Evidence mapPaperPMID 42310888Full record

ArticleDiabetes, obesity & metabolism2026

Effect of a Novel GLP-1 Analogue Ecnoglutide on the Pharmacokinetics of Rosuvastatin and Digoxin in Healthy Participants.

Fengshan Li, Chunfeng Du, Qin Yu, Shiyin Feng, Linrui Cai, Zhuo Chen, Qin Zou, Weiyi Guo, Dan Du, Feng Hu and 10 more

Abstract readClinical Trial, Phase I
In one paragraph

Article in Diabetes, obesity & metabolism, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Cited by 1 paper.

0numbers the graph read from it
0cells of the map it votes in
1citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

1 citing paper in PubMed.

  1. Article
4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

20 authors.

Fengshan LiNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.ORCID https://orcid.org/0000-0003-1115-2766
Chunfeng DuNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Qin YuNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Shiyin FengNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Linrui CaiNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Zhuo ChenNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Qin ZouNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Weiyi GuoNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Dan DuNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Feng HuNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Xiaohong LiuNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Yalin HuangNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Shuxia ShiNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Wei ShiNational Drug Clinical Trial Institution of West China Second University Hospital, Sichuan University, Chengdu, China.
Lei GuanHangzhou Sciwind Biosciences Co., Ltd., Hangzhou, China.
Liu YangHangzhou Sciwind Biosciences Co., Ltd., Hangzhou, China.
Qing ZhengHangzhou Sciwind Biosciences Co., Ltd., Hangzhou, China.
Yao LiHangzhou Sciwind Biosciences Co., Ltd., Hangzhou, China.
Rui LiuHangzhou Sciwind Biosciences Co., Ltd., Hangzhou, China.
Ming YangHangzhou Sciwind Biosciences Co., Ltd., Hangzhou, China.

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

aimEvaluate ecnoglutide (XW003) effects on rosuvastatin and digoxin pharmacokinetics (PKs) in healthy adults.

methodsThis was an open-label, single-sequence crossover Phase 1 study. Eligible participants received rosuvastatin (10 mg, single dose) and digoxin (0.25 mg, single dose) in two periods: Once before subcutaneous treatment with ecnoglutide and once during steady-state subcutaneous ecnoglutide (1.2 mg). Coadministration effect was assessed via PK parameters of both drugs.

resultsA total of 28 volunteers received at least one dose of study drug. Co-administration of ecnoglutide did not affect rosuvastatin and digoxin to a clinically relevant degree. For the area under the concentration-time curve from time zero to infinity, the geometric mean (GM) ratio (with ecnoglutide vs. alone) [90% confidence interval (CI)] was 106% (94%, 120%) for rosuvastatin and 84% (76%, 94%) for digoxin. Additionally, the maximum plasma concentration (C

conclusionBased on the PK and safety evaluations, ecnoglutide does not cause clinically significant PK interactions with rosuvastatin or digoxin. Consequently, no dose adjustments for rosuvastatin or digoxin are required when ecnoglutide is co-administered. However, close clinical and plasma monitoring is advised during the coadministration of digoxin, especially in patients with renal impairment.

Indexed as

DigoxinGlucagon-Like Peptide 1Hydroxymethylglutaryl-CoA Reductase InhibitorsRosuvastatin CalciumAdultCross-Over StudiesDrug InteractionsFemaleHealthy VolunteersHumansMaleMiddle AgedYoung AdultDigoxinGlucagon-Like Peptide 1Hydroxymethylglutaryl-CoA Reductase InhibitorsRosuvastatin Calciumdrug–drug interactionecnoglutide (XW003)glucagon‐like peptide‐1 analogueobesity

Identifiers

PMID42310888
PMCPMC13449077

What Socratic holds

Textmetadata
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Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.