Evidence map›Paper›PMID 42028604›Full record

Trial reportCirculation. Heart failure2026

Modest Contribution of Bradykinin to Blood Pressure Reduction by Sacubitril/Valsartan in Chronic Heart Failure.

Deepak K Gupta, Lynne W Stevenson, Erica M Garner, Christopher Maulion, Hui Nian, Patricia R Wright, Adina F Turcu, Shouzou Wei, Nancy J Brown

Registry-linked trialAbstract readRandomized Controlled Trial
In one paragraph

Trial report in Circulation. Heart failure, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. It is linked to trial NCT04113109 (Mechanisms Underlying Hypotensive Response to ARB/NEP Inhibition - Aim 2), which is not on this map. Cited by 1 paper.

0numbers the graph read from it
0cells of the map it votes in
1citing papers in PubMed
–field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

NCT04113109 phase4completednot on this map

Mechanisms Underlying Hypotensive Response to ARB/NEP Inhibition - Aim 2

TypeinterventionalSponsorVanderbilt University Medical CenterRan2019 to 2025Enrolled46ConditionsHeart FailureArmsLCZ 696, Icatibant, placebo, Para-aminohippurate, Iohexol
3 · Its place in the literature

Who cites it

1 citing paper in PubMed.

  1. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

9 authors.

Deepak K GuptaVanderbilt Translational and Clinical Cardiovascular Research Center and Division of Cardiovascular Medicine (D.K.G., L.W.S.), Vanderbilt University Medical Center, Nashville, TN.ORCID 0000-0003-2191-3485
Lynne W StevensonVanderbilt Translational and Clinical Cardiovascular Research Center and Division of Cardiovascular Medicine (D.K.G., L.W.S.), Vanderbilt University Medical Center, Nashville, TN.ORCID 0000-0002-8626-5258
Erica M GarnerDivision of Endocrinology, Diabetes, and Metabolism (E.M.G.), Vanderbilt University Medical Center, Nashville, TN.ORCID 0000-0001-8703-2678
Christopher MaulionDivision of Cardiovascular Medicine, Yale University School of Medicine, New Haven, CT (C.M.).ORCID 0000-0002-2510-4266
Hui NianDepartment of Biostatistics (H.N.), Vanderbilt University Medical Center, Nashville, TN.ORCID 0000-0003-0047-8330
Patricia R WrightDivision of Clinical Pharmacology (P.R.W., S.W.), Vanderbilt University Medical Center, Nashville, TN.
Adina F TurcuDivision of Metabolism, Endocrinology, and Diabetes, University of Michigan School of Medicine, Ann Arbor (A.F.T.).ORCID 0000-0001-9831-6190
Shouzou WeiDivision of Clinical Pharmacology (P.R.W., S.W.), Vanderbilt University Medical Center, Nashville, TN.
Nancy J BrownYale University School of Medicine, New Haven, CT (N.J.B.).ORCID 0000-0001-7109-3142

Funding

Vanderbilt Institute for Clinical and Translational Research (VICTR) -Identifying correlates of functional immunity in SARS-CoV-2 convalescent plasmaUL1TR002243 · NCATS · VANDERBILT UNIVERSITY MEDICAL CENTER · PI Paul A. Harris, Wesley H Self · 2017 to 2026
$130.7M
Improving Diagnostic Accuracy for Acute Heart FailureR01HL153607 · NHLBI · VANDERBILT UNIVERSITY MEDICAL CENTER · PI COLLINS, SEAN PATRICK, GUPTA, DEEPAK · 2021 to 2024
$5.9M
Mechanism(s) Underlying Hypotensive Response to ARB/NEP InhibitionR01HL145293 · NHLBI · YALE UNIVERSITY · PI BROWN, NANCY J., STEVENSON, LYNNE W · 2020 to 2024
$3.1M
NCATS NIH HHS UL1 TR002243NHLBI NIH HHS R01 HL145293NHLBI NIH HHS R01 HL153607
6 · The paper itself

Abstract

backgroundSymptomatic hypotension can limit sacubitril/valsartan therapy. Neprilysin inhibition may augment vasodilators, such as bradykinin. We hypothesized that bradykinin contributes to blood pressure (BP) lowering with sacubitril/valsartan in stable ambulatory patients with heart failure and reduced ejection fraction <50%.

methodsIn a randomized, double-blind crossover trial, participants received intravenous infusion of the bradykinin B2 receptor inhibitor icatibant and a matching placebo for 6 hours following sacubitril/valsartan dosing at acute initiation (n=36) and after 8 weeks of chronic therapy (n=30). The primary end point was maximal change in mean arterial pressure (MAP). Plasma natriuretic peptides, urine cyclic GMP, urine volume, sodium excretion, renal plasma flow, and renovascular resistance were measured.

resultsThe first dose of sacubitril/valsartan (50 mg) significantly lowered MAP by a mean maximum of ≈10 mm Hg, which was similar during icatibant and placebo. Within 6 hours after the first sacubitril/valsartan dose, plasma ANP (atrial natriuretic peptide [1-28]) and urine cGMP/creatinine increased significantly, whereas B-type NP (1-32) and NT-proBNP (N-terminal pro B-type natriuretic peptide) did not. Icatibant partially blunted the rise in urine cGMP/creatinine, but did not affect other parameters. After 8 weeks of sacubitril/valsartan titrated to maximally tolerated doses, baseline ANP (1-28) remained increased, and baseline MAP and NT-proBNP were decreased compared with before sacubitril/valsartan initiation. MAP decreased further after dose administration of sacubitril/valsartan, and the mean maximal reduction in MAP was significantly attenuated during icatibant compared with placebo (9 versus 12 mm Hg;

conclusionsBP lowering with sacubitril/valsartan occurs with both acute and chronic dosing. ANP (1-28) appears to mediate the initial BP reduction, whereas bradykinin contributes to BP lowering after dosing during chronic therapy. Clarifying these mechanisms may inform clinical management to optimize the benefit of this important heart failure and reduced ejection fraction therapy. REGISTRATION: URL: https://www.clinicaltrials.gov; Unique identifier: NCT04113109.

Indexed as

AminobutyratesAngiotensin Receptor AntagonistsBlood PressureBradykininBradykinin B2 Receptor AntagonistsHeart FailureTetrazolesAgedBiphenyl CompoundsChronic DiseaseCross-Over StudiesCyclic GMPDouble-Blind MethodDrug CombinationsFemaleHumansAminobutyratesAngiotensin Receptor AntagonistsBiphenyl CompoundsBradykininBradykinin B2 Receptor AntagonistsCyclic GMPDrug CombinationsicatibantNatriuretic Peptide, BrainPeptide Fragmentssacubitril and valsartan sodium hydrate drug combinationTetrazolesValsartanblood pressurebradykininheart failurehypotensionneprilysin

Identifiers

PMID42028604
PMCPMC13171156

What Socratic holds

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Read underepoch 390

Registered trials

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.