Evidence mapPaperPMID 40667753Full record

ArticleFuture medicinal chemistry2025

Design and synthesis of novel quinoline-piperazines fused to a phenylhydrazinecarbothioamide scaffold as promising α-glucosidase inhibitors with anti-diabetic potential.

Mehran Ghasemi, Fateme Bagheri, Fatemeh Sadat Khajeh Mohammadilar, Aida Iraji, Vahid Lotfi, Reza Karimi, Maryam Dehghan, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Mohammad Mahdavi and 1 more

Abstract read
In one paragraph

Article in Future medicinal chemistry, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

11 authors.

Mehran GhasemiNatural and Medical Sciences Research Center, University of Nizwa, Nizwa, Oman.
Fateme BagheriStem Cells Technology Research Center, Shiraz University of Medical Sciences, Shiraz, Iran.
Fatemeh Sadat Khajeh MohammadilarEndocrinology and Metabolism Research Center, Endocrinology and Metabolism Clinical Sciences Institute, Tehran University of Medical Sciences, Tehran, Iran.
Aida IrajiStem Cells Technology Research Center, Shiraz University of Medical Sciences, Shiraz, Iran.
Vahid LotfiEndocrinology and Metabolism Research Center, Endocrinology and Metabolism Clinical Sciences Institute, Tehran University of Medical Sciences, Tehran, Iran.
Reza KarimiSchool of Chemistry, College of Science, University of Tehran, Tehran, Iran.
Maryam DehghanSchool of Chemistry, College of Science, University of Tehran, Tehran, Iran.
Somayeh MojtabaviDepartment of Pharmaceutical Biotechnology, Faculty of Pharmacy, Tehran University of Medical Sciences, Tehran, Iran.
Mohammad Ali FaramarziDepartment of Pharmaceutical Biotechnology, Faculty of Pharmacy, Tehran University of Medical Sciences, Tehran, Iran.
Mohammad MahdaviEndocrinology and Metabolism Research Center, Endocrinology and Metabolism Clinical Sciences Institute, Tehran University of Medical Sciences, Tehran, Iran.
Ahmed Al-HarrasiNatural and Medical Sciences Research Center, University of Nizwa, Nizwa, Oman.

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

aimsThis study focused on the design, synthesis, and dual MATERIALS &

methodsA series of quinoline-benzoylhydrazine compounds were synthesized and evaluated as α-glucosidase inhibitors. The most active compound was subjected to the kinetic study plus molecular docking and molecular dynamics simulations to elucidate the mechanism of inhibition and stability.

resultsAll synthesized compounds exhibited strong α-glucosidase inhibition. Among them,

conclusionThe results confirm that quinoline-piperazine derivatives bearing phenylhydrazinecarbothioamide moieties are promising scaffolds for α-glucosidase inhibition.

Indexed as

alpha-GlucosidasesDrug DesignGlycoside Hydrolase InhibitorsHydrazinesHypoglycemic AgentsPiperazinesQuinolinesThioamidesHumansMolecular Docking SimulationMolecular Dynamics SimulationMolecular StructureStructure-Activity Relationshipalpha-GlucosidasesGlycoside Hydrolase InhibitorsHydrazinesHypoglycemic AgentsPiperazinesQuinolinesThioamidesDiabetes mellitusMolecular dynamics simulationPiperazineQuinolineα-glucosidase

Identifiers

PMID40667753
PMCPMC12279276

What Socratic holds

Textmetadata
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.