Evidence mapPaperPMID 41801080Full record

ArticleCNS neuroscience & therapeutics2026

Elucidating Trigonelline's Therapeutic Mechanisms for Traumatic Brain Injury Through Integrated Network Pharmacology and In Vivo Validation.

Qian Zhang, Yuefan Zhang, Zhibing Song, Zixiang Tang, Guoqiang Wang, Xiang Yang, Jincai Li, Tiejun Li

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Article in CNS neuroscience & therapeutics, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 1 paper.

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1citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

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3 · Its place in the literature

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1 citing paper in PubMed.

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4 · The record

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5 · Who and what money

Authors and funding

8 authors.

Qian ZhangSchool of Traditional Chinese Medicine, Bozhou University, Bozhou, China.ORCID https://orcid.org/0009-0005-4232-9773
Yuefan ZhangSchool of Medicine, Shanghai University, Shanghai, China.
Zhibing SongSchool of Biological and Medical Engineering, Donghua University, Shanghai, China.
Zixiang TangSchool of Traditional Chinese Medicine, Bozhou University, Bozhou, China.
Guoqiang WangSchool of Traditional Chinese Medicine, Bozhou University, Bozhou, China.
Xiang YangZhangjiagang TCM Hospital, Affiliated to Nanjing University of Chinese Medicine, Suzhou, China.
Jincai LiSchool of Traditional Chinese Medicine, Bozhou University, Bozhou, China.ORCID https://orcid.org/0000-0002-0353-3617
Tiejun LiDepartment of Pharmacy, Punan Hospital, Shanghai, China.

Funding

Bozhou Municipal Key Laboratory of Modern Traditional Chinese Medicine Manufacturing 002006Key Specialty Construction Project of Pudong Health and Family Planning Commission of Shanghai PWZzk2022-08National Natural Science Foundation of China 82204929University Synergy Innovation Program of Anhui Province GXXT-2023-073
6 · The paper itself

Abstract

backgroundTraumatic brain injury (TBI) triggers complex pathological cascades, including inflammation, oxidative stress, apoptosis, and gliosis, particularly during the acute phase after injury. Trigonelline has been reported to exert neuroprotective effects in experimental models; however, its molecular mechanisms in acute TBI remain insufficiently defined.

objectiveThis study aimed to elucidate the molecular targets and mechanisms by which trigonelline attenuates acute TBI using an integrated network pharmacology and experimental validation approach.

methodsA trigonelline-target interaction network was constructed based on network pharmacology, followed by GO/KEGG analyses to predict the biological processes and pathways involved. Molecular docking was conducted to validate the binding affinity of trigonelline with key targets. Animal experiments were carried out to confirm the mechanistic predictions.

resultsNetwork pharmacology identified GAPDH, IL6, ALB, TNF, and IL1B as major hub genes associated with trigonelline. GO/KEGG analyses suggested that the neuroprotective effects of trigonelline against TBI primarily involved the MAPK and PI3K-Akt pathways. In vivo assays demonstrated that trigonelline treatment significantly reduced brain water content, inflammation, and oxidative stress levels within 72 h post-injury, while ameliorating histopathological damage, as confirmed by ELISA, HE, and LFB staining. TUNEL, NeuN, and FJB staining further revealed that trigonelline attenuated TBI-induced neuronal apoptosis. Western blotting demonstrated that trigonelline suppressed MMP-9 and AQP4 expression and attenuated the triggering of the MAPK signaling pathway.

conclusionBy attenuating MAPK signaling and apoptosis, trigonelline mitigates neural damage following TBI. The present findings provide experimental evidence supporting the neuroprotective effects of trigonelline in an acute TBI model.

Indexed as

AlkaloidsBrain Injuries, TraumaticNetwork PharmacologyNeuroprotective AgentsAnimalsMaleMolecular Docking SimulationOxidative StressRatsRats, Sprague-DawleyAlkaloidsNeuroprotective AgentstrigonellineMAPK pathwaymolecular dockingnetwork pharmacologytraumatic brain injurytrigonelline

Identifiers

PMID41801080
PMCPMC12970217

What Socratic holds

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.