Evidence mapPaperPMID 40660408Full record

ArticleAlzheimer's research & therapy2025

The efficacy and pharmacological mechanism of Guilingji to prevent Alzheimer's disease.

Fengrui Hu, Yaling Lei, Rui Han, Bo Yang, Yanlin Liang, Jing Luan, Bei Zhang, Shan Wang, Xingchun Gou

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Article in Alzheimer's research & therapy, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 1 paper.

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0cells of the map it votes in
1citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

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2 · The registry

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3 · Its place in the literature

Who cites it

1 citing paper in PubMed.

  1. Review
4 · The record

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5 · Who and what money

Authors and funding

9 authors.

Fengrui Hu *Shaanxi Key Laboratory of Brain Disorders & Institute of Basic and Translational Medicine, Xi'an Medical University, Xi'an, 710021, China.
Yaling Lei *Shaanxi Provincial Hospital of Traditional Chinese Medicine, Xi'an, 710003, China.
Rui Han *Shaanxi Key Laboratory of Brain Disorders & Institute of Basic and Translational Medicine, Xi'an Medical University, Xi'an, 710021, China.
Bo YangShanxi Guangyuyuan Sinopharm Co., Ltd., Jinzhong, 030800, China.
Yanlin LiangShanxi Guangyuyuan Sinopharm Co., Ltd., Jinzhong, 030800, China.
Jing LuanShaanxi Key Laboratory of Brain Disorders & Institute of Basic and Translational Medicine, Xi'an Medical University, Xi'an, 710021, China.
Bei ZhangDepartment of Neurology, The First Affiliated Hospital of Xi'an Medical University, Xi'an, 710077, China.
Shan WangShaanxi Key Laboratory of Brain Disorders & Institute of Basic and Translational Medicine, Xi'an Medical University, Xi'an, 710021, China. wangshan_jzs@xiyi.edu.cn.
Xingchun GouShaanxi Key Laboratory of Brain Disorders & Institute of Basic and Translational Medicine, Xi'an Medical University, Xi'an, 710021, China. go@xiyi.edu.cn.

Funding

National Natural Science Foundation of China NO.82201599Natural Science Basic Research Program of Shaanxi Province 2022JQ-814Scientific Research Program Funded by Education Department of Shaanxi Provincial Government NO.23JK0654
6 · The paper itself

Abstract

backgroundEffective treatments for Alzheimer's disease (AD) are limited, so preventing or delaying its onset is crucial. Previous clinical trials have shown the safety and potential efficacy of the Chinese herbal formula Guilingji (GLJ), but its preventive effect on AD and mechanism are still unclear.

methodsIn this study, a network pharmacology approach was employed to elucidate the mechanism of GLJ in AD. Behavioral assessments and biochemical experiments were conducted on APPswe/PS1ΔE9 transgenic (APP/PS1) mice. The pivotal pathways and biological processes were validated in vitro AD model using HT22 and BV-2 cells stimulated by Aβ1-42. Additionally, molecular docking was utilized to illustrate the binding affinity of GLJ's active components to key genes implicated in AD prevention.

resultsNetwork pharmacology analysis identified 482 common targets associated with the active components of GLJ. KEGG enrichment analysis highlighted the PI3K-AKT and retrograde endocannabinoid signaling pathways as the key mechanisms. GLJ significantly postponed cognitive decline, suppressed Aβ plaque accumulation, mitigated neuronal damage, and reduced inflammatory responses in glial cells in AD mice. GLJ and its compounds quercetin and carvone assist in neuron survival by regulating the PI3K/AKT pathway and the apoptotic proteins Bcl-2 and Bax. Additionally, GLJ, kaempferol and stigmasterol enhance microglial clearance of Aβ through the CB2 receptor. Moreover, molecular docking suggested that quercetin and carvone interacted effectively with PI3K, while kaempferol and stigmasterol combined well with CB2.

conclusionsGLJ effectively delays AD progression by modulating critical pathological pathways such as neuronal survival, neuroinflammation, and Aβ clearance through a synergistic multi-target approach, offering a promising avenue for AD prevention.

Indexed as

Alzheimer DiseaseDrugs, Chinese HerbalAmyloid beta-PeptidesAnimalsDisease Models, AnimalHumansMaleMiceMice, TransgenicMolecular Docking SimulationNetwork PharmacologyPeptide FragmentsSignal TransductionAmyloid beta-PeptidesDrugs, Chinese HerbalPeptide FragmentsAlzheimer’s diseaseAβ neurotoxicityGuilingjiMicroglia phagocytosisNeuronal damage

Identifiers

PMID40660408
PMCPMC12257861

What Socratic holds

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.