Evidence map›Paper›PMID 41889258›Full record

ArticleInorganic chemistry2026

Dual-Action NSAID-Gold(I) Alkynyl Hybrids for Synergistic Anti-Inflammatory and Anticancer Therapy of Colorectal Cancer.

Javier Sáez, Luis Vicente Herrera-Marcos, María Jesús Rodríguez-Yoldi, M Concepción Gimeno, Elena Cerrada

Abstract read
In one paragraph

Article in Inorganic chemistry, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
–field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

5 authors.

Javier SáezDepartamento de Química Inorgánica, Instituto de Síntesis Química Y Catálisis Homogénea (ISQCH). Universidad de Zaragoza-C.S.I.C, Zaragoza 50009, Spain.
Luis Vicente Herrera-MarcosDepartamento de anatomía E Histología Humanas, Facultad de Ciencias de la Salud Y Del Deporte, Pl. Universidad 3, Huesca 22002, Spain.
María Jesús Rodríguez-YoldiDepartamento de farmacología Y Fisiología, Medicina Legal Y Forense. Unidad de Fisiología, Facultad de Veterinaria, Ciber de Fisiopatología de la Obesidad Y Nutrición (CIBERobn), Instituto Agroalimentario de Aragón (IA2), Zaragoza 50013, Spain.
M Concepción GimenoDepartamento de Química Inorgánica, Instituto de Síntesis Química Y Catálisis Homogénea (ISQCH). Universidad de Zaragoza-C.S.I.C, Zaragoza 50009, Spain.ORCID 0000-0003-0553-0695
Elena CerradaDepartamento de Química Inorgánica, Instituto de Síntesis Química Y Catálisis Homogénea (ISQCH). Universidad de Zaragoza-C.S.I.C, Zaragoza 50009, Spain.ORCID 0000-0003-2457-3674

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Colorectal cancer (CRC) remains a major global health challenge, in which chronic inflammation and redox dysregulation are key drivers of tumor progression. Here, we report a rationally designed family of NSAID-derived alkyne ligands coordinated to JohnPhos-gold(I) fragments, affording eight new alkynyl gold(I) derivatives. Complexes based on naproxen, ibuprofen, and salicylic acid derivatives display potent antiproliferative activity against Caco-2/TC7 colon cancer cells, outperforming oxaliplatin and being comparable to auranofin, while showing markedly reduced cytotoxicity in breast cancer lines and nonmalignant cells, thus indicating promising selectivity. Mechanistic studies revealed that the most active complex, [Au(L1)JP] (

Indexed as

AlkynesAnti-Inflammatory Agents, Non-SteroidalAntineoplastic AgentsColorectal NeoplasmsGoldApoptosisCell Line, TumorCell ProliferationCyclooxygenase 2Drug Screening Assays, AntitumorHumansMolecular StructureAlkynesAnti-Inflammatory Agents, Non-SteroidalAntineoplastic AgentsCyclooxygenase 2Gold

Identifiers

PMID41889258
PMCPMC13058884

What Socratic holds

Textmetadata
LicenceCC BY
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.