Evidence map›Paper›PMID 42310164›Full record

ArticlePsychopharmacology2026

Novel dopamine 4 receptor ligands differentially ameliorate ADHD-like behaviors in spontaneously hypertensive rats.

Ike C de la Peña, Samantha Andino, Ashley Amis, Mohammad A Alkhatib, Tian Li, Thomas M Keck, Comfort A Boateng

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Article in Psychopharmacology, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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0citing papers in PubMed
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1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

5 · Who and what money

Authors and funding

7 authors.

Ike C de la PeñaDepartment of Pharmaceutical and Administrative Sciences, Loma Linda University School of Pharmacy, Loma Linda, CA, 92350, USA. idelapena@llu.edu.ORCID http://orcid.org/0000-0003-2046-522X
Samantha AndinoDepartment of Pharmaceutical and Administrative Sciences, Loma Linda University School of Pharmacy, Loma Linda, CA, 92350, USA.
Ashley AmisDepartment of Pharmaceutical and Administrative Sciences, Loma Linda University School of Pharmacy, Loma Linda, CA, 92350, USA.
Mohammad A AlkhatibDepartment of Chemistry and Biochemistry, Department of Biological and Biomedical Sciences, College of Science and Mathematics, Rowan University, Glassboro, NJ, USA.
Tian LiDepartment of Basic Pharmaceutical Sciences, High Point University Fred Wilson School of Pharmacy, High Point, NC, USA.
Thomas M KeckDepartment of Chemistry and Biochemistry, Department of Biological and Biomedical Sciences, College of Science and Mathematics, Rowan University, Glassboro, NJ, USA. keckt@rowan.edu.ORCID http://orcid.org/0000-0003-1845-9373
Comfort A BoatengDepartment of Basic Pharmaceutical Sciences, High Point University Fred Wilson School of Pharmacy, High Point, NC, USA. cboateng@highpoint.edu.ORCID http://orcid.org/0000-0003-1907-431X

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

rationaleDopamine D4 receptors (D4Rs) have been implicated in the pathophysiology of attention-deficit/hyperactivity disorder (ADHD), yet their precise role and therapeutic relevance remain underexplored. Highly selective D4R compounds may provide a valuable tool to elucidate D4R function and assess their potential as non-stimulant ADHD treatments.

objectivesThis study examined the behavioral effects of two novel D4R drugs, namely, FMJ-01-38 (high-efficacy partial agonist) and FMJ-01-54 (full antagonist) in adolescent spontaneously hypertensive rats (SHR/NCrl), a validated ADHD animal model, and Wistar (control) rats.

methodsRats received intraperitoneal injections of FMJ-01-38 or FMJ-01-54 (5-10 mg/kg), or vehicle prior to behavioral assays assessing locomotor activity (open field tests), recognition memory (novel object preference test), spatial working memory (Y-maze test), and impulsivity (delay discounting task).

resultsFMJ-01-38 dose-dependently reduced locomotor hyperactivity and improved spontaneous alternation in SHR/NCrl; at 5 mg/kg, it also enhanced novel object preference and reduced impulsive choice and action, indicating attenuation of ADHD-like behaviors and improved cognitive function. FMJ-01-54 produced similar improvements in Y-maze and novel-object performance without altering locomotor activity or impulsivity of SHR/NCrl, suggesting selective cognitive improvement. In Wistar rats, FMJ-01-38 increased novel object preference only at the 5 mg/kg dose, while FMJ-01-54 treatment did not produce any significant behavioral effects.

conclusionsThese findings demonstrate that D4R modulation, through either partial agonism or antagonism, differentially ameliorates ADHD-related behaviors and improves cognitive performance. Both FMJ-01-38 and FMJ-01-54 produced minimal effects in control animals, suggesting pathology-specific efficacy and highlighting D4R ligands as promising non-stimulant therapeutic candidates for ADHD.

Indexed as

ADHDD4R full antagonistD4R partial agonistDopamine D4 receptorFMJ-01-38FMJ-01-54

Identifiers

PMID42310164

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.