Evidence mapPaperPMID 41994902Full record

Trial reportDiabetes, obesity & metabolism2026

Pharmacokinetic Bioequivalence of Orforglipron Tablets and Capsules in Healthy Participants With Obesity or Overweight.

Xiaosu Ma, Ying Grace Li, Sohini Raha, David C Sperry, David E Coutant, Shobha Bhattachar

Registry-linked trialAbstract readClinical Trial, Phase IMulticenter StudyRandomized Controlled Trial
In one paragraph

Trial report in Diabetes, obesity & metabolism, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. It is linked to trial NCT06440980 (A Multiple-Dose Study to Investigate the Bioequivalence of Orforglipron), which is not on this map. Cited by 7 papers.

0numbers the graph read from it
0cells of the map it votes in
7citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

NCT06440980 phase1completednot on this map

A Multiple-Dose Study to Investigate the Bioequivalence of Orforglipron (LY3502970) Capsules and Orforglipron Tablets in Participants With Obesity or Overweight Who Are Otherwise Healthy.

TypeinterventionalSponsorEli Lilly and CompanyRan2024 to 2025Enrolled533ConditionsHealthy, Obese, Overweight, ObesityArmsOrforglipron
3 · Its place in the literature

Who cites it

7 citing papers in PubMed.

  1. Trial
  2. Trial
  3. Article
  4. Article
  5. Article
  6. Article
  7. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

6 authors.

Xiaosu MaEli Lilly and Company, Indianapolis, Indiana, USA.
Ying Grace LiEli Lilly and Company, Indianapolis, Indiana, USA.
Sohini RahaEli Lilly and Company, Indianapolis, Indiana, USA.
David C SperryEli Lilly and Company, Indianapolis, Indiana, USA.
David E CoutantEli Lilly and Company, Indianapolis, Indiana, USA.
Shobha BhattacharEli Lilly and Company, Indianapolis, Indiana, USA.

Funding

Eli Lilly and Company
6 · The paper itself

Abstract

aimsTo evaluate the bioequivalence of orally administered orforglipron tablets and capsules in participants with obesity or overweight who were otherwise healthy. MATERIALS AND

methodsThis phase 1, multicenter, open-label, multiple-dose, dose-escalation study was conducted in 429 healthy adults. Study participants received each orforglipron capsule and tablet dose strength once daily for 7 days in the fasted state at capsule doses of 1, 3, 6, 12, 24, or 36 mg and corresponding tablet doses of 0.8, 2.5, 5.5, 9, 14.5, and 17.2 mg. The primary endpoint was steady-state area under the concentration-time curve from 0 to 24 h (AUC

resultsBioequivalence was demonstrated between capsules and dose-adjusted tablets across all six doses. The 90% confidence interval of the ratios of the geometric least-squares means of AUC

conclusionsOnce-daily orforglipron capsules and dose-adjusted tablets demonstrated pharmacokinetic bioequivalence at all tested doses and showed similar safety and tolerability profiles, with mostly mild treatment-emergent adverse events consistent with previous orforglipron clinical trials. ClinicalTrials .gov Identifier: NCT06440980.

Indexed as

Anti-Obesity AgentsObesityOverweightAdministration, OralAdolescentAdultArea Under CurveCapsulesDose-Response Relationship, DrugFemaleFluorine CompoundsHumansMaleMiddle AgedOxadiazolesTabletsAnti-Obesity AgentsCapsulesFluorine CompoundsorforglipronOxadiazolesTabletsantiobesity drugGLP‐1obesity therapypharmacokinetics

Identifiers

PMID41994902
PMCPMC13243956

What Socratic holds

Textmetadata
LicenceCC BY-NC
Read underepoch 390

Registered trials

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.