Evidence mapPaperPMID 40774999Full record

ArticleScientific reports2025

The therapeutic potential of pegylated arginase I treatment in glioblastoma.

Marcus Kwong Lam Fung, Shing Chan, Stella Sun, Ping De Zhang, Gilberto Ka Kit Leung, Godfrey Chi Fung Chan

Abstract read
In one paragraph

Article in Scientific reports, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 3 papers.

0numbers the graph read from it
0cells of the map it votes in
3citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

3 citing papers in PubMed.

  1. Article
  2. Review
  3. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

6 authors.

Marcus Kwong Lam FungDepartment of Paediatrics & Adolescent Medicine, School of Clinical Medicine, LKS Faculty of Medicine, The University of Hong Kong, Pok Fu Lam, HKSAR, China.
Shing ChanDepartment of Paediatrics & Adolescent Medicine, School of Clinical Medicine, LKS Faculty of Medicine, The University of Hong Kong, Pok Fu Lam, HKSAR, China.
Stella SunDepartment of Surgery, School of Clinical Medicine, LKS Faculty of Medicine, The University of Hong Kong, Pok Fu Lam, HKSAR, China.
Ping De ZhangDepartment of Surgery, School of Clinical Medicine, LKS Faculty of Medicine, The University of Hong Kong, Pok Fu Lam, HKSAR, China.
Gilberto Ka Kit LeungDepartment of Surgery, School of Clinical Medicine, LKS Faculty of Medicine, The University of Hong Kong, Pok Fu Lam, HKSAR, China.
Godfrey Chi Fung ChanDepartment of Paediatrics & Adolescent Medicine, School of Clinical Medicine, LKS Faculty of Medicine, The University of Hong Kong, Pok Fu Lam, HKSAR, China. gcfchan@hku.hk.

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

This study used in vitro experiments and an orthotopic glioblastoma (GBM) mouse model to test the efficacy of human pegylated arginase I formulation, BCT-100, against the incurable cancer, GBM. Arginine auxotrophy in GBM was verified in silico and in vitro by absence of OTC and ASS1 expression. BCT-100 inhibited growth and induced cell death in four GBM cell lines in vitro. Transcriptomics of U87 and U373 treated with BCT-100 responded differently. BCT-100-treated U87 showed autophagy induction. Cytotoxicity enhancement was observed in four cell lines treated with BCT-100 + chloroquine (CQ). CQ + BCT-100 induced caspase-dependent and caspase-independent cell death in luciferase-transfected U87 (U87(lf+)). BCT-100 or CQ monotherapy, but not BCT-100+ CQ, prolonged survival of intracranial U87(lf+)-bearing mice similarly without suppressing tumor growth. Mouse microglia cell BV2 protected U87(lf+) from BCT100-induced cytotoxicity in transwell co-culture. Etoposide suppressed BV2's protection to U87(lf+) upon BCT-100 treatment by suppressing the growth and inducing cell death of BV2, suggesting microglial suppression as a strategy for enhancing the efficacy of BCT-100. Microglial protection may explain the in vitro and in vivo discrepancies. Further investigation into microglia/GBM interactions may help improve the efficacy of arginine deprivation therapy against GBM.

Indexed as

Antineoplastic AgentsArginaseBrain NeoplasmsGlioblastomaPolyethylene GlycolsAnimalsArginineCell Line, TumorCell ProliferationChloroquineHumansMiceMicrogliaXenograft Model Antitumor AssaysAntineoplastic AgentsARG1 protein, humanArginaseArginineChloroquinePolyethylene GlycolsArginine deprivationCombination therapyGlioblastomaMicrogliaPegylated arginase ITumor microenvironment

Identifiers

PMID40774999
PMCPMC12331973

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.