Evidence mapPaperPMID 41467933Full record

ArticleCell biochemistry and biophysics2026

Dioxopiperidinamide Derivative SKT-36 Alleviates scopolamine-induced Cognitive and Neurobehavioral Impairments in an In-vivo Zebrafish Model.

Sanjay Gopi, S Madesh, Karthikeyan Ramamurthy, S Kaliraj, Bader O Almutairi, Ki Choon Choi, Ajay Guru, Kathiravan Muthu Kumaradoss, Jesu Arockiaraj

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Article in Cell biochemistry and biophysics, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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1 · What the graph read from it

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The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

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3 · Its place in the literature

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4 · The record

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5 · Who and what money

Authors and funding

9 authors.

Sanjay GopiToxicology and Pharmacology Laboratory, Department of Biotechnology, Faculty of Science and Humanities, SRM Institute of Science and Technology, Kattankulathur, 603203, Chengalpattu District, Tamil Nadu, India.
S MadeshToxicology and Pharmacology Laboratory, Department of Biotechnology, Faculty of Science and Humanities, SRM Institute of Science and Technology, Kattankulathur, 603203, Chengalpattu District, Tamil Nadu, India.
Karthikeyan RamamurthyToxicology and Pharmacology Laboratory, Department of Biotechnology, Faculty of Science and Humanities, SRM Institute of Science and Technology, Kattankulathur, 603203, Chengalpattu District, Tamil Nadu, India.
S KalirajDepartment of Chemistry, Faculty of Engineering and Technology, SRM Institute of Science and Technology, Kattankulathur, 603203, Chengalpattu District, Tamil Nadu, India.
Bader O AlmutairiDepartment of Zoology, College of Science, King Saud University, P.O. Box 2455, Riyadh, 11451, Saudi Arabia.
Ki Choon ChoiGrassland and Forage Division, National Institute of Animal Science, RDA, Wanju-gun, Republic of Korea, 31000.
Ajay GuruMarwadi University Research Center, Marwadi University, Rajkot, 360003, Gujarat, India. ajayguru040996@gmail.com.
Kathiravan Muthu KumaradossDr APJ Abdul Kalam Research Lab, Department of Pharmaceutical Chemistry, SRM College of Pharmacy, Faculty of Medicine and Health Sciences, SRM Institute of Science and Technology, Kattankulathur, 603203, Chengalpattu District, Tamil Nadu, India.
Jesu ArockiarajToxicology and Pharmacology Laboratory, Department of Biotechnology, Faculty of Science and Humanities, SRM Institute of Science and Technology, Kattankulathur, 603203, Chengalpattu District, Tamil Nadu, India. jesuaroa@srmist.edu.in.

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Dementia, characterized by cognitive decline and synaptic dysfunction, presents significant therapeutic challenges. This study explores the potential of SKT-36, a novel Dioxopiperidinamide (DOPA) derivative, in reversing scopolamine (SCP)-induced cognitive deficits in an in-vivo zebrafish model. SKT-36 exhibits high neuroprotective potential due to its inherent antioxidant and anti-inflammatory properties. Network pharmacology analysis revealed 637 intersecting targets linking SKT-36 with dementia-associated genes such as STAT3, GSK3B, and HSP90AB1 identified as key hubs. Molecular docking also confirmed highly favorable binding affinity of SKT-36 with Danio rerio of AChE, exhibited a binding energy of -6.58 kcal/mol. For in vivo analysis, zebrafish were treated with SKT-36 at 10 µM and 7.5 µM, and the effects were assessed using neurobehavioral, biochemical, and gene expression studies. SKT-36 at 10 µM significantly enhanced locomotor activity, reduced anxiety-like behavior, and improved spatial and recognition memory, as shown by various behavioral tests. Biochemically, SKT-36 reduced oxidative stress markers and restored antioxidant enzyme activities. Also, superior acetylcholinesterase (AChE) inhibitory activity compared to standard treatments was seen suggesting effective cholinergic modulation. Gene expression analysis indicated SKT-36’s anti-inflammatory and neuroprotective effects, normalizing genes related to inflammation and neuronal plasticity. Histological analysis confirmed reduced neuronal damage and amyloid-beta plaque accumulation observed in the optic tectum regions. These findings highlight SKT-36 as a promising therapeutic agent for dementia, offering neuroprotective and cognitive benefits.

Indexed as

Behavior, AnimalCognitive DysfunctionNeuroprotective AgentsPiperidinesScopolamineAcetylcholinesteraseAnimalsAntioxidantsCholinesterase InhibitorsDisease Models, AnimalMaleMolecular Docking SimulationOxidative StressZebrafishAcetylcholinesteraseAntioxidantsCholinesterase InhibitorsNeuroprotective AgentsPiperidinesScopolamineDementiaDioxopiperidinamideMemory impairmentNeurobehavioral disabilityScopolamine

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.