Evidence map›Paper›PMID 40938862›Full record

ArticlePloS one2025

Using systems biology and drug repositioning approaches to discover FDA-approved drugs candidates for endometriosis treatment.

Samira Sanami, Shahrzad Aghaamoo, Sajjad Ahmad, Ali Fazli, Bahareh Mansouri, Jonas Ivan Nobre Oliveira, Mojgan Rahmanian

Abstract read
In one paragraph

Article in PloS one, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 2 papers.

0numbers the graph read from it
0cells of the map it votes in
2citing papers in PubMed
–field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

2 citing papers in PubMed.

  1. Review
  2. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

7 authors.

Samira SanamiAbnormal Uterine Bleeding Research Center, Semnan University of Medical Sciences, Semnan, Iran.
Shahrzad AghaamooAbnormal Uterine Bleeding Research Center, Semnan University of Medical Sciences, Semnan, Iran.
Sajjad AhmadDepartment of Health and Biological Sciences, Abasyn University, Peshawar, Pakistan.
Ali FazliAbnormal Uterine Bleeding Research Center, Semnan University of Medical Sciences, Semnan, Iran.
Bahareh MansouriAbnormal Uterine Bleeding Research Center, Semnan University of Medical Sciences, Semnan, Iran.
Jonas Ivan Nobre OliveiraDepartment of Biophysics and Pharmacology, Federal University of Rio Grande do Norte, Natal, Rio Grande do Norte, Brazil.
Mojgan RahmanianAbnormal Uterine Bleeding Research Center, Semnan University of Medical Sciences, Semnan, Iran.ORCID https://orcid.org/0009-0009-7122-5227

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Endometriosis is characterized by the presence of endometrial tissue outside the uterine cavity. The administration of drugs designated for this condition has significant adverse effects, such as signs of estrogen insufficiency and suppression of ovulation. Considering this issue, this study aims to employ drugs repurposing approaches for the treatment of endometriosis. The GSE120103 dataset was selected to assess the expression of genes involved in endometriosis, then differentially expressed genes (DEGs) were identified using the "Limma" package in R Studio. Functional and pathway enrichment analysis of 708 up-regulated and 414 down-regulated DEGs was performed using ShinyGO 0.81 and DAVID tools. the Search Tool for the Retrieval of Interacting Genes/Proteins (STRING) was then used to build a protein-protein interaction (PPI) network of up-regulated DEGs, followed by Cytoscape software to identify hub genes. Vascular endothelial growth factor receptor 2 (VEGFR2) and interleukin-6 (IL-6) were identified as hub genes, assessments suggested that VEGFR2 may be a more promising possibility for druggability than IL-6. 16 FDA-approved drugs targeting VEGFR2 were identified, and molecular docking analysis indicated that ponatinib (-9.6 kcal/mol) had a more favorable binding energy than the co-crystal ligand (-9.2 kcal/mol). Moreover, molecular dynamics (MD) simulation analysis demonstrated considerable stability of the VEGFR2-ponatinib complex over a 100 nanoseconds (ns) timescale. The findings of this study indicate that ponatinib may provide considerable therapeutic promise for the treatment of endometriosis. Nevertheless, additional experimental investigations are required to evaluate its therapeutic efficacy.

Indexed as

Drug RepositioningEndometriosisSystems BiologyDrug ApprovalFemaleGene Regulatory NetworksHumansInterleukin-6Molecular Docking SimulationProtein Interaction MapsUnited StatesUnited States Food and Drug AdministrationVascular Endothelial Growth Factor Receptor-2Interleukin-6Vascular Endothelial Growth Factor Receptor-2

Identifiers

PMID40938862
PMCPMC12431326

What Socratic holds

Textmetadata
LicenceCC BY
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Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.