Evidence mapPaperPMID 41455835Full record

ArticleScientific reports2025

Anticancer potential of Dendrocnide meyeniana through phytochemical profiling, ADMET analysis, molecular docking, and in silico cytotoxicity evaluation.

Edlyn E Pooten, Khristina G Judan Cruz, Evaristo A Abella, Anna Karen C Laserna, Abul Baskhar Mir Md Khademul Islam, Kozo Watanabe

Abstract read
In one paragraph

Article in Scientific reports, 2025. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

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3 · Its place in the literature

Who cites it

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4 · The record

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5 · Who and what money

Authors and funding

6 authors.

Edlyn E PootenCentre for Marine Environmental Studies (CMES), Ehime University, Bunkyo-cho-3, Matsuyama, Ehime, 790-8577, Japan.
Khristina G Judan CruzCentre for Marine Environmental Studies (CMES), Ehime University, Bunkyo-cho-3, Matsuyama, Ehime, 790-8577, Japan. kjcruz@clsu.edu.ph.
Evaristo A AbellaDepartment of Biological Sciences, Central Luzon State University, 3120, Science City of Muñoz, Nueva Ecija, Philippines.
Anna Karen C LasernaCentral Instrumentation Facility, Office of the Vice Chancellor for Research and Innovation, De La Salle University, 2401 Taft Avenue, Malate, 1004, Manila, Philippines.
Abul Baskhar Mir Md Khademul IslamDepartment of Genetic Engineering & Biotechnology, University of Dhaka, Dhaka, Bangladesh.
Kozo WatanabeCentre for Marine Environmental Studies (CMES), Ehime University, Bunkyo-cho-3, Matsuyama, Ehime, 790-8577, Japan. watanabe.kozo.mj@ehime-u.ac.jp.

Funding

Japan Society for the Promotion of Science (JSPS) Core-to-Core Program B. Asia-Africa Science Platforms; JSPS Bilateral Joint Research Projects; Ministry of Education, Culture, Sports, Science and Technology, Japan (MEXT); Leading Academia in Marine and Environment Pollution Research (LaMer) JPJSCCB20240008; 120248601
6 · The paper itself

Abstract

Phytochemicals are widely explored for cancer therapeutics due to their structural diversity and broad pharmacological activities. This study investigated the phytochemical composition and anticancer potential of Dendrocnide meyeniana using integrated in silico approaches. Gas chromatography-mass spectrometry (GC-MS) and ultra-high-performance liquid chromatography-quadrupole time-of-flight mass spectrometry (UHPLC-QTOF-MS) identified 78 compounds, confirming the plant's rich chemical diversity. Four cancer-related targets- EGFR, p53, MMP7 and CDK8/Cyclin C were selected for molecular docking to identify potential inhibitors. Drug-likeness and ADMET profiling of nine bioactive candidates revealed Cryptotanshinone as the most promising compound, exhibiting favorable pharmacokinetic and safety properties. Molecular docking showed that Cryptotanshinone possessed strong binding affinities toward EGFR ( -8.8 kcal/mol), p53 (-8.7 kcal/mol), MMP7 (-8.7 kcal/mol), and CDK8/Cyclin C (-9.8 kcal/mol), comparable to or exceeding the reference drug Erlotinib (-9.0 kcal/mol for EGFR). Toxicity prediction indicated no hepatotoxic, mutagenic, or cytotoxic effects, though the compound showed potential carcinogenic activity possibly linked to pathway-specific interaction in cell-cycle regulation. Molecular dynamics simulation further validated the stability of the Cryptotanshinone-EGFR complex, exhibiting moderate RMSD values and limited structural fluctuations indicative of stable interactions. Collectively, these findings highlight Cryptotanshinone from D. meyeniana as a promising natural lead for anticancer drug development, characterized by strong binding affinity, favorable pharmacokinetics, and structural stability in silico. Further in vitro and in vivo studies are warranted to confirm its therapeutic efficacy and safety.

Indexed as

Antineoplastic Agents, PhytogenicPhytochemicalsCell Line, TumorComputer SimulationErbB ReceptorsHumansMolecular Docking SimulationPhenanthrenesAntineoplastic Agents, PhytogeniccryptotanshinoneEGFR protein, humanErbB ReceptorsPhenanthrenesPhytochemicalsADMETDendrocnide meyenianaGC-MSIn silicoMolecular dockingUHPLC-QTOF-MS

Identifiers

PMID41455835
PMCPMC12823615

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.