Evidence mapPaperPMID 41803158Full record

ArticleScientific reports2026

Organic solution advanced spray-dried microparticulate dry powder of doxycycline hyclate for lung delivery.

Hanan Alameddin, Wafaa Alabsi, Basanth Babu Eedara, Neftali Ortega Alarcon, Richard L De Armond, Saif Mashaqi, Sairam Parthasarathy, Roberto Guzman, Heidi M Mansour

Abstract read
In one paragraph

Article in Scientific reports, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

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Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

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0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

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PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

9 authors.

Hanan AlameddinThe University of ArizonaR. Ken Coit College of PharmacySkaggs Pharmaceutical Sciences Center, Tucson, AZ, USA. hananalameddin@arizona.edu.
Wafaa AlabsiThe University of ArizonaR. Ken Coit College of PharmacySkaggs Pharmaceutical Sciences Center, Tucson, AZ, USA.
Basanth Babu EedaraThe University of ArizonaR. Ken Coit College of PharmacySkaggs Pharmaceutical Sciences Center, Tucson, AZ, USA.
Neftali Ortega AlarconThe University of ArizonaR. Ken Coit College of PharmacySkaggs Pharmaceutical Sciences Center, Tucson, AZ, USA.
Richard L De ArmondThe University of Arizona Health Sciences Center for Sleep Circadian and Neurosciences Research, Tucson, AZ, USA.
Saif MashaqiThe University of Arizona Health Sciences Center for Sleep Circadian and Neurosciences Research, Tucson, AZ, USA.
Sairam ParthasarathyThe University of Arizona Health Sciences Center for Sleep Circadian and Neurosciences Research, Tucson, AZ, USA.
Roberto GuzmanThe University of ArizonaR. Ken Coit College of PharmacySkaggs Pharmaceutical Sciences Center, Tucson, AZ, USA.
Heidi M MansourThe University of ArizonaR. Ken Coit College of PharmacySkaggs Pharmaceutical Sciences Center, Tucson, AZ, USA.

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Obstructive sleep apnea (OSA) is a common sleep disorder characterized by the upper airway collapse, leading to interrupted breathing and reduced oxygen levels during sleep. This condition often results in chronic inflammation and is associated with various long-term health problems. To address OSA-related inflammation, an FDA-approved drug, Doxycycline, was formulated in this study as a dry powder inhaler due to its favorable anti-inflammatory properties that was tested in subsequent cellular and animal studies of OSA. This comprehensive and systematic study aimed to develop inhalable excipient-free spray-dried (SD) one-component drug powders of Doxycycline. Advanced organic solution spray-drying in closed mode, with three different feed pump rates (10%, 50%, and 100%), was used to design and produce Doxycycline microparticles in the solid state successfully. The SD Doxycycline formulations comprised hollow, spherical, dimpled particles (<2 μm). The solid-state characterization of SD formulations confirmed the amorphous nature of Doxycycline after spray drying with a glass transition temperature between 82.73 °C and 89.29 °C. However, compared to the raw drug, residual water content was higher in the SD formulation, ranging from 6.4 ± 0.02% w/w in SD Doxycycline at the low feed pump rate to 6.79 ± 0.06% w/w in SD Doxycycline at the high feed pump rate. SD formulations showed good aerosolization behavior with a Respirable Fraction (RF) of >60% with NeoHaler inhaler device (63.19 ± 7.59 to 68.53 ± 3.73%) while HandiHaler showed lower RF (39.61± 0.57 to 53.90 ± 8.03%). The fine particle fraction (FPF) was higher in the NeoHaler group (24.91 ± 1.17 to 36.72 ± 2.01%) compared to HandiHaler (19.61 ± 5.41 to 33.76 ± 5.21%). This could be explained by the difference in median aerodynamic diameter (8.21 ± 2.68 to 4.69± 1.27 μm) in the NeoHaler group compared to (3.07 ± 0.36 to 3.67 ± 0.59 μm) HandiHaler group. Furthermore, in vitro cell viability as a function of lung cell type and drug dose showed 10 µM of Doxycycline as a safe concentration for the A549, H358, H441, and Calu-3 epithelial-like immortal human cell lines. Inhalable dry powder formulation of Doxycycline could offer new treatment options for patients suffering from sleep apnea.

Indexed as

DoxycyclineDrug Delivery SystemsLungAdministration, InhalationAerosolsAnimalsDry Powder InhalersHumansParticle SizePowdersSpray DryingAerosolsDoxycyclinePowdersAerosolizationDoxycyclineDry Powder Inhaler (DPI)Lung inflammationObstructive Sleep Apnea (OSA)Spray drying

Identifiers

PMID41803158
PMCPMC13096535

What Socratic holds

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.