Evidence mapPaperPMID 40476344Full record

ArticleJournal of neurochemistry2025

Multi-Omic Analysis of Glutamate Excitotoxicity in Primary Neuronal Cultures.

Jennifer H Nguyen, Xiaolu Zhang, Hunter M Eby, Khaled Alganem, William G Ryan, Ali Sajid Lmami, Anna E Lundh, Anvitha R Madhavaram, James D Bretz, Ethel Tackie-Yarboi and 4 more

Abstract read
In one paragraph

Article in Journal of neurochemistry, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 2 papers.

0numbers the graph read from it
0cells of the map it votes in
2citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

2 citing papers in PubMed.

  1. Trial
  2. Review
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

14 authors.

Jennifer H NguyenDepartment of Neurosciences and Psychiatry, University of Toledo, Toledo, Ohio, USA.ORCID https://orcid.org/0009-0008-8708-0117
Xiaolu ZhangDepartment of Neurosciences and Psychiatry, University of Toledo, Toledo, Ohio, USA.
Hunter M EbyDepartment of Neurosciences and Psychiatry, University of Toledo, Toledo, Ohio, USA.
Khaled AlganemDepartment of Neurosciences and Psychiatry, University of Toledo, Toledo, Ohio, USA.
William G RyanDepartment of Neurosciences and Psychiatry, University of Toledo, Toledo, Ohio, USA.
Ali Sajid LmamiDepartment of Neurosciences and Psychiatry, University of Toledo, Toledo, Ohio, USA.
Anna E LundhDepartment of Neurosciences and Psychiatry, University of Toledo, Toledo, Ohio, USA.
Anvitha R MadhavaramDepartment of Medicinal and Biological Chemistry, University of Toledo, Toledo, Ohio, USA.
James D BretzDepartment of Medical Microbiology and Immunology, University of Toledo, Toledo, Ohio, USA.
Ethel Tackie-YarboiDepartment of Medicinal and Biological Chemistry, University of Toledo, Toledo, Ohio, USA.
Kelsee ZajacDepartment of Medicinal and Biological Chemistry, University of Toledo, Toledo, Ohio, USA.
William S MesserDepartment of Medicinal and Biological Chemistry, University of Toledo, Toledo, Ohio, USA.
Isaac T SchieferDepartment of Medicinal and Biological Chemistry, University of Toledo, Toledo, Ohio, USA.
Robert E McCullumsmithDepartment of Neurosciences and Psychiatry, University of Toledo, Toledo, Ohio, USA.

Funding

Translational assessment of brain bioenergetic function in schizophreniaR01MH121102 · NIMH · UNIVERSITY OF MARYLAND BALTIMORE · PI Christopher Marano, Robert E McCullumsmith · 2021 to 2024
$2.9M
Cross platform analysis of drug targets and toxicity of bath saltsU01DA054330 · UNIVERSITY OF TOLEDO HEALTH SCI CAMPUS · 2025 to 2025
$556k
Development of Attenuated Furoxans as Novel Therapies for Alzheimer's DiseaseR01AG057598 · NIA · UNIVERSITY OF TOLEDO HEALTH SCI CAMPUS · PI Isaac T Schiefer · 2022 to 2022
$386k
NIA NIH HHS AG057598NIA NIH HHS R01 AG057598NIDA NIH HHS U01 DA054330NIMH NIH HHS MH107487NIMH NIH HHS MH121102NIMH NIH HHS R01 MH107487NIMH NIH HHS R01 MH121102
6 · The paper itself

Abstract

Glutamate excitotoxicity plays a critical role in neurodegeneration by triggering NMDA receptor hyperactivation, leading to elevated synaptic calcium levels and subsequent neuronal death. To better understand how glutamate affects neurons in neurological diseases, we conducted a comprehensive analysis of molecular changes at the transcriptome and kinome levels. We used primary cortical cultures from rat embryos to study glutamate-induced excitotoxicity. Intermediate doses of glutamate (250 μM) produced significant neurotoxic effects, whereas high and low doses resulted in less cell mortality, aligning with previous findings related to calcium influx. Transcriptional analysis identified BTG2, NPAS4, and CCN1 as the most significantly differentially expressed genes following 250 μM glutamate treatment in neurons. Dkk2, a Wnt antagonist, exhibited the highest log fold change among the significantly differentially expressed genes. Gene set enrichment analysis identified 1127 significant pathways. Perturbagen analysis revealed 2811 unique concordant signatures and 1071 unique discordant signatures. Kinome array profiling indicated activation of PKA and PKG kinases, which regulate signaling pathways essential for synaptic plasticity-related gene expression. Multi-omic integration of transcriptome and kinome data revealed enrichment of response to oxidative stress, actin filament organization, and regulation of apoptotic processes pathways. The Wnt signaling pathway emerged as a pivotal factor in the early stages of axon differentiation and growth, as well as in shaping axonal behavior and dendrite development. Moreover, the interplay between MAPK and Wnt signaling pathways likely impacts cellular differentiation processes. Our findings highlight a prominent role for p38/MAPK and stress-activated MAPK pathways, with specific activation of the MAPK/ERK signaling pathway in response to excitotoxic neuronal damage in vitro. In conclusion, glutamate excitotoxicity induces molecular changes at the transcriptome and kinome levels that include elements of the MAPK and WNT biological pathways.

Indexed as

Glutamic AcidNeuronsAnimalsCells, CulturedMultiomicsRatsRats, Sprague-DawleyTranscriptomeGlutamic Acidglutamate excitotoxicitykinomicsMAPK signalingmultiomicstranscriptomics

Identifiers

PMID40476344
PMCPMC12142573

What Socratic holds

Textmetadata
LicenceCC BY-NC-ND
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.