Evidence mapPaperPMID 41501134Full record

ArticleScientific reports2026

In-silico screening of marine fungal metabolites identifies potential FtsZ inhibitors against MDR-tuberculosis through docking and molecular dynamics analysis.

Meghana S R, Yogesh H S, Sibghatullah Muhammad Ali Sangi, Anitha K N, Sadik Shaik, Sreeharsha Nagaraja, Girish Meravanige, Mohammed Monirul Islam, Pavan Kumar Sreenivasalu, Rashed M Almuqbil and 4 more

Abstract read
In one paragraph

Article in Scientific reports, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 2 papers.

0numbers the graph read from it
0cells of the map it votes in
2citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

2 citing papers in PubMed.

  1. Article
  2. Frontiers in bioinformatics · 2026
    Review
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

14 authors.

Meghana S RDepartment of Pharmacognosy, KLE College of Pharmacy, 560010, Rajajinagar, Bengaluru, India.
Yogesh H SDepartment of Pharmacology, Nitte College of Pharmaceutical sciences (Nitte Deemed to be University), Bengaluru, 560064, Karnataka, India.
Sibghatullah Muhammad Ali SangiBasic Medical Sciences Department, Dar Al Uloom University, Riyadh, 13314, Saudi Arabia.
Anitha K NDepartment of Pharmacology, Government College of Pharmacy, Bengaluru, 560027, Karnataka, India.
Sadik ShaikDepartment of Pharmacology, East Point College of Pharmacy, Bengaluru, 560049, Karnataka, India.
Sreeharsha NagarajaDepartment of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, 31982, Saudi Arabia.
Girish MeravanigeDepartment of Biomedical Sciences, College of Medicine, King Faisal University, Al-Ahsa, 31982, Saudi Arabia.
Mohammed Monirul IslamDepartment of Biomedical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, 31982, Saudi Arabia.
Pavan Kumar SreenivasaluDepartment of Restorative Dentistry and Endodontics, College of Dentistry, King Faisal University, Al-Ahsa, 31982, Saudi Arabia.
Rashed M AlmuqbilDepartment of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, 31982, Saudi Arabia.
Shahzad ChohanDepartment of Biomedical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, 31982, Saudi Arabia.
Bipindra PandeyDepartment of Pharmacy, Madan Bhandari Academy of Health Sciences, Hetauda, Nepal.
Shankar ThapaDepartment of Pharmacy, Madan Bhandari Academy of Health Sciences, Hetauda, Nepal.
Ayomide Victor AtokiDepartment of Biochemistry, Kampala International University, Ishaka- Bushenyi, Uganda. atokiav@kiu.ac.ug.ORCID http://orcid.org/0000-0003-1914-973X

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Tuberculosis (TB) remains a major global health challenge, intensified by the rise of multidrug-resistant (MDR) and extensively drug-resistant (XDR) strains of Mycobacterium tuberculosis. The bacterial cell division protein FtsZ, a key GDPase required for cytokinesis, represents a promising target for novel anti-TB therapeutics. This study aimed to identify potential FtsZ inhibitors among marine fungal metabolites using molecular docking, molecular dynamics (MD) simulations, and MM/GBSA analyses. Docking was performed with AutoDock Vina v1.2.0, followed by 200 ns MD simulations using Desmond to evaluate complex stability. Among 100 screened metabolites, Xanalteric acid II showed the strongest binding affinity (- 10.9 kcal/mol), interacting with Arg140 and Thr130 within the active site, outperforming the co-crystallized ligand (- 9.1 kcal/mol) and moxifloxacin (- 7.7 kcal/mol). The FtsZ-Xanalteric acid II complex exhibited stable RMSD and compact radius of gyration throughout the simulation. MM/GBSA analysis revealed a strong binding free energy (ΔG_bind = - 74.77 ± 4.95 kcal/mol), dominated by van der Waals and lipophilic interactions. PCA, FEL, and DCCM analyses confirmed the structural rigidity and energetic stability of the complex. These findings highlight Xanalteric acid II as a promising marine-derived inhibitor of FtsZ and support the potential of marine metabolites in developing next-generation anti-TB agents.

Indexed as

Antitubercular AgentsBacterial ProteinsCytoskeletal ProteinsFungiMycobacterium tuberculosisTuberculosis, Multidrug-ResistantMolecular Docking SimulationMolecular Dynamics SimulationProtein BindingAntitubercular AgentsBacterial ProteinsCytoskeletal ProteinsFtsZ protein, BacteriaFtsZ inhibitionMarine fungal metabolitesMM/GBSAMolecular dynamicsTuberculosis

Identifiers

PMID41501134
PMCPMC12855928

What Socratic holds

Textmetadata
LicenceCC BY-NC-ND
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.