Evidence map›Paper›PMID 41317193›Full record

ReviewNaunyn-Schmiedeberg's archives of pharmacology2026

Viniferin and its derivatives: a comprehensive review of structural variations and promising pharmacological applications in disease prevention and therapeutic development.

Ahmed M El-Dessouki, Kareem A Attallah, Aya H Eid, Eman S Zaki, Samar S Khalaf, Riham A El-Shiekh, Nada M Kamel, Rana M ElBishbishy, Ahmed H Elosaily

Abstract readReview
In one paragraph

Review in Naunyn-Schmiedeberg's archives of pharmacology, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 1 paper.

0numbers the graph read from it
0cells of the map it votes in
1citing papers in PubMed
–field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

1 citing paper in PubMed.

  1. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

9 authors.

Ahmed M El-DessoukiPharmacology and Toxicology Department, Faculty of Pharmacy6 of October City, Ahram Canadian University, Giza, 12566, Egypt.
Kareem A AttallahResearch and Development Department, Biotechnology Research Center, 23 July St., Industrial Zone, New Damietta, 34517, Egypt.ORCID http://orcid.org/0000-0002-5886-1466
Aya H EidPharmacology and Toxicology Department, Faculty of Pharmacy, Heliopolis University, Cairo, Egypt.
Eman S ZakiPharmacology and Toxicology Department, Faculty of Pharmacy, Heliopolis University, Cairo, Egypt.
Samar S KhalafBiochemistry Department Faculty of Pharmacy, Heliopolis University, Cairo, Egypt. Samar.samir@hu.edu.eg.ORCID http://orcid.org/0000-0003-4986-8567
Riham A El-ShiekhDepartment of Pharmacognosy, Faculty of Pharmacy, Cairo University, Cairo, 11562, Egypt.
Nada M KamelDepartment of Pharmacology and Toxicology, Faculty of Pharmacy, Cairo University, Kasr El-Aini Street, Cairo, 11562, Egypt.
Rana M ElBishbishyDepartment of Pharmacology and Toxicology, Faculty of Pharmacy, Cairo University, Kasr El-Aini Street, Cairo, 11562, Egypt.
Ahmed H ElosailyDepartment of Pharmacognosy, Faculty of Pharmacy, Ahram Canadian University, Giza, 12573, Egypt.

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Viniferin, a resveratrol-derived compound that belongs to a group of plant-produced stilbenoids, functions as a natural defense against microbial invasion, toxins, infections, and ultraviolet radiation. Alpha-(α-) viniferin (trimer), beta-(β-) viniferin (dimer), delta-(δ-) viniferin (oxidative dehydrodimer), epsilon-(ε-) viniferin (distinct dehydrodimer), gamma-(γ-) viniferin (isomeric oligomer), vitisin A (R-viniferin), and vitisin B (R2-viniferin) are structurally diverse forms with distinct pharmacological activities. Antioxidant studies showed that ε-viniferin exhibited a 2,2-diphenyl-1-picrylhydrazyl (DPPH) free radical scavenging half-maximal inhibitory concentration (IC₅₀) of about 80 µM. Also, suppression of nuclear factor kappa B, cyclooxygenase-2, and prostaglandin E₂ are anti-inflammatory mechanisms. R2-viniferin demonstrated an IC₅₀ of 9.7 µM against hepatocellular carcinoma HepG2 cells at 72 h, mediated through apoptosis and cell-cycle arrest, according to anticancer studies that demonstrated dose-dependent cytotoxicity. There have been reports of additional activity against models of glioblastoma and prostate cancer. In metabolic disorders, oral α-viniferin (20-40 mg/kg/day) improved lipid and glucose homeostasis in mice fed a high-fat diet, and it additionally improved liver and renal biomarkers such as blood urea nitrogen, creatinine, alanine aminotransferase, and aspartate aminotransaminase. Several bacterial strains have shown signs of preliminary antimicrobial action. By reducing excitotoxicity and oxidative stress, viniferins also have neuroprotective effects. They also have anti-melanogenic properties by blocking the tyrosinase and melanogenesis pathways. Collectively, viniferins demonstrate pleiotropic pharmacologic activities by defined molecular mechanisms and quantifiable dose-dependent effects. The properties classify viniferins as new multifunctional drug candidates for discovery and nutraceuticals, but they highlight the need for standardized pharmacologic assays, further preclinical validation, and pharmacokinetic optimization towards clinical use.

Indexed as

BenzofuransStilbenesAnimalsAnti-Inflammatory AgentsAntioxidantsHumansStructure-Activity RelationshipAnti-Inflammatory AgentsAntioxidantsBenzofuransStilbenesChemistryDrug discoveryFunctional foodsHealth benefitsPharmacologyViniferin

Identifiers

PMID41317193
PMCPMC13053555

What Socratic holds

Textmetadata
LicenceCC BY
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Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.