Evidence mapPaperPMID 41915115Full record

Trial reportAdvances in therapy2026

Safety, Tolerability and PK Characteristics of RM301B Eye Drops: A Single-Centre, Randomized, Double-Blind, Dose-Escalation, Placebo-Controlled Phase I Clinical Trial.

Zhishu Bao, Wendan Xu, Ruoyu Li, Haihui Wei, Qing Dong, Ziang Xu, Linlin Li, Chenglong Li, Huixiang Ma, Jia Qu and 2 more

Abstract readRandomized Controlled TrialClinical Trial, Phase I
PubMed Publisher
In one paragraph

Trial report in Advances in therapy, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

12 authors.

Zhishu Bao *National Engineering Research Center of Ophthalmology and Optometry, Eye Hospital, Wenzhou Medical University, Wenzhou, 325027, China.
Wendan Xu *National Engineering Research Center of Ophthalmology and Optometry, Eye Hospital, Wenzhou Medical University, Wenzhou, 325027, China.
Ruoyu Li *National Engineering Research Center of Ophthalmology and Optometry, Eye Hospital, Wenzhou Medical University, Wenzhou, 325027, China.
Haihui WeiNational Engineering Research Center of Ophthalmology and Optometry, Eye Hospital, Wenzhou Medical University, Wenzhou, 325027, China.
Qing DongChengdu Ruimu Biopharmaceuticals Co., Ltd., Chengdu, 611135, China.
Ziang XuNational Engineering Research Center of Ophthalmology and Optometry, Eye Hospital, Wenzhou Medical University, Wenzhou, 325027, China.
Linlin LiNational Engineering Research Center of Ophthalmology and Optometry, Eye Hospital, Wenzhou Medical University, Wenzhou, 325027, China.
Chenglong LiNational Engineering Research Center of Ophthalmology and Optometry, Eye Hospital, Wenzhou Medical University, Wenzhou, 325027, China.
Huixiang MaNational Engineering Research Center of Ophthalmology and Optometry, Eye Hospital, Wenzhou Medical University, Wenzhou, 325027, China. mahuixiang2022@163.com.
Jia QuNational Engineering Research Center of Ophthalmology and Optometry, Eye Hospital, Wenzhou Medical University, Wenzhou, 325027, China. qujia@eye.ac.cn.
Liangde XuNational Engineering Research Center of Ophthalmology and Optometry, Eye Hospital, Wenzhou Medical University, Wenzhou, 325027, China. xuld@eye.ac.cn.
Hong WangNational Engineering Research Center of Ophthalmology and Optometry, Eye Hospital, Wenzhou Medical University, Wenzhou, 325027, China. wanghongbio@wmu.edu.cn.ORCID http://orcid.org/0000-0001-8391-3806

Funding

Key Research and Development Program of Zhejiang Province 2023C03031National Key Research and Development Program for Active Health and Aging Response 2023YFC3604000National Natural Science Foundation of China 32370679National Natural Science Foundation of China 92581118
6 · The paper itself

Abstract

introductionRM301B eye drops are a dexamethasone (DEX)-based formulation indicated for treating macular oedema associated with retinal vein occlusion (RVO). Non-clinical pharmacodynamic studies have demonstrated that RM301B eye drops have a certain inhibitory effect on retinal oedema. This study aimed to evaluate the safety, tolerability, and pharmacokinetic (PK) characteristics of RM301B eye drops following administration in healthy subjects.

methodsA single-centre, randomized, double-blind, placebo-controlled, dose-escalation Phase I clinical study. In the single-dose study, ten subjects received once-daily RM301B or placebo. In the multiple ascending dose study, 30 subjects received 3, 6, or 8 daily instillations for 7 days. Safety and tolerability were monitored throughout the study, with plasma samples collected for PK analysis.

resultsNo serious adverse events (SAEs) occurred in the study. All mild adverse events (AEs) were determined to be unrelated to RM301B. PK results indicated detectable plasma concentrations (0.10-0.40 ng/ml) only in individual subjects within 5 h post-single dose and at specific time points following multiple dosing. Mean area under the curve from time zero to t (AUC

conclusionsRM301B eye drops demonstrated safety and good tolerability in subjects, characterized by minimal plasma exposure, a short half-life, and no significant accumulation. Subsequent trials will evaluate the safety and efficacy of RM301B in patients with macular oedema associated with RVO.

trial registrationChiCTR2500111837 (retrospectively registered on November 6, 2025).

Indexed as

DexamethasoneMacular EdemaOphthalmic SolutionsAdultArea Under CurveDose-Response Relationship, DrugDouble-Blind MethodFemaleHumansMaleMiddle AgedYoung AdultDexamethasoneOphthalmic SolutionsDexamethasonePharmacokineticsPhase I clinical trialRM301B eye drops

Identifiers

What Socratic holds

Textmetadata
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.