Evidence map›Paper›PMID 41444645›Full record

ArticleHuman genomics2025

Two cases of TBL1XR1 heterozygous variants in children: a new splicing site variant identification and functional analysis through molecular docking and molecular dynamics simulation.

Yaxue Xie, Ziyan Zhang, Gang Zhu, Zhichao Li, Huiling Zhang, Jiaqi Zhang, Lin Wan, Guang Yang

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In one paragraph

Article in Human genomics, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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5 · Who and what money

Authors and funding

8 authors.

Yaxue Xie *Department of Pediatrics, The First Medical Center of Chinese PLA General Hospital, Beijing, 100853, China.
Ziyan Zhang *Department of Pediatrics, The First Medical Center of Chinese PLA General Hospital, Beijing, 100853, China.
Gang ZhuDepartment of Pediatrics, The First Medical Center of Chinese PLA General Hospital, Beijing, 100853, China.
Zhichao LiDepartment of Pediatrics, The First Medical Center of Chinese PLA General Hospital, Beijing, 100853, China.
Huiling ZhangDepartment of Pediatrics, The First Medical Center of Chinese PLA General Hospital, Beijing, 100853, China.
Jiaqi ZhangDepartment of Pediatrics, The First Medical Center of Chinese PLA General Hospital, Beijing, 100853, China.
Lin WanDepartment of Pediatrics, The First Medical Center of Chinese PLA General Hospital, Beijing, 100853, China.
Guang YangDepartment of Pediatrics, The First Medical Center of Chinese PLA General Hospital, Beijing, 100853, China. yangg301@126.com.

Funding

Beijing Natural Science Foundation 7222187Capital's Funds for Health Improvement and Research 2024-2-5082Innovation Talent Fund of Senior Department of Pediatrics, The Seventh Medical Center of PLA General Hospital QZX-04-EKLHJH-3the general project of National Key Research and Development Program of China 2022YFC2705300the general project of National Key Research and Development Program of China 2023YFC2706405the key project of innovation cultivation fund of the Seventh Medical Center of Chinese PLA General Hospital qzx-2023-1
6 · The paper itself

Abstract

backgroundTransducin β-like 1 X-linked receptor 1 (TBL1XR1) protein is an important component of NCoR/SMRT complex. The variants of TBL1XR1 are associated with Pierpont syndrome (PS) and developmental delay (DD). This study aimed to discover new TBL1XR1 variants, their clinical manifestations, and protein-level changes.

methodsWhole-exome sequencing was used to identify patients with TBL1XR1 variants in 2024. Minigene assay was used to investigate specific splice site, which was further validated by Sanger sequencing. Structural changes in the TBL1XR1 protein were analyzed using PyMOL and molecular dynamics (MD) simulations. Potential binding partners were predicted via Genecards, STRING, and Cytoscape, while molecular docking was employed to assess how variants affect protein complex interactions.

resultsTwo novel TBL1XR1 variants (c.1048-8_1049del and c.865-7A>G) were identified in two patients. Patient 1 exhibits global developmental delay (GDD), while patient 2 displays with facial dysmorphism and autism spectrum disorder. c.865-7A>G is a non-canonical splicing variant causing abnormal mRNA splicing. SpliceAI and RDDC predicted its splicing pattern. Minigene analysis found a 6 bp (TCTCAG) insertion in mRNA, leading to two amino acid (SQ) insertion in the TBL1XR1 protein. Therefore, P2 was diagnosed with PS. Variant changed the local hydrogen bond network and electrostatic potential. MD simulations showed variant changed the conformation of TBL1XR1 protein. Protein–protein interaction analysis selected NCOR1 for docking with TBL1XR1. Their interaction was reduced after the insertion of SQ, which may contribute to the occurrence of PS.

conclusionThis study reported two patients manifesting with GDD and PS, which were identified with two novel variants of TBL1XR1 (c.1048-8_1049del, p.(N350X)) and (c.865-7A>G, p.K288_T289insSQ), respectively. c.865-7A>G variant might lead to PS by reducing its interaction with NCOR1.

Indexed as

Developmental DisabilitiesNuclear ProteinsReceptors, Cytoplasmic and NuclearRepressor ProteinsChildChild, PreschoolExome SequencingFemaleHeterozygoteHumansMaleMolecular Docking SimulationMolecular Dynamics SimulationMutationRNA Splice SitesRNA SplicingNuclear ProteinsReceptors, Cytoplasmic and NuclearRepressor ProteinsRNA Splice SitesTBL1XR1 protein, humanMinigeneMolecular dockingMolecular dynamicsPierpont syndromeTBL1XR1

Identifiers

PMID41444645
PMCPMC12781238

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