Evidence mapPaperPMID 41810128Full record

Trial reportDrug design, development and therapy2026

Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of Intravenous Administration JMKX003142 in Chinese Healthy Subjects: A Randomized, Double-Blind, Placebo-Controlled, Single, and Multiple Ascending Dose Phase I Clinical Trial.

Cheng Cui, Jixiang Zhu, Zhiping Liu, Jingyao Liu, Xiaomin Huang, Yi Liu, Jingqiu Hu, Lingli Zhang, Xue Zhang, Yila Sha and 2 more

Registry-linked trialAbstract readRandomized Controlled TrialClinical Trial, Phase I
In one paragraph

Trial report in Drug design, development and therapy, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. It is linked to trial NCT06344533 (Phase I Clinical Study to Evaluate the Safety, Tolerability, and Pharmacokinetic Characteristics of JMKX003142 Injection Administered Randomly, Double-blind, Placebo-controlled, Single-ascending Dose and Multiple-ascending Doses in Chinese Healthy Adult Subjects), which is not on this map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

NCT06344533 phase1unknown statusnot on this map

Phase I Clinical Study to Evaluate the Safety, Tolerability, and Pharmacokinetic Characteristics of JMKX003142 Injection Administered Randomly, Double-blind, Placebo-controlled, Single-ascending Dose and Multiple-ascending Doses in Chinese Healthy Adult Subjects

TypeinterventionalSponsorJemincareRan2024 to 2025Enrolled78ConditionsHealthy AdultArmsJMKX003142 Injection, Placebo
3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

12 authors.

Cheng CuiDrug Clinical Trial Center, Department of Pharmacy, Peking University Third Hospital, Beijing, 100191, People's Republic of China.
Jixiang ZhuDrug Clinical Trial Center, Department of Pharmacy, Peking University Third Hospital, Beijing, 100191, People's Republic of China.
Zhiping LiuDrug Clinical Trial Center, Department of Pharmacy, Peking University Third Hospital, Beijing, 100191, People's Republic of China.
Jingyao LiuDrug Clinical Trial Center, Department of Pharmacy, Peking University Third Hospital, Beijing, 100191, People's Republic of China.
Xiaomin HuangDrug Clinical Trial Center, Department of Pharmacy, Peking University Third Hospital, Beijing, 100191, People's Republic of China.
Yi LiuClinical Development Center, Shanghai Jeyou Pharmaceutical Co.,Ltd., Shanghai, 200120, People's Republic of China.
Jingqiu HuClinical Development Center, Shanghai Jeyou Pharmaceutical Co.,Ltd., Shanghai, 200120, People's Republic of China.
Lingli ZhangClinical Development Center, Shanghai Jeyou Pharmaceutical Co.,Ltd., Shanghai, 200120, People's Republic of China.
Xue ZhangClinical Development Center, Shanghai Jeyou Pharmaceutical Co.,Ltd., Shanghai, 200120, People's Republic of China.
Yila ShaClinical Development Center, Shanghai Jeyou Pharmaceutical Co.,Ltd., Shanghai, 200120, People's Republic of China.
Dongyang LiuDrug Clinical Trial Center, Department of Pharmacy, Peking University Third Hospital, Beijing, 100191, People's Republic of China.ORCID 0000-0002-0608-8192
Haiyan LiDrug Clinical Trial Center, Department of Pharmacy, Peking University Third Hospital, Beijing, 100191, People's Republic of China.

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Purpose: This study is the first-in-human study to evaluate the safety, tolerability, pharmacokinetics (PK), and pharmacodynamics (PD) profiles of single ascending doses (SAD) and multiple ascending doses (MAD) of JMKX003142 injection in healthy Chinese subjects. Patients and Methods: In this Phase I, randomized, double-blind, placebo-controlled study, 48 subjects in the SAD (0.1-6 mg) study received intravenous injection of JMKX003142 or placebo in ascending dose. Thirty subjects in the MAD (1-4 mg) study received an intravenous injection of JMKX003142 or placebo once a day for five consecutive days. The primary endpoint was the safety and tolerability of JMKX003142 injection, with the secondary and exploratory endpoints focusing on its PK and PD profiles, respectively. Results: The JMKX003142 injection exhibited favourable safety and tolerability, with all treatment-emergent adverse events (TEAEs) being mild. No serious adverse events, deaths or discontinuations due to TEAEs were observed. Following single and multiple intravenous injections of JMKX003142, the maximum concentration (C Conclusion: Overall, both single and multiple intravenous injections of JMKX003142 have been demonstrated to be safe, well tolerated, and to possess excellent PK characteristics as well as significant diuretic activity. Trial Registration: This study was registered with ClinicalTrials.gov (NCT06344533).

Indexed as

Antidiuretic Hormone Receptor AntagonistsReceptors, VasopressinAdministration, IntravenousAdultChinaDose-Response Relationship, DrugDouble-Blind MethodEast Asian PeopleFemaleHealthy VolunteersHumansInjections, IntravenousMaleYoung AdultAntidiuretic Hormone Receptor AntagonistsAVPR2 protein, humanReceptors, Vasopressinactive arginine vasopressin V2 receptor antagonistJMKX003142pharmacodynamicspharmacokineticssafetytolerability

Identifiers

PMID41810128
PMCPMC12970034

What Socratic holds

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Registered trials

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.