Evidence map›Paper›PMID 41423449›Full record

ArticleNature communications2025

Restoration of PKM1 improves functional maturation of human stem-cell derived-β cell by regulating PEP metabolism.

Haopeng Lin, Xin Liu, Feng Zhang, Deqi Chen, Xiaoxiao Xie, Qifei Dong, Jiawei Yan, Jiaxiang Yin, Zirong Bi, Zhihua Dou and 10 more

Abstract read
In one paragraph

Article in Nature communications, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 1 paper.

0numbers the graph read from it
0cells of the map it votes in
1citing papers in PubMed
–field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

1 citing paper in PubMed.

  1. Review
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

20 authors.

Haopeng LinSchool of Biomedical Engineering, Guangzhou Medical University, Guangzhou, China.
Xin LiuGuangzhou National Laboratory, Guangzhou, China.
Feng ZhangGuangzhou National Laboratory, Guangzhou, China.
Deqi ChenGuangzhou National Laboratory, Guangzhou, China.
Xiaoxiao XieSchool of Biomedical Engineering, Guangzhou Medical University, Guangzhou, China.
Qifei DongGuangzhou National Laboratory, Guangzhou, China.
Jiawei YanGuangzhou National Laboratory, Guangzhou, China.
Jiaxiang YinGuangzhou National Laboratory, Guangzhou, China.
Zirong BiGuangzhou National Laboratory, Guangzhou, China.
Zhihua DouGuangzhou National Laboratory, Guangzhou, China.
Yingling JiangGuangzhou National Laboratory, Guangzhou, China.
Kuo JiangGuangzhou National Laboratory, Guangzhou, China.
Tongran ZhangGuangzhou National Laboratory, Guangzhou, China.
Peng XueGuangzhou National Laboratory, Guangzhou, China.
Wei PengGuangzhou National Laboratory, Guangzhou, China.ORCID http://orcid.org/0000-0002-0949-4487
Lihua ChenGuangzhou National Laboratory, Guangzhou, China.ORCID http://orcid.org/0000-0003-3369-1875
Tao XuSchool of Biomedical Engineering, Guangzhou Medical University, Guangzhou, China. xutao@ibp.ac.cn.ORCID http://orcid.org/0000-0002-8260-9754
Zonghong LiGuangzhou National Laboratory, Guangzhou, China. Li_zonghong@gzlab.ac.cn.ORCID http://orcid.org/0000-0002-5153-0007
Yanying GuoDepartment of Endocrinology and Metabolism, People's Hospital of Xinjiang Uygur Autonomous Region, Xinjiang Clinical Research Center for Diabetes, Xinjiang Key Laboratory of Cardiovascular Homeostasis and Regeneration Research, Urumqi, China. gyy@xjrmyy.com.
Huisheng LiuSchool of Biomedical Engineering, Guangzhou Medical University, Guangzhou, China. Liu_huisheng@gzlab.ac.cn.ORCID http://orcid.org/0000-0001-5371-7943

Funding

Guangzhou Medical University (Guangzhou Medical College) 06-445-1247National Natural Science Foundation of China (National Science Foundation of China) 2021YFA1101300, 2020YFA0908200, 32570979
6 · The paper itself

Abstract

Human stem cell-derived β (SC-β) cells still exhibit limited glucose response required for insulin secretion due to glycolytic bottlenecks, yet how these metabolic abnormalities impact glucose response and functional maturation of SC-β cells remains unclear. In this study, we identify a metabolic checkpoint located at PEP accumulation that impedes the functional maturation, which is rescued by restoration of pyruvate kinase M1 (PKM1). Glucose-tracing metabolomics in human stem cell-derived islets reveal abnormal glycolytic PEP accumulation at resting condition, associated with impaired calcium response and insulin secretion upon high glucose or glycolytic metabolite stimulation. Mechanistically, elevated PEP significantly raises intracellular basal calcium levels and downregulates expression of genes involved in TCA cycle as elucidated by single cell transcriptomics. Furthermore, the activity of pyruvate kinase, which metabolizes PEP, is notably reduced due to low PKM1 expression. Overexpression of PKM1 alleviates PEP accumulation, restores TCA-related gene expression, and enhances glucose-stimulated calcium responses and insulin secretion. Together, our findings reveal a critical role of PKM1-regulated PEP metabolism in SC-β cell functional maturation and highlight the importance of metabolic reprogramming for advancing stem cell-based therapies for diabetes.

Indexed as

Insulin-Secreting CellsPyruvate KinaseCalciumCell DifferentiationCitric Acid CycleGlucoseGlycolysisHumansInsulin SecretionStem CellsThyroid Hormone-Binding ProteinsCalciumGlucosePyruvate KinaseThyroid Hormone-Binding Proteins

Identifiers

PMID41423449
PMCPMC12830896

What Socratic holds

Textmetadata
LicenceCC BY-NC-ND
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.