Evidence map›Paper›PMID 40406932›Full record

ArticleCNS neuroscience & therapeutics2025

Ligustrazine Alleviates Blood-Brain Barrier Damage by Downregulating Expression of miR-297c-5p.

Shaoyu Guan, Ruichen Jiang, Xudong Wang, Tong Chen, Ping Yi, Tian Li, Teng Ma, Fang Wang

Abstract read
In one paragraph

Article in CNS neuroscience & therapeutics, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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0citing papers in PubMed
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1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

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Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

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PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

8 authors.

Shaoyu GuanPharmaceutical Sciences Research Division, Department of Pharmacy, Medical Supplies Centre of PLA General Hospital/Medical School of Chinese PLA, Beijing, China.
Ruichen JiangDepartment of Clinical Medicine, Beijing University of Chinese Medicine, Beijing, China.
Xudong WangDepartment of Dermatology, The Seventh Medical Center of Chinese PLA General Hospital/Medical School of Chinese PLA, Beijing, China.
Tong ChenDepartment of Cardiology, The Sixth Medical Centre, Chinese PLA General Hospital/Medical School of Chinese PLA, Beijing, China.
Ping YiDepartment of Orthopaedics, China-Japan Friendship Hospital, Beijing, China.
Tian LiTianjin Key Laboratory of Acute Abdomen Disease-Associated Organ Injury and ITCWM Repair, Institute of Integrative Medicine of Acute Abdominal Diseases, Tianjin Nankai Hospital, Tianjin Medical University, Tianjin, China.ORCID 0000-0002-8281-4459
Teng MaDepartment of Trauma Orthopedics, General Hospital of Ningxia Medical University, Yinchuan, China.
Fang WangMedical Imaging Center of People's Hospital of Ningxia Hui Autonomous Region/Ningxia Medical University, Yinchuan, China.

Funding

2022 Ningxia Hui Autonomous Region Natural Science Foundation (General) Project 2022AAC03390
6 · The paper itself

Abstract

objectiveLigustrazine (LSZ), an ingredient of Ligusticum chuanxiong, has long been used to treat neurovascular diseases in China. This study investigates its protective effects for the impairment of the blood-brain barrier (BBB) and the underlying mechanisms.

methodsIn this study, the impacts of LSZ on the BBB function were firstly assessed in b. End3 cells in vitro. Oxygen-glucose deprivation (OGD) served as an injury factor and western blot (WB) analyzed the expressions of occludin and ZO-1, two tight junction proteins (TJs), essential for maintaining the integrity of the BBB. After bioinformatics analysis of the transcriptome in vivo, qRT-PCR of miR-297c-5p was conducted and a dual-luciferase reporter assay was used to verify the target protein, occludin, which was confirmed by hippocampal insertion using guide cannulas and microinfection of RNA oligos.

resultsA 3-h deprivation of OGD of b. End3 cells resulted in noticeable reductions in the level of occludin and ZO-1. However, administration of LSZ (0.1 μM) effectively restored these decreases. In normal mice, administration of LSZ (25 mg/kg, i.p., once daily for 9 days) resulted in a notable reduction in miR-297c-5p. In the middle cerebral artery occlusion (MCAO) mouse model, increased miR-297c-5p was also reversed by LSZ administration. Bioinformatics analysis revealed one of the targets of miR-297c-5p includes occludin. MiR-297c-5p was found to directly target occludin in the dual-luciferase reporter assay. Transfection of miR-297c-5p agomir into b. End3 cells resulted in a significant reduction in the level of occludin, while transfection of antagomir led to an increase in occludin. Besides, stereotaxic injection of AAV-miR-297c-5p into the hippocampus reduced occludin level in vivo. Ultimately, hippocampal microinfection of RNA oligos provided a confirmation that miR-297c-5p was downregulated by LSZ in MCAO mice with up-regulated occludin expression.

conclusionIn conclusion, the present findings provide new insights into regulating occludin by LSZ through downregulation of miR-297c-5p.

Indexed as

Blood-Brain BarrierDown-RegulationMicroRNAsNeuroprotective AgentsPyrazinesAnimalsCell HypoxiaGlucoseMaleMiceMice, Inbred C57BLOccludinZonula Occludens-1 ProteinGlucoseMicroRNAsNeuroprotective AgentsOccludinPyrazinestetramethylpyrazineZonula Occludens-1 Proteinblood–brain barrierligustrazinemiR‐297c‐5ptight junction

Identifiers

PMID40406932
PMCPMC12099305

What Socratic holds

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.