Evidence mapPaperPMID 40216698Full record

ArticleCell biochemistry and biophysics2025

The Impact of Liraglutide, a GLP-1 Receptor Agonist, on High Glucose-Induced Inflammation, Apoptosis, Oxidative Stress, and NLRP3 Signaling.

Mustafa Gokce, Dilek Ozturk Civelek, Aylin Vidin Sen, Eray Metin Guler, Erkan Civelek, Birsel Sonmez Uydes Dogan, F Ilkay Alp Yildirim

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Article in Cell biochemistry and biophysics, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 3 papers.

0numbers the graph read from it
0cells of the map it votes in
3citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

3 citing papers in PubMed.

  1. Review
  2. Article
  3. Review
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

7 authors.

Mustafa GokceIstanbul University, Faculty of Pharmacy, Department of Pharmacology, Istanbul, Turkey.
Dilek Ozturk CivelekBezmialem Vakif University, Faculty of Pharmacy, Department of Pharmacology, Istanbul, Turkey.
Aylin Vidin SenIstanbul University, Faculty of Pharmacy, Department of Pharmacology, Istanbul, Turkey.
Eray Metin GulerHealth Sciences University, Hamidiye Medical School, Department of Medical Biochemistry, Istanbul, Turkey.
Erkan CivelekIstanbul University, Faculty of Pharmacy, Department of Pharmacology, Istanbul, Turkey.
Birsel Sonmez Uydes DoganIstanbul University, Faculty of Pharmacy, Department of Pharmacology, Istanbul, Turkey.
F Ilkay Alp YildirimIstanbul University, Faculty of Pharmacy, Department of Pharmacology, Istanbul, Turkey. ilkayalp@istanbul.edu.tr.

Funding

Bezmialem Vakif University BAP unit 20220203Istanbul University BAP unit TSA-2022-38649TUBITAK 1002-Rapid Support Program 720075
6 · The paper itself

Abstract

Diabetes-related endothelial dysfunction, alteration in cell signaling, increased oxidative stress and activation of pro-inflammatory processes are the main causes of diabetes-related vascular complications. Glucagon-like peptide-1 (GLP-1) and its receptor (GLP-1R) play a crucial role in regulating glucose homeostasis, insulin secretion, and reducing inflammation. GLP-1R agonists have been explored for their potential in mitigating diabetes-related vascular dysfunction. The NOD-like receptor protein 3 (NLRP3) inflammasome, a key protein complex in immune response, activates caspase-1 and promotes proinflammatory cytokine secretion. High glucose levels activate NLRP3 in macrophages via reactive oxygen species and mitochondrial dysfunction. This study aims to investigate the effects of GLP-1 receptor agonist, Liraglutide, on cell proliferation, inflammation, oxidative stress and NLRP3-related signaling pathways in human umbilical vein endothelial cells (HUVEC) and human coronary artery endothelial cell (HCAEC) cultures. HUVEC and HCAEC were incubated with Liraglutide (10 and 100 nM, 48 h) either in normoglycemic (5.5 mM) or hyperglycemic (25 mM) condition. Cell proliferation, oxidative stress, mRNA and protein expressions of ASC, caspase-1, NLRP3 which are. components of NLRP3 inflammasome, were determined. Our results showed that, Liraglutide significantly reduced hyperglycemia-induced oxidative stress, mRNA and protein expressions of NLRP3 inflammasome and proinflammatory cytokine levels, as well as cell membrane damage in HUVEC and HCAEC. Our results indicate that Liraglutide may have the potential on preventing hyperglycemia-induced cellular damage by reducing inflammation and immune response activation both in human venous and arterial endothelial cells.

Indexed as

ApoptosisGlucagon-Like Peptide-1 Receptor AgonistsGlucoseLiraglutideNLR Family, Pyrin Domain-Containing 3 ProteinOxidative StressSignal TransductionCell ProliferationGlucagon-Like Peptide-1 ReceptorHumansHuman Umbilical Vein Endothelial CellsInflammasomesInflammationReactive Oxygen SpeciesGlucagon-Like Peptide-1 ReceptorGlucagon-Like Peptide-1 Receptor AgonistsGlucoseInflammasomesLiraglutideNLR Family, Pyrin Domain-Containing 3 ProteinNLRP3 protein, humanReactive Oxygen SpeciesEndothelial dysfunctionHyperglycemiaInflammationLiraglutideNLRP3

Identifiers

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.