Evidence map›Paper›PMID 41219567›Full record

ArticlePharmaceutical research2025

Development and Optimization of Myricetin Loaded Inhalable Microsphere to Treat COPD.

Suhas Shivaji Siddheshwar, Darshana Jagtap, Someshwar Dattatraya Mankar, Arti Changdev Ghorpade, Santosh Bhausaheb Dighe, Sanjay Bhawar

Abstract read
PubMed Publisher
In one paragraph

Article in Pharmaceutical research, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
–field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

6 authors.

Suhas Shivaji SiddheshwarDepartment of Pharmaceutics, Pravara Rural College of Pharmacy, Loni, Maharashtra, India. drssiddheshwar@gmail.com.ORCID http://orcid.org/0000-0002-7944-9470
Darshana JagtapDepartment of Pharmaceutics, Pravara Rural College of Pharmacy, Loni, Maharashtra, India.ORCID http://orcid.org/0009-0002-2647-9534
Someshwar Dattatraya MankarDepartment of Pharmaceutics, Pravara Rural College of Pharmacy, Loni, Maharashtra, India.ORCID http://orcid.org/0000-0003-3991-9412
Arti Changdev GhorpadeDepartment of Pharmaceutics, Pravara Rural College of Pharmacy, Loni, Maharashtra, India.ORCID http://orcid.org/0009-0003-7843-5688
Santosh Bhausaheb DigheDepartment of Pharmacology, Pravara Rural College of Pharmacy, Loni, Maharashtra, India, 413736.ORCID http://orcid.org/0000-0003-3260-2981
Sanjay BhawarDepartment of Pharmacology, Pravara Rural College of Pharmacy, Loni, Maharashtra, India, 413736.ORCID http://orcid.org/0000-0002-5345-0799

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

objectivesTo develop and optimize myricetin-loaded inhalable microspheres using ionotropic gelation technique for sustained pulmonary delivery in Chronic Obstructive Pulmonary Disease (COPD) treatment.

methodsMyricetin-loaded microspheres were prepared using varying concentrations of gellan gum and sodium alginate through a 3

resultsThe optimized formulation (DF4) exhibited spherical morphology with ideal particle size for pulmonary delivery (7.72 μm), high entrapment efficiency (72.84%), and negative zeta potential ensuring colloidal stability. This formulation demonstrated excellent aerodynamic properties (FPF 31.71%), sustained drug release over 12 h, and remarkable stability over 6 months under both accelerated and real-time storage conditions. The formulation showed significant bronchodilatory activity with 63.47% relaxation at 25 μg/ml, achieving approximately 80.8% efficacy compared to theophylline anhydrous.

conclusionThe optimized myricetin-loaded inhalable microspheres represent a promising pulmonary delivery system for COPD management, offering advantages of sustained drug release, improved lung deposition, and significant bronchodilatory effect. This formulation holds potential for reducing dosing frequency, enhancing patient compliance, and improving therapeutic outcomes in COPD patients, warranting further in vivo studies before clinical translation.

Indexed as

Bronchodilator AgentsFlavonoidsMicrospheresPulmonary Disease, Chronic ObstructiveAdministration, InhalationAlginatesAnimalsChemistry, PharmaceuticalDelayed-Action PreparationsDrug LiberationDrug StabilityGoatsParticle SizePolysaccharides, BacterialTheophyllineTracheaAlginatesBronchodilator AgentsDelayed-Action PreparationsFlavonoidsgellan gummyricetinPolysaccharides, BacterialTheophyllinebronchodilatory activitycontrolled releaseCOPDfactorial designinhalable microspheresionotropic gelationmyricetin

Identifiers

What Socratic holds

Textmetadata
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.