Evidence mapPaperPMID 40453214Full record

ArticleDrug design, development and therapy2025

A Novel Flavonoid Derivative of Icariside II (YS-10) Improves Erectile Dysfunction in a Diabetic Rat Model by Inhibiting Ferroptosis via Activation of the Nrf2/HO-1/GPX4 Pathway.

Yang Liu, Guan-Nan Liu, Ya-Rong Zha, Chen-Li Pan, Yong-de Xu, Hong-Wei Li, Yue-Yue Zang, Wan-Qi Wang, Jun-Jie Yao, Jun-Tao Sun and 2 more

Abstract read
In one paragraph

Article in Drug design, development and therapy, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 2 papers.

0numbers the graph read from it
0cells of the map it votes in
2citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

2 citing papers in PubMed.

  1. Article
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4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

12 authors.

Yang LiuChangchun University of Chinese Medicine, Changchun, Jilin Province, People's Republic of China.ORCID 0000-0002-4702-5809
Guan-Nan LiuChangchun University of Chinese Medicine, Changchun, Jilin Province, People's Republic of China.
Ya-Rong ZhaChangchun University of Chinese Medicine, Changchun, Jilin Province, People's Republic of China.
Chen-Li PanChangchun University of Chinese Medicine, Changchun, Jilin Province, People's Republic of China.
Yong-de XuDepartment of Urology, Beijing Friendship Hospital, Capital Medical University, Beijing, 100050, People's Republic of China.
Hong-Wei LiChangchun University of Chinese Medicine, Changchun, Jilin Province, People's Republic of China.
Yue-Yue ZangChangchun University of Chinese Medicine, Changchun, Jilin Province, People's Republic of China.
Wan-Qi WangChangchun University of Chinese Medicine, Changchun, Jilin Province, People's Republic of China.
Jun-Jie YaoChangchun University of Chinese Medicine, Changchun, Jilin Province, People's Republic of China.
Jun-Tao SunChangchun University of Chinese Medicine, Changchun, Jilin Province, People's Republic of China.
Yong YangDepartment of Urology, The Affiliated Hospital of Changchun University of Chinese Medicine, Changchun, Jilin Province, People's Republic of China.ORCID 0000-0002-2907-3030
Zhi-Tao WeiDepartment of Urology, The Affiliated Hospital of Changchun University of Chinese Medicine, Changchun, Jilin Province, People's Republic of China.ORCID 0000-0002-1285-9328

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Objective: This study aimed to evaluate the therapeutic potential of YS-10, a novel flavonoid derivative of icariside II (ICA II), and to explore its mechanism of action in a diabetic rat model of erectile dysfunction (DMED). Methods: Twenty-four male Sprague-Dawley rats were divided into four groups: control, DMED, DMED + ICA II (2.5 mg/kg/day), and DMED + YS-10 (2.5 mg/kg/day). Treatments lasted for 4 weeks followed by a 3-day washout. Erectile function was assessed, and penile tissues were analyzed by histology, immunohistochemistry, ELISA, and Western blot. In vitro, primary corpus cavernosum endothelial cells (CCECs) were treated with advanced glycation end products (AGEs), YS-10, Fer-1 (ferroptosis inhibitor), or ML385 (Nrf2 inhibitor) to evaluate oxidative stress and ferroptosis. Results: In vivo, both YS-10 and ICA II (2.5 mg/kg/day) significantly improved erectile function in diabetic rats, increased smooth muscle content, reduced collagen deposition, and enhanced endothelial marker (CD31) expression in penile tissue ( Conclusion: YS-10 improves erectile function in diabetic rats by reducing oxidative stress and inhibiting ferroptosis via activation of the Nrf2/HO-1/GPX4 pathway. At 2.5 mg/kg/day, YS-10 was effective, well-tolerated, and showed efficacy comparable to ICA II. These findings support its potential as a promising candidate for diabetes-related erectile dysfunction therapy.

Indexed as

Diabetes Mellitus, ExperimentalErectile DysfunctionFerroptosisFlavonoidsAnimalsCells, CulturedDisease Models, AnimalDose-Response Relationship, DrugHeme Oxygenase-1Heme Oxygenase (Decyclizing)MaleMolecular StructureNF-E2-Related Factor 2Oxidative StressPhospholipid Hydroperoxide Glutathione PeroxidaseRatsbaohuoside IFlavonoidsglutathione peroxidase 4, ratHeme Oxygenase-1Heme Oxygenase (Decyclizing)Hmox1 protein, ratNfe2l2 protein, ratNF-E2-Related Factor 2Phospholipid Hydroperoxide Glutathione PeroxidaseStreptozocindiabetes mellituserectile dysfunctionferroptosisGPX4ICA IINrf2YS-10

Identifiers

PMID40453214
PMCPMC12126984

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.