Evidence map›Paper›PMID 42315993›Full record

ArticleChemMedChem2026

Synthesis of Novel d-Glucopyranuronamide-Based Nucleos(t)ide Analogs Bearing (Triazolyl)methyl Phosph(on)ate Motifs With Anticancer and Antibacterial Potential.

Domingos M Manuel, Tânia Moreira, Sérgio R Filipe, Veronika Vojáčková, Radek Jorda, Nuno M Xavier

Abstract read
In one paragraph

Article in ChemMedChem, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
–field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

6 authors.

Domingos M ManuelResearch Institute for Medicines (iMed.ULisboa), Faculty of Pharmacy, Universidade de Lisboa, Lisboa, Portugal.
Tânia MoreiraCentro de Química Estrutural, Institute of Molecular Sciences, Faculdade de Ciências, Universidade de Lisboa, Lisboa, Portugal.
Sérgio R FilipeLaboratory of Bacterial Cell Surfaces and Pathogenesis, UCIBIO-Applied Molecular Biosciences Unit - Associate Laboratory i4HB - Institute for Health and Bioeconomy, Dep. de Ciências da Vida, Faculdade de Ciências e Tecnologia, Universidade Nova de Lisboa, Caparica, 2825-149 Caparica, Portugal.
Veronika VojáčkováDepartment of Experimental Biology, Faculty of Science, Palacký University Olomouc, Olomouc, Czech Republic.
Radek JordaDepartment of Experimental Biology, Faculty of Science, Palacký University Olomouc, Olomouc, Czech Republic.
Nuno M XavierResearch Institute for Medicines (iMed.ULisboa), Faculty of Pharmacy, Universidade de Lisboa, Lisboa, Portugal.ORCID 0000-0001-8739-8768

Funding

Fundação para a Ciência e a Tecnologia CEECIND/03881/2018Fundação para a Ciência e a Tecnologia EXPL/MED-QUI/1017/2021Fundação para a Ciência e a Tecnologia LA/P/0056/2020Fundação para a Ciência e a Tecnologia UID/04138/2025Fundação para a Ciência e a Tecnologia UIDB/00100/2020Fundação para a Ciência e a Tecnologia UIDP/00100/2020Fundação para a Ciência e a Tecnologia UID/PRR/04138/2025Fundação para a Ciência e a Tecnologia UID/PRR2/04138/2025
6 · The paper itself

Abstract

The synthesis and evaluation of the antiproliferative and antibacterial potential of novel d-glucuronamide-based nucleoside analogs and isonucleotides is reported. The synthesized molecules comprise an anomeric (triazolyl)methyl phosphonate or phosphate motif and a dodecyl chain or a (triazolyl)ethyl purine system at the amide moiety. Their synthesis involved a 1,3-dipolar cycloaddition between N-propargyl or N-dodecyl glucuronamidyl azides with propargyl alcohol or propargyl bromide and further O-phosphorylation or Arbuzov reaction, respectively, to furnish glucuronamidyl (triazolyl)methyl phosphate/phosphonate derivatives. N-Propargyl glucuronamidyl derivatives were then engaged in cycloaddition with 9-azidoethyl-6-chloropurine to afford 6-chloropurine isonucleotides. Isonucleoside (triazolyl)methyl phosphonate/phosphates containing a 3-O-dodecyl moiety displayed significant antiproliferative activities in chronic myeloid leukemia (K562) and breast cancer (MCF-7) cells with GI

Indexed as

Anti-Bacterial AgentsAntineoplastic AgentsTriazolesCell ProliferationDose-Response Relationship, DrugDrug Screening Assays, AntitumorEscherichia coliHumansMCF-7 CellsMicrobial Sensitivity TestsMolecular StructureNucleosidesStructure-Activity RelationshipAnti-Bacterial AgentsAntineoplastic AgentsNucleosidesTriazolesantibacterial agentsanticancer agentscycloadditiond‐glucuronamidenucleoside and nucleotide analogs

Identifiers

PMID42315993
PMCPMC13279754

What Socratic holds

Textmetadata
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.