Evidence mapPaperPMID 41185102Full record

ArticleAnimal models and experimental medicine2025

Pimobendan alleviates myocyte apoptosis and fibrosis associated with mitral regurgitation by targeting endoplasmic reticulum stress.

Pakit Boonpala, Sushawadee Tongta, Nakkawee Saengklub, Vudhiporn Limprasutr, Sirinapa Srikam, Wilawan Ji-Au, Tussapon Boonyarattanasoonthorn, Yaowalak Panyasing, Sarawut Kumphune, Sarinee Kalandakanond-Thongsong and 1 more

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Article in Animal models and experimental medicine, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 1 paper.

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0cells of the map it votes in
1citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

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The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

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Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

1 citing paper in PubMed.

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4 · The record

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5 · Who and what money

Authors and funding

11 authors.

Pakit BoonpalaDepartment of Physiology, Faculty of Veterinary Science, Chulalongkorn University, Bangkok, Thailand.
Sushawadee TongtaChulalongkorn University Laboratory Animal Center (CULAC), Chulalongkorn University, Bangkok, Thailand.
Nakkawee SaengklubDepartment of Physiology, Faculty of Pharmacy, Mahidol University, Bangkok, Thailand.ORCID 0000-0001-8537-7576
Vudhiporn LimprasutrChulalongkorn University Laboratory Animal Center (CULAC), Chulalongkorn University, Bangkok, Thailand.ORCID 0000-0003-0769-0297
Sirinapa SrikamDepartment of Pathology, Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.
Wilawan Ji-AuDepartment of Pathology, King Chulalongkorn Memorial Hospital, Bangkok, Thailand.
Tussapon BoonyarattanasoonthornChulalongkorn University Laboratory Animal Center (CULAC), Chulalongkorn University, Bangkok, Thailand.
Yaowalak PanyasingDepartment of Pathology, Faculty of Veterinary Science, Chulalongkorn University, Bangkok, Thailand.
Sarawut KumphuneBiomedical Engineering Institute (BMEI), Chiang Mai University, Chiang Mai, Thailand.
Sarinee Kalandakanond-ThongsongDepartment of Physiology, Faculty of Veterinary Science, Chulalongkorn University, Bangkok, Thailand.
Anusak KijtawornratDepartment of Physiology, Faculty of Veterinary Science, Chulalongkorn University, Bangkok, Thailand.ORCID 0000-0002-7872-3183

Funding

The 100th Anniversary Chulalongkorn University Fund for Doctoral Scholarshipthe 90th Anniversary of Chulalongkorn University Fund GCUGR1125641042Dthe National Budget to CULAC 390252002the Thailand Science Research and Innovation Fund at Chulalongkorn University HEAF673100100
6 · The paper itself

Abstract

backgroundEndoplasmic reticulum (ER) stress is an important factor in the development of numerous cardiovascular disorders; nevertheless, the association between ER stress and mitral regurgitation (MR) remains inadequately characterized. The molecular mechanism of pimobendan (PIMO) that contributes to the delay in congestive heart failure (CHF) in MR associated with apoptosis and fibrosis is still unclear. Our aim was to examine the impact of PIMO on ER stress, apoptosis, and fibrosis in a chronic MR rat model.

methodsMR was surgically induced in 10 Sprague-Dawley rats, with 5 serving as sham operation controls. At 8 weeks postsurgery, the MR animals were randomly allocated into two groups: MR and MR + PIMO groups. PIMO was administered twice daily through oral gavage for 4 weeks, whereas the sham and MR groups were administered similar quantities of drinking water. Echocardiography was conducted before the delivery of PIMO as a baseline measure and at the end of the study. At the end of the investigation, hearts were procured for histopathological and ER stress evaluations.

resultsPIMO significantly maintained heart function and structural remodeling in the MR animals. PIMO significantly reduced MR-induced myocyte apoptosis (p = 0.044) and fibrosis (p = 0.002) by reducing the messenger RNA expression of genes associated with ER stress (GRP78 [glucose-regulated protein 78], ATF4 [activating transcription factor 4], and CHOP [C/ERP homologous protein]) compared to the MR group (p < 0.05, p < 0.01, and p < 0.001, respectively).

conclusionPIMO demonstrated cardioprotective benefits on heart function, myocyte apoptosis, and fibrosis by regulating ER stress in an MR-induced CHF rat model.

Indexed as

ApoptosisEndoplasmic Reticulum StressMitral Valve InsufficiencyMyocytes, CardiacAnimalsDisease Models, AnimalFibrosisMaleRatsRats, Sprague-Dawleyapoptosisendoplasmic reticulum (ER) stressfibrosismitral regurgitationmitral regurgitation rat modelpimobendan

Identifiers

PMID41185102
PMCPMC12746179

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.