dependent relaxation and reducing constriction via AMPK/SIRT1 pathways. These properties could improve vascular health in patients with hypertension and related conditions. Further studies are needed to explore new indications for SGLT2 inhibitors.

Indexed as

AMP-Activated Protein KinasesBenzhydryl CompoundsGlucosidesHypertensionSignal TransductionSirtuin 1AnimalsAortaMaleMesenteric Artery, SuperiorPhenylephrineRatsRats, Inbred SHRRats, Inbred WKYSodium-Glucose Transporter 2 InhibitorsVasoconstrictionAMP-Activated Protein KinasesBenzhydryl CompoundsempagliflozinGlucosidesPhenylephrineSirt1 protein, ratSirtuin 1Sodium-Glucose Transporter 2 InhibitorsAMPKempagliflozinSGLT2 inhibitorssirtuin 1spontaneously hypertensive ratvasoprotection

Identifiers

PMID40214461
PMCPMC11987869

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.