Evidence mapPaperPMID 40468373Full record

ArticleBMC complementary medicine and therapies2025

Integrative investigation on Hippocratea africana root: insights from cardio-protective, anti-oxidative stress activities, isolation, GC/MS, and pharmacological significance profiling.

Edet Effiong Asanga, Kufre Uyo Noah, Jude Efiom Okokon, Chinedum Martins Ekeleme, Imaobong Etima Udoh, Augustine Bassey, Martin Osita Anagboso, Aniekeme Ndisa Inyang

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Article in BMC complementary medicine and therapies, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 1 paper.

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0cells of the map it votes in
1citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

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The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

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3 · Its place in the literature

Who cites it

1 citing paper in PubMed.

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4 · The record

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5 · Who and what money

Authors and funding

8 authors.

Edet Effiong AsangaDepartment of Biochemistry, Arthur Jarvis University, Akpabuyo, Cross River State, Nigeria. edyasangae1@gmail.com.
Kufre Uyo NoahDepartment of Pharmacology and Toxicology, University of Uyo, Uyo, Akwa Ibom State, Nigeria.
Jude Efiom OkokonDepartment of Pharmacology and Toxicology, University of Uyo, Uyo, Akwa Ibom State, Nigeria.
Chinedum Martins EkelemeDepartment of Biochemistry, Delta State University of Science and Technology, Ozoro, Delta State, Nigeria.
Imaobong Etima UdohDepartment of Zoology and Environmental Biology, University of Calabar, Calabar, Cross River State, Nigeria.
Augustine BasseyDepartment of Clinical Pharmacology and Therapeutics, University of Uyo, Uyo, Akwa Ibom State, Nigeria.
Martin Osita AnagbosoDepartment of Microbiology, Madonna University Nigeria, Elele Campus, PortHarcourt, Rivers State, Nigeria.
Aniekeme Ndisa InyangDepartment of Biochemistry, Arthur Jarvis University, Akpabuyo, Cross River State, Nigeria.

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

backgroundHippocratea africana root is scientifically used in cardiotoxicity treatment; therefore, this study was designed to validate this claims through the evaluation of its cardioprotective activity, isolation, and characterization of its constituents, as well as in silico profiling of these ligands against antioxidant enzymes.

methodsStandard protocols were followed in the extraction, fractionation, isolation, characterization, evaluation of cardio-protective activity (marker enzymes, oxidative stress markers, and histological section), retrieval of target proteins (SOD, CAT, GPx, and GSH), ADMET, and docking studies. Column and thin layer chromatography as well as GC/MS aided the isolation and characterization of compounds; SWISSADME and ADMET lab 2 enhanced the evaluation of pharmacokinetic properties; PyRx for docking analysis; Biovia discovery studio and PyMol software for 2D and 3D visualization of the ligand-protein interactions.

resultsThe root extract administration significantly (p < 0.05) reduced the serum levels of CK-MB, LDH, and troponin I that were elevated after doxorubicin administration; however, the levels of GSH, GST, SOD, GPx, and CAT that were decreased after doxorubicin administration were significantly (p < 0.05) elevated whereas the raised MDA level was reduced after treatment with the extract and fractions of the plant. Also, the histological sections in the extract-treated rats showed reductions in pathological features as compared with the negative control group. Moreover, the chemical pathological changes were consistent with histopathological observations suggesting marked cardio-protective potentials. Furthermore, the chromatographic analyses yielded bulked fractions {D3 (11 mg), E6 (25 mg), and E8 (21 mg)} and their GC/MS analyses revealed dihydroartemisinin; retinoic acid, methyl ester; α-thujene; α-terpinolene; 9,12,15-octadecatrienal; α-terpineol etc. with already reported antioxidant activities. These ligands (dihydroartemisinin; retinoic acid, methyl ester) obeyed Lipinski's criteria, had remarkable pharmacokinetic profiles, and their docking analyses revealed that they modulated antioxidant enzymes with better binding affinities than vitamin C.

conclusionGiven the demonstrated antidotal and cardioprotective properties of the plant root, it presents a promising candidate for mitigating doxorubicin-induced toxicities and could be effectively utilized as a supportive therapy in such contexts.

Indexed as

AntioxidantsCardiotonic AgentsOxidative StressPlant ExtractsAnimalsDoxorubicinGas Chromatography-Mass SpectrometryMaleMolecular Docking SimulationPlant RootsRatsRats, WistarAntioxidantsCardiotonic AgentsDoxorubicinPlant ExtractsADMETAntioxidantCardioprotectiveChromatographyGC/MSHippocratea africanaMolecular dockingOxidative stress

Identifiers

PMID40468373
PMCPMC12135251

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.