Evidence mapPaperPMID 42226756Full record

ArticleDrug design, development and therapy2026

Pharmacokinetics and Pharmacodynamics of Dapagliflozin in Obese and Nonobese Healthy Adults Following Multiple Administration.

Hae Won Lee, Hyungjin Kim, Ji Seo Park, Jae Hwa Lee, Jin Ju Park, Mi-Ri Gwon, Joo-Youn Cho, Sook Jin Seong, Young-Ran Yoon

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Article in Drug design, development and therapy, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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1 · What the graph read from it

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Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

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3 · Its place in the literature

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4 · The record

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5 · Who and what money

Authors and funding

9 authors.

Hae Won LeeSchool of Medicine, Kyungpook National University and Department of Clinical Pharmacology and Therapeutics, Kyungpook National University Hospital, Daegu, 41944, Republic of Korea.ORCID 0000-0001-7299-5332
Hyungjin KimSchool of Medicine, Kyungpook National University and Department of Clinical Pharmacology and Therapeutics, Kyungpook National University Hospital, Daegu, 41944, Republic of Korea.ORCID 0009-0004-1487-1293
Ji Seo ParkSchool of Medicine, Kyungpook National University and Department of Clinical Pharmacology and Therapeutics, Kyungpook National University Hospital, Daegu, 41944, Republic of Korea.
Jae Hwa LeeSchool of Medicine, Kyungpook National University and Department of Clinical Pharmacology and Therapeutics, Kyungpook National University Hospital, Daegu, 41944, Republic of Korea.ORCID 0000-0002-1886-7038
Jin Ju ParkSchool of Medicine, Kyungpook National University and Department of Clinical Pharmacology and Therapeutics, Kyungpook National University Hospital, Daegu, 41944, Republic of Korea.
Mi-Ri GwonSchool of Medicine, Kyungpook National University and Department of Clinical Pharmacology and Therapeutics, Kyungpook National University Hospital, Daegu, 41944, Republic of Korea.
Joo-Youn ChoDepartment of Clinical Pharmacology and Therapeutics, Seoul National University College of Medicine and Hospital, Seoul, Republic of Korea.ORCID 0000-0001-9270-8273
Sook Jin SeongSchool of Medicine, Kyungpook National University and Department of Clinical Pharmacology and Therapeutics, Kyungpook National University Hospital, Daegu, 41944, Republic of Korea.
Young-Ran YoonSchool of Medicine, Kyungpook National University and Department of Clinical Pharmacology and Therapeutics, Kyungpook National University Hospital, Daegu, 41944, Republic of Korea.ORCID 0000-0003-2166-7579

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Background: Dapagliflozin, a sodium-glucose cotransporter 2 inhibitor, lowers blood glucose levels by preventing renal glucose reabsorption, resulting in urinary glucose excretion. Because dapagliflozin-induced glycosuria produces a modest reduction in body weight, it may benefit patients with type 2 diabetes who are overweight or obese. Pathophysiologic alterations associated with obesity may lead to clinically significant differences in drug pharmacokinetic (PK) and pharmacodynamic (PD) properties. Purpose: This study aimed to evaluate the PK and PD characteristics of dapagliflozin in obese and nonobese healthy adults and assess the effect of obesity on these profiles by comparing outcomes between the two groups following multiple oral doses. Methods: In this open-label, multiple-dose study, dapagliflozin 10 mg tablets were administered once daily for 5 days to healthy adults. Serial blood samples for PK analysis were collected before and up to 48 h after the last dose on day 5. PK parameters were determined using noncompartmental analysis.Sensitivity analyses were conducted, including correlation analysis of PK parameters with weight or BMI using Pearson's correlation coefficients ( Results: Thirteen nonobese and nine obese participants completed the study. The geometric mean ratio (obese/nonobese) (90% CIs) of the area under the plasma concentration-time curve during a dosing interval at steady state (AUC Conclusion: The AUC

Indexed as

Benzhydryl CompoundsGlucosidesHypoglycemic AgentsObesitySodium-Glucose Transporter 2 InhibitorsAdministration, OralAdultBlood GlucoseDose-Response Relationship, DrugFemaleHealthy VolunteersHumansMaleMiddle AgedTabletsYoung AdultBenzhydryl CompoundsBlood GlucosedapagliflozinGlucosidesHypoglycemic AgentsSodium-Glucose Transporter 2 InhibitorsTabletsdapagliflozinobesitypharmacodynamicspharmacokineticstype 2 diabetes

Identifiers

PMID42226756
PMCPMC13222617

What Socratic holds

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.