Evidence mapPaperPMID 42007495Full record

ArticleCPT: pharmacometrics & systems pharmacology2026

Population Pharmacokinetics and Pharmacokinetics-Pharmacodynamics Analyses of Elafibranor to Support Dose Selection in Primary Biliary Cholangitis.

Qing Xi Ooi, Karl Brendel, Stijn van Beek, Jurij Aguiar Zdovc, Maddlie Bardol, Marion Dehez

Abstract read
In one paragraph

Article in CPT: pharmacometrics & systems pharmacology, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

6 authors.

Qing Xi OoiPharmetheus, Uppsala, Sweden.ORCID https://orcid.org/0000-0003-4310-9842
Karl BrendelIpsen, Paris, France.ORCID https://orcid.org/0009-0004-7551-0758
Stijn van BeekPharmetheus, Uppsala, Sweden.
Jurij Aguiar ZdovcPharmetheus, Uppsala, Sweden.ORCID https://orcid.org/0000-0001-8680-3792
Maddlie BardolPharmetheus, Uppsala, Sweden.
Marion DehezIpsen, Paris, France.

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Elafibranor 80 mg/day is approved for second-line primary biliary cholangitis (PBC) treatment. We present pharmacokinetic (PK) analyses of elafibranor and its metabolite, GFT1007, and pharmacokinetic-pharmacodynamic (PKPD) analyses describing the relationship between their exposure and responses in alkaline phosphatase (ALP) and total bilirubin (TB). PK data originated from 17 clinical trials. Separate elafibranor and GFT1007 PK models were developed using nonlinear mixed-effects modeling. Effects of covariates on PK parameters were explored. PKPD data originated from one phase II and one phase III trial; separate ALP and TB models were developed using a sequential approach. The sum of the areas under the plasma-concentration time curve during a dosing interval at steady state of elafibranor and GFT1007 (AUC

Indexed as

Liver Cirrhosis, BiliaryModels, BiologicalAlkaline PhosphataseArea Under CurveBilirubinDose-Response Relationship, DrugFemaleHumansMaleAlkaline PhosphataseBilirubindoseefficacylivermodel based drug developmentpopulation pharmacodynamicspopulation pharmacokineticssimulation

Identifiers

PMID42007495
PMCPMC13274737

What Socratic holds

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LicenceCC BY-NC
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Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.