Evidence mapPaperPMID 41280890Full record

ArticleFrontiers in immunology2025

A novel GCGR/GLP-1R dual-agonist TB001 ameliorates kidney fibrosis via inhibiting PERK-mediated endoplasmic reticulum stress pathway.

Weijie Lai, Linjie Peng, Jianliang Min, Longhui Qiu, Chang Wang, Shuangjin Yu, Qihao Li, Ruobing Li, Xianxing Jiang, Guodong Chen

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Article in Frontiers in immunology, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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1 · What the graph read from it

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The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

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3 · Its place in the literature

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4 · The record

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5 · Who and what money

Authors and funding

10 authors.

Weijie Lai *Organ Transplant Center, The First Affiliated Hospital of Sun Yat-sen University, Guangzhou, China.
Linjie Peng *The Second Affiliated Hospital of Southern University of Science and Technology, Shenzhen, China.
Jianliang Min *School of Medicine, Jiaying University, Meizhou, China.
Longhui Qiu *Organ Transplant Center, The First Affiliated Hospital of Sun Yat-sen University, Guangzhou, China.
Chang WangOrgan Transplant Center, The First Affiliated Hospital of Sun Yat-sen University, Guangzhou, China.
Shuangjin YuOrgan Transplant Center, The First Affiliated Hospital of Sun Yat-sen University, Guangzhou, China.
Qihao LiOrgan Transplant Center, The First Affiliated Hospital of Sun Yat-sen University, Guangzhou, China.
Ruobing LiOrgan Transplant Center, The First Affiliated Hospital of Sun Yat-sen University, Guangzhou, China.
Xianxing JiangSchool of Pharmaceutical Sciences, Sun Yat-sen University, Sun Yat-sen University, Guangzhou, China.
Guodong ChenOrgan Transplant Center, The First Affiliated Hospital of Sun Yat-sen University, Guangzhou, China.

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Background: Chronic kidney disease (CKD) affects over one million individuals worldwide and remain a critical economic and healthcare burden. Renal fibrosis is the hallmark of CKD. Previous reports showed that GLP-1R agonists could help prevent kidney fibrosis in diabetic patients. In this study, we aimed to determine the efficacy of a novel GLP-1R and GCGR co-agonist, TB001 in the development of renal fibrosis using both Methods: Unilateral ureteral obstruction (UUO) surgery was performed on adult B6 mice to establish a mouse model of kidney fibrosis. Mice that underwent sham surgery served as the control group. UUO mice were treated with vehicle or TB001 daily post-surgery and were sacrificed at day 14. Tissue samples were collected for immunohistochemistry and kidney mRNA gene expression analysis. Mouse tubular cells (mTECs) stimulated with TGF-β were used to model kidney fibrosis Results: Compared with vehicle treatment, TB001 treatment significantly improved renal histopathology and reduced interstitial collagen deposition and macrophage infiltration in obstructed kidneys. Both Conclusion: This study demonstrated that TB001, a novel GCGR/GLP-1R co-agonist, effectively attenuates renal fibrosis in pre-clinical models, potentially through the inhibition of PERK-mediated ER stress in tubular cells.

Indexed as

Endoplasmic Reticulum StressGlucagon-Like Peptide-1 Receptor AgonistsReceptors, GlucagonRenal Insufficiency, ChronicAnimalsCells, CulturedDisease Models, AnimaleIF-2 KinaseEpithelial-Mesenchymal TransitionFibrosisKidney TubulesMaleMiceMitochondriaEif2ak3 protein, mouseeIF-2 KinaseGlucagon-Like Peptide-1 Receptor AgonistsReceptors, GlucagonEMTer stressGCGRGLP-1rpERKrenal fibrosis

Identifiers

PMID41280890
PMCPMC12636095

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.