Evidence mapPaperPMID 40243772Full record

ArticleInternational journal of molecular sciences2025

Neuroprotective Effects of Cilomilast and Chlorogenic Acid Against Scopolamine-Induced Memory Deficits via Modulation of the cAMP/PKA-CREB-BDNF Pathway.

Esraa M Mosalam, Soha M Atya, Noha M Mesbah, Shady Allam, Eman T Mehanna

Abstract read
In one paragraph

Article in International journal of molecular sciences, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 10 papers.

0numbers the graph read from it
0cells of the map it votes in
10citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

10 citing papers in PubMed.

  1. Article
  2. Review
  3. Article
  4. Article
  5. Article
  6. Article
  7. Article
  8. Article
  9. Oral Supplementation withNutrients · 2025
    Article
  10. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

5 authors.

Esraa M MosalamBiochemistry Department, Faculty of Pharmacy, Menoufia University, Shebin EL-Kom 32511, Menoufia, Egypt.ORCID 0000-0003-4630-4125
Soha M AtyaDepartment of Biochemistry, Faculty of Pharmacy, Suez Canal University, Ismailia 41522, Ismailia, Egypt.ORCID 0009-0004-1083-1315
Noha M MesbahDepartment of Biochemistry, Faculty of Pharmacy, Suez Canal University, Ismailia 41522, Ismailia, Egypt.ORCID 0000-0002-8863-968X
Shady AllamDepartment of Pharmacology and Toxicology, Faculty of Pharmacy, Menoufia University, Shebin EL-Kom 32511, Menoufia, Egypt.ORCID 0000-0002-5633-4128
Eman T MehannaDepartment of Biochemistry, Faculty of Pharmacy, Suez Canal University, Ismailia 41522, Ismailia, Egypt.ORCID 0000-0003-2759-2889

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Alzheimer's disease (AD) is a neurodegenerative disorder characterized by cognitive decline, neuroinflammation and neuronal damage. This study aimed to investigate the neuroprotective effects of cilomilast (CILO), a phosphodiesterase-4 (PDE4) inhibitor, alone and in combination with chlorogenic acid (CGA), a natural polyphenol, against scopolamine (SCOP)-induced cognitive impairment in mice. Forty male albino mice were divided into five groups: normal control, SCOP control, CGA + SCOP, CILO + SCOP and CILO + CGA + SCOP. Behavioral assessments, including the Y-maze and pole climbing tests, demonstrated that SCOP significantly impaired cognition, while treatment with CILO and CGA reversed these deficits, with the combination group showing the greatest improvement. Histopathological analyses revealed that CILO and CGA reduced neuronal damage and amyloid beta (Aβ) accumulation. Immunohistochemical and biochemical assessments confirmed a decrease in neuroinflammatory markers, including tumor necrosis factor-alpha (TNF-α) and nuclear factor kappa B (NF-κB). Molecular analyses showed that CILO restored cyclic adenosine monophosphate (cAMP) levels, leading to activation of protein kinase A (PKA), cAMP response element-binding protein (CREB) and brain-derived neurotrophic factor (BDNF), key regulators of neuronal plasticity and survival. CGA enhanced these effects by further inhibiting PDE4, amplifying the neuroprotective response. These findings suggest that PDE4 inhibitors, particularly in combination with CGA, may represent promising therapeutic strategies for AD-related cognitive impairment.

Indexed as

Chlorogenic AcidMemory DisordersNeuroprotective AgentsSignal TransductionAnimalsBrain-Derived Neurotrophic FactorCyclic AMPCyclic AMP-Dependent Protein KinasesCyclic AMP Response Element-Binding ProteinDisease Models, AnimalMaleMicePhosphodiesterase 4 InhibitorsScopolamineBdnf protein, mouseBrain-Derived Neurotrophic FactorChlorogenic AcidCreb1 protein, mouseCyclic AMPCyclic AMP-Dependent Protein KinasesCyclic AMP Response Element-Binding ProteinNeuroprotective AgentsPhosphodiesterase 4 InhibitorsScopolamineAlzheimer’scAMP/PKA–CREB–BDNF pathwaychlorogenic acidcilomilastneuroinflammationphosphodiesterase 4

Identifiers

PMID40243772
PMCPMC11988773

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.