Evidence map›Paper›PMID 40705771›Full record

ArticleJournal of medicinal chemistry2025

Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution.

Tania Ciaglia, Valeria Napolitano, Maria Rosaria Miranda, Danila La Gioia, Simona Musella, Aniello Schiano Moriello, Fabrizio Merciai, Veronica Di Sarno, Simona De Vita, Ester Colarusso and 13 more

Abstract read
In one paragraph

Article in Journal of medicinal chemistry, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
–field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

23 authors.

Tania CiagliaDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
Valeria NapolitanoDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
Maria Rosaria MirandaDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
Danila La GioiaDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
Simona MusellaDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
Aniello Schiano MorielloInstitute of Biomolecular Chemistry, Consiglio Nazionale delle Ricerche, Comprensorio Olivetti, Via Campi Flegrei, 34, 80078 Pozzuoli, Naples, Italy.
Fabrizio MerciaiDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
Veronica Di SarnoDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
Simona De VitaDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.ORCID 0000-0002-8203-3580
Ester ColarussoDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
Gerardina SmaldoneDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
Francesca Di MatteoDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
Eduardo Maria SommellaDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.ORCID 0000-0001-8654-6431
Poulami KumarInstitute of Biomolecular Chemistry, Consiglio Nazionale delle Ricerche, Comprensorio Olivetti, Via Campi Flegrei, 34, 80078 Pozzuoli, Naples, Italy.
Marco AllaràInstitute of Biomolecular Chemistry, Consiglio Nazionale delle Ricerche, Comprensorio Olivetti, Via Campi Flegrei, 34, 80078 Pozzuoli, Naples, Italy.
Alessia LigrestiInstitute of Biomolecular Chemistry, Consiglio Nazionale delle Ricerche, Comprensorio Olivetti, Via Campi Flegrei, 34, 80078 Pozzuoli, Naples, Italy.ORCID 0000-0003-1787-3900
Isabel M Gomez-MonterreyDepartment of Pharmacy, University Federico II of Naples, Via D. Montesano 49, 80131 Naples, Italy.ORCID 0000-0001-6688-2606
Giuseppe BifulcoDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.ORCID 0000-0002-1788-5170
Gianluigi LauroDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.ORCID 0000-0001-5065-9717
Pietro CampigliaDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.ORCID 0000-0002-1069-2181
Carmine OstacoloDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.ORCID 0000-0003-3715-8680
Vincenzo VestutoDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.
Alessia BertaminoDepartment of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy.ORCID 0000-0002-5482-6276

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Molecular diversity is one of the most pursued objectives in drug discovery, and diversity-oriented synthesis (DOS) perfectly responds to the achievement of this goal. In this paper, we describe a DOS approach applied to the antitumor field with the aim of identifying new anticancer structures and their associated targets. To accomplish this ambitious project, after an initial stage of phenotypic evaluation, we set up an integrated platform of inverse virtual screening (IVS), bioinformatics, and omics to predict the biological targets of the most promising compounds

Indexed as

Antineoplastic AgentsComputational BiologyDrug DiscoveryApoptosisCell Line, TumorDrug Screening Assays, AntitumorHumansAntineoplastic Agents

Identifiers

PMID40705771
PMCPMC12362587

What Socratic holds

Textmetadata
LicenceCC BY
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.